| DB00470 | Dronabinol | approved, illicit | yes | agonist | Details |
| DB00486 | Nabilone | approved, investigational | yes | partial agonist | Details |
| DB05201 | V24343 | investigational | unknown | | Details |
| DB11745 | Otenabant | investigational | unknown | | Details |
| DB05077 | SLV319 | investigational | unknown | | Details |
| DB05750 | AVE-1625 | investigational | unknown | | Details |
| DB06155 | Rimonabant | approved, investigational | yes | antagonist | Details |
| DB02955 | Ricinoleic acid | experimental | unknown | | Details |
| DB09061 | Cannabidiol | approved, investigational | yes | antagonistmodulator | Details |
| DB09288 | Propacetamol | experimental | yes | antagonist | Details |
| DB14011 | Nabiximols | investigational | yes | | Details |
| DB14009 | Medical Cannabis | experimental, investigational | yes | negative modulator | Details |
| DB11755 | Tetrahydrocannabivarin | investigational | yes | antagonist | Details |