| Patidegib | Organic compounds | Organoheterocyclic compounds | Piperidines | Not Available | Details |
| Somatorelin | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| JNJ-42396302 | Organic compounds | Organic nitrogen compounds | Organonitrogen compounds | Amines | Details |
| AFN-1252 | Organic compounds | Organoheterocyclic compounds | Diazanaphthalenes | Naphthyridines | Details |
| SJ-733 | Organic compounds | Organoheterocyclic compounds | Isoquinolines and derivatives | Isoquinolones and derivatives | Details |
| Samatasvir | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| Urapidil | Organic compounds | Organoheterocyclic compounds | Diazinanes | Piperazines | Details |
| Naveglitazar | Organic compounds | Benzenoids | Benzene and substituted derivatives | Diphenylethers | Details |
| Letrazuril | Organic compounds | Benzenoids | Benzene and substituted derivatives | Diphenylacetonitriles | Details |
| Indantadol | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| Isoquercetin | Organic compounds | Phenylpropanoids and polyketides | Flavonoids | Flavonoid glycosides | Details |
| Emapunil | Organic compounds | Organoheterocyclic compounds | Imidazopyrimidines | Purines and purine derivatives | Details |
| Protionamide | Organic compounds | Organoheterocyclic compounds | Pyridines and derivatives | Not Available | Details |
| Metenkefalin | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| 4SC-203 | Organic compounds | Organoheterocyclic compounds | Diazanaphthalenes | Benzodiazines | Details |
| Rolofylline | Organic compounds | Organoheterocyclic compounds | Imidazopyrimidines | Purines and purine derivatives | Details |
| Beloranib | Organic compounds | Phenylpropanoids and polyketides | Cinnamic acids and derivatives | Cinnamic acid esters | Details |
| Icaritin | Organic compounds | Phenylpropanoids and polyketides | Flavonoids | Flavones | Details |
| ATX-914 | Organic compounds | Organoheterocyclic compounds | Diazines | Pyrimidines and pyrimidine derivatives | Details |
| Lurbinectedin | Organic compounds | Alkaloids and derivatives | Harmala alkaloids | Not Available | Details |
| PF-04995274 | Organic compounds | Organoheterocyclic compounds | Benzisoxazoles | Not Available | Details |
| Modufolin | Organic compounds | Organoheterocyclic compounds | Pteridines and derivatives | Pterins and derivatives | Details |
| Soblidotin | Organic compounds | Organic acids and derivatives | Peptidomimetics | Hybrid peptides | Details |
| Relamorelin | Organic compounds | Organic acids and derivatives | Peptidomimetics | Hybrid peptides | Details |
| WP-1066 | Organic compounds | Organoheterocyclic compounds | Pyridines and derivatives | Halopyridines | Details |
| Intepirdine | Organic compounds | Organoheterocyclic compounds | Diazinanes | Piperazines | Details |
| Salirasib | Organic compounds | Lipids and lipid-like molecules | Prenol lipids | Sesquiterpenoids | Details |
| Mubritinib | Organic compounds | Benzenoids | Benzene and substituted derivatives | Phenylbutylamines | Details |
| Lumretuzumab | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Aviscumine | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |