Bone Density Conservation Agents

Name
Bone Density Conservation Agents
Accession Number
DBCAT000089
Description

Agents that inhibit BONE RESORPTION and/or favor BONE MINERALIZATION and BONE REGENERATION. They are used to heal BONE FRACTURES and to treat METABOLIC BONE DISEASES such as OSTEOPOROSIS.

Drugs
DrugDrug Description
24,25-DihydroxycholecalciferolNot Annotated
AbaloparatideA parathyroid hormone-related protein (PTHrP) analog used for the treatment of osteoporosis in patients with a high risk of fracture.
Alendronic acidA bisphosphonate drug that prevents osteoclastic bone resorption which is used for the prevention and treatment of osteoporosis.
AlfacalcidolA vitamin D analogue used for the management of hypocalcemia, secondary hyperparathyroidism, and osteodystrophy in patients with chronic renal failure, as well as some types of rickets and osteomalacia.
BazedoxifeneA selective estrogen receptor modulator (SERM) used to treat moderate to severe vasomotor symptoms in menopause and osteoporosis alone or in combination with conjugated estrogens.
CalcifediolAn active metabolite of vitamin D used to treat hyperparathyroidism as well as to combat hypocalcemia in dialysis patients.
Calcitonin porcineCalcitonin is a polypeptide hormone secreted by the parafollicular cells of the thyroid gland in mammals. It inhibits bone resorption and lowers both serum and urinary calcium concentrations. Human calcitonin...
CalcitriolAn active metabolite of vitamin D that is used to treat hyperparathyroidism and is also used in dialysis patients to combat hypocalcemia.
CholecalciferolA form of Vitamin D used in the treatment of specific medical conditions such as refractory rickets, hypoparathyroidism, and familial hypophosphatemia, as well as osteoporosis and chronic kidney disease.
Clodronic acidA bisphosphonate used to treat osteoporosis in postmenopausal women, hypercalcemia of malignancy, and osteolysis.
DenosumabA RANK ligand (RANKL) inhibitor used for the management of osteoporosis in patients at high risk for bone fractures.
DihydrotachysterolA synthetic analog of vitamin D that does not require renal activation like vitamin D2 or Vitamin D3.
DoxercalciferolA synthetic vitamin D2 analog used to treat secondary hyperparathyroidism in patients with chronic kidney disease with or without therapy of dialysis.
ElcatoninNot Annotated
EldecalcitolInvestigated for use/treatment in osteoporosis.
ErgocalciferolA vitamin found in many supplement products.
Etidronic acidA bisphosphonate drug that prevents osteoclastic bone resorption; used for the prevention and treatment of osteoporosis.
Human calcitoninHuman calcitonin is indicated for the treatment of Paget's disease in the cases where the use of salmon calcitonin may provoke the generation of high-titer of antibodies. Paget's disease is...
IbandronateA bisphosphonate used to treat osteoporosis in postmenopausal women.
Incadronic acidIncadronate has been investigated in the treatment of myeloma, leukemia, and other cancers. It has also been investigated in patients with hypercalcemia of malignancy.
Nandrolone decanoateAn anabolic steroid indicated for the management of the anemia of renal insufficiency by increasing hemoglobin and red cell mass.
Olpadronic acidOlpadronic acid is a small molecule drug. Olpadronic acid has a monoisotopic molecular weight of 263.03 Da.
Pamidronic acidA bisphosphonate used to treat Paget's disease, to treat hypercalcemia of malignancy, and to treat osteolytic bone lesions.
ParicalcitolA vitamin D analog used to treat hyperparathyroidism associated with stage 3 or greater chronic kidney disease.
ProcalcitoninProcalcitonin is under investigation in clinical trial NCT03440060 (Procalcitonin-guided Antibiotic Therapy During Severe Exacerbation of COPD).
RaloxifeneA selective estrogen receptor modulator that is used to prevent and treat osteoporosis and reduce the risk of invasive breast cancer in high-risk postmenopausal women.
Risedronic acidA bisphosphonate used to treat osteoporosis and Paget's disease.
Salmon calcitoninA synthetic peptide form of calcitonin used to inhibit bone resorption in the treatment of hypercalcemia, osteoporosis, and Paget's disease.
Strontium ranelateA medication used for the management of severe osteoporosis in high-risk postmenopausal women and adult men.
TeriparatideA recombinant parathyroid hormone used for the treatment of osteoporosis.
Tiludronic acidA bisphosphonate used for the treatment of Paget's disease of bone.
ToremifeneA first generation nonsteroidal selective estrogen receptor modulator used to treat certain breast cancers.
Vitamin DAn ingredient found in a variety of supplements and vitamins.
Zoledronic acidA bisphosphonate used to treat malignancy associated hypercalcemia, multiple myeloma, and bone metastasis from solid tumors.
Drugs & Drug Targets
DrugTargetType
24,25-Dihydroxycholecalciferol25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrialenzyme
24,25-Dihydroxycholecalciferol1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrialenzyme
24,25-DihydroxycholecalciferolCatalasetarget
24,25-DihydroxycholecalciferolVitamin D-binding proteincarrier
AbaloparatideParathyroid hormone/parathyroid hormone-related peptide receptortarget
Alendronic acidFarnesyl pyrophosphate synthasetarget
Alendronic acidTyrosine-protein phosphatase non-receptor type 4target
Alendronic acidReceptor-type tyrosine-protein phosphatase Starget
Alendronic acidReceptor-type tyrosine-protein phosphatase epsilontarget
Alendronic acidV-type proton ATPase catalytic subunit Atarget
Alendronic acidHydroxylapatitetarget
AlfacalcidolAlpha globincarrier
AlfacalcidolVitamin D-binding proteincarrier
AlfacalcidolRetinoic acid receptor RXR-alphatarget
Alfacalcidol25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrialtarget
AlfacalcidolVitamin D3 receptortarget
BazedoxifeneEstrogen receptortarget
BazedoxifeneUDP-glucuronosyltransferase 1A10enzyme
BazedoxifeneUDP-glucuronosyltransferase 1A8enzyme
BazedoxifeneEstrogen receptor betatarget
BazedoxifeneEstrogen receptortarget
BazedoxifeneUDP-glucuronosyltransferase 1A4enzyme
Calcifediol1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrialenzyme
CalcifediolVitamin D3 receptortarget
Calcifediol25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrialenzyme
CalcitriolHomeobox protein Hox-A10target
CalcitriolVitamin D3 receptortarget
Calcitriol1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrialenzyme
CalcitriolCytochrome P450 3A4enzyme
CalcitriolVitamin D-binding proteincarrier
CholecalciferolCytochrome P450 2C8enzyme
CholecalciferolCytochrome P450 1A1enzyme
CholecalciferolVitamin D3 receptortarget
CholecalciferolCytochrome P450 3A4enzyme
CholecalciferolCytochrome P450 2J2enzyme
CholecalciferolSterol 26-hydroxylase, mitochondrialenzyme
CholecalciferolVitamin D 25-hydroxylaseenzyme
CholecalciferolCholesterol side-chain cleavage enzyme, mitochondrialenzyme
CholecalciferolVitamin D-binding proteincarrier
Clodronic acidHydroxylapatitetarget
Clodronic acidADP/ATP translocase 3target
Clodronic acidProstaglandin G/H synthase 2enzyme
Clodronic acidADP/ATP translocase 1target
Clodronic acidADP/ATP translocase 2target
DenosumabTumor necrosis factor ligand superfamily member 11target
DihydrotachysterolVitamin D3 receptortarget
DoxercalciferolVitamin D3 receptortarget
DoxercalciferolSterol 26-hydroxylase, mitochondrialenzyme
EldecalcitolVitamin D3 receptortarget
Ergocalciferol1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrialenzyme
Ergocalciferol25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrialenzyme
ErgocalciferolSterol 26-hydroxylase, mitochondrialenzyme
ErgocalciferolVitamin D 25-hydroxylaseenzyme
ErgocalciferolVitamin D-binding proteincarrier
ErgocalciferolVoltage-dependent calcium channeltarget
ErgocalciferolRibulose-phosphate 3-epimeraseenzyme
ErgocalciferolCholesterol side-chain cleavage enzyme, mitochondrialenzyme
ErgocalciferolVitamin D3 receptortarget
Etidronic acidADP/ATP translocase 3target
Etidronic acidADP/ATP translocase 2target
Etidronic acidADP/ATP translocase 1target
Etidronic acidV-type proton ATPase catalytic subunit Atarget
Etidronic acidReceptor-type tyrosine-protein phosphatase Starget
Etidronic acidHydroxylapatitetarget
Human calcitoninAminopeptidase Nenzyme
Human calcitoninAlpha-actinin-1target
Human calcitoninAlpha-N-acetylglucosaminidaseenzyme
Human calcitoninPhosphoglucomutase-1enzyme
Human calcitoninCalcitonin receptortarget
IbandronateGeranylgeranyl pyrophosphate synthasetarget
IbandronateHydroxylapatitetarget
IbandronateFarnesyl pyrophosphate synthasetarget
Incadronic acidCaspase-3target
Incadronic acidFarnesyl pyrophosphate synthasetarget
Incadronic acidCaspase-4target
Incadronic acidCaspase-7target
Nandrolone decanoateAndrogen receptortarget
Nandrolone decanoateAromataseenzyme
Nandrolone decanoateAmine oxidase [flavin-containing] Benzyme
Nandrolone decanoateAmine oxidase [flavin-containing] Aenzyme
Nandrolone decanoateProtein c-Fostarget
Nandrolone decanoate5-hydroxytryptamine 2 receptortarget
Nandrolone decanoate5-hydroxytryptamine receptor 1Btarget
Nandrolone decanoateInsulin-like growth factor 1 receptortarget
Nandrolone decanoateDopamine receptortarget
Nandrolone decanoateUDP-glucuronosyltransferase 2B7enzyme
Nandrolone decanoateUDP-glucuronosyltransferase 1A4enzyme
Nandrolone decanoateUDP-glucuronosyltransferase 2B4enzyme
Nandrolone decanoateUDP-glucuronosyltransferase 1A3enzyme
Nandrolone decanoateUDP-glucuronosyltransferase 1A1enzyme
Nandrolone decanoateUDP-glucuronosyltransferase 1A10enzyme
Nandrolone decanoateSex hormone-binding globulincarrier
Pamidronic acidFarnesyl pyrophosphate synthasetarget
Pamidronic acidHydroxylapatitetarget
Pamidronic acidGeranylgeranyl pyrophosphate synthasetarget
Pamidronic acidCaspase-3target
Pamidronic acidCaspase-9target
ParicalcitolUDP-glucuronosyltransferase 1A4enzyme
ParicalcitolCytochrome P450 3A4enzyme
Paricalcitol1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrialenzyme
ParicalcitolVitamin D3 receptortarget
RaloxifeneUDP-glucuronosyltransferase 1A8enzyme
RaloxifeneCytochrome P450 2C8enzyme
RaloxifeneSolute carrier organic anion transporter family member 1B1transporter
RaloxifeneSolute carrier organic anion transporter family member 1B3transporter
RaloxifeneATP-dependent translocase ABCB1transporter
RaloxifeneBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RaloxifeneAlbumincarrier
RaloxifeneUDP-glucuronosyltransferase 1A1enzyme
RaloxifeneTrefoil factor 1target
RaloxifeneUDP-glucuronosyltransferase 1A10enzyme
RaloxifeneATP-binding cassette sub-family C member 4transporter
RaloxifeneATP-binding cassette sub-family C member 3transporter
RaloxifeneATP-binding cassette sub-family C member 2transporter
RaloxifeneSerpin B9target
RaloxifeneCytochrome P450 3A4enzyme
RaloxifeneAlpha-1-acid glycoprotein 1carrier
RaloxifeneAromataseenzyme
RaloxifeneCytochrome P450 2B6enzyme
RaloxifeneEstrogen receptortarget
RaloxifeneAldehyde oxidaseenzyme
RaloxifeneEstrogen receptor betatarget
Risedronic acidFarnesyl pyrophosphate synthasetarget
Risedronic acidHydroxylapatitetarget
Risedronic acidProstaglandin G/H synthase 2enzyme
Salmon calcitoninCalcitonin receptortarget
Strontium ranelateExtracellular calcium-sensing receptortarget
TeriparatideParathyroid hormonetarget
TeriparatideParathyroid hormone/parathyroid hormone-related peptide receptortarget
Tiludronic acidReceptor-type tyrosine-protein phosphatase epsilontarget
Tiludronic acidTyrosine-protein phosphatase non-receptor type 6target
Tiludronic acidAlbumincarrier
Tiludronic acidAdenosine triphosphate (ATP)target
Tiludronic acidHydroxylapatitetarget
Tiludronic acidV-ATPase Subunitstarget
Tiludronic acidTyrosine-protein phosphatase non-receptor type 12target
ToremifeneEstrogen receptortarget
ToremifeneSex hormone-binding globulintarget
ToremifeneCytochrome P450 1A1enzyme
ToremifeneATP-dependent translocase ABCB1transporter
ToremifeneCytochrome P450 3A4enzyme
ToremifeneEstrogen receptortarget
Vitamin DVitamin D3 receptortarget
Vitamin DVitamin D-binding proteintarget
Vitamin DVitamin D 25-hydroxylaseenzyme
Vitamin D25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrialenzyme
Vitamin DCytochrome P450 3A4enzyme
Zoledronic acidMultidrug resistance-associated protein 1transporter
Zoledronic acidHydroxylapatitetarget
Zoledronic acidGeranylgeranyl pyrophosphate synthasetarget
Zoledronic acidFarnesyl pyrophosphate synthasetarget