LY-2183240

DB17035ExperimentalSmall molecule

LY-2183240 is an inhibitor of endocannabinoid reuptake/breakdown.

Mechanism: Pharmacologically active on Cannabinoid receptor 1, Fatty-acid amide hydrolase 1, and Monoglyceride lipase
Curator reviewed
Formula / weight: C₁₇H₁₇N₅O · 307.357 g/mol (avg)
Also known as: 1h-tetrazole-1-carboxamide, 5-((1,1'-biphenyl)-4-ylmethyl)-n,n-dimethyl- · 5-(biphenyl-4-ylmethyl)-n,n-dimethyl-1h-tetrazole-1-carboxamide
Code names: LY-2183240

Resolves to

Compound

Structure

InChIKeyGZNIYOXWFCDBBJ-UHFFFAOYSA-NSMILESCN(C)C(=O)N1N=NN=C1CC1=CC=C(C=C1)C1=CC=CC=C1

Targets

What you can answer from here — as of July 08, 2026

3Protein targetsEach mapped to UniProt, with action and pharmacological action

Listed above

5+ReferencesStructured and connected to the statements they support

Which drugs share a target with LY-2183240, and which of those have an active Phase 3 trial?

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