Valemetostat

DB18314InvestigationalSmall molecule

Valemetostat: Overview.

Chemical structure of Valemetostat
Formula / weight
C26H34ClN3O4 · 488.03 g/mol (avg)
Also known as
Ezh1/2 inhibitor ds-3201

Resolves to

Compound
UNII60RD0234VECAS1809336-39-7ChEMBLCHEMBL4597193
Structure
InChIKeySSDRNUPMYCFXGM-UYPAYLBCSA-NSMILES[H][C@@]1(CC[C@@H](CC1)N(C)C)[C@@]1(C)OC2=C(O1)C(C)=C(C=C2Cl)C(=O)NCC1=C(C)C=C(C)NC1=O
Targets
Q92800EZH1Q15910EZH2

What you can answer from here — as of September 23, 2026

2Protein targetsEach mapped to UniProt, with action and pharmacological action
Listed above
15Clinical trialsPhase, status and sponsor resolved per trial
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2+ReferencesStructured and connected to the statements they support
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Which drugs share a target with Valemetostat, and which of those have an active Phase 3 trial?

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