| MSX-122 | Organic compounds | Benzenoids | Benzene and substituted derivatives | Benzylamines | Details |
| NB-001 | Organic compounds | Organoheterocyclic compounds | Imidazopyrimidines | Purines and purine derivatives | Details |
| Mibampator | Organic compounds | Benzenoids | Benzene and substituted derivatives | Biphenyls and derivatives | Details |
| Carlumab | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Turofexorate isopropyl | Organic compounds | Organoheterocyclic compounds | Indoles and derivatives | Indoles | Details |
| Nivocasan | Organic compounds | Organoheterocyclic compounds | Isoquinolines and derivatives | Not Available | Details |
| RO-5028442 | Organic compounds | Organoheterocyclic compounds | Indoles and derivatives | Indolecarboxylic acids and derivatives | Details |
| N-sulfoglucosamine sulfohydrolase recombinant | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| AZD-7295 | Organic compounds | Benzenoids | Benzene and substituted derivatives | Anilides | Details |
| Felcisetrag | Organic compounds | Organoheterocyclic compounds | Benzimidazoles | Not Available | Details |
| Monteplase | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Perfosfamide | Organic compounds | Organic nitrogen compounds | Organonitrogen compounds | Nitrogen mustard compounds | Details |
| Fenpropidin | Organic compounds | Benzenoids | Benzene and substituted derivatives | Phenylpropanes | Details |
| ASP-3026 | Organic compounds | Organoheterocyclic compounds | Piperidines | Phenylpiperidines | Details |
| Dolastatin 10 | Organic compounds | Organic acids and derivatives | Peptidomimetics | Hybrid peptides | Details |
| Daporinad | Organic compounds | Benzenoids | Benzene and substituted derivatives | Benzoyl derivatives | Details |
| Firategrast | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| Dipraglurant | Organic compounds | Organoheterocyclic compounds | Imidazopyridines | Not Available | Details |
| Demcizumab | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Etanidazole | Organic compounds | Organic nitrogen compounds | Organonitrogen compounds | Amines | Details |
| Brontictuzumab | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Tiplimotide | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Bindarit | Organic compounds | Organoheterocyclic compounds | Benzopyrazoles | Indazoles | Details |
| CC-115 | Organic compounds | Organoheterocyclic compounds | Pyridines and derivatives | Pyridyltriazoles | Details |
| DTP-348 | Organic compounds | Organoheterocyclic compounds | Azoles | Imidazoles | Details |
| Amuvatinib | Organic compounds | Organoheterocyclic compounds | Diazinanes | Piperazines | Details |
| Z-160 | Organic compounds | Benzenoids | Benzene and substituted derivatives | Diphenylmethanes | Details |
| CGI-1842 | Organic compounds | Benzenoids | Benzene and substituted derivatives | N-phenylureas | Details |
| GSK-690693 | Organic compounds | Organoheterocyclic compounds | Imidazopyridines | Imidazo-[4,5-c]pyridines | Details |
| AKN-028 | Organic compounds | Organoheterocyclic compounds | Indoles and derivatives | Indoles | Details |