Ditekiren

DB19992ExperimentalSmall molecule

Ditekiren is a small molecule drug. The usage of the INN stem '-kiren' in the name indicates that Ditekiren is a renin inhibitor. Ditekiren has a monoisotopic molecular weight of...

Mechanism: Pharmacologically active on Renin
Curator reviewed
Formula / weight: C₅₀H₇₅N₉O₈ · 930.205 g/mol (avg)
Code names: MCMC-6317 · U-71038

Resolves to

Compound

UNII5355S3W1ISCAS103336-05-6ChEMBLCHEMBL1790497

Structure

InChIKeySASWSEQJAITMKS-JJNNLWIXSA-NSMILES

CC[C@H](C)[C@H](NC(=O)[C@@H](C[C@H](O)[C@H](CC(C)C)NC(=O)[C@H](CC1=CN=CN1)N(C)C(=O)[C@H](CC1=CC=CC=C1)NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C)C(=O)NCC1=CC=CC=N1

Targets

P00797REN

Transporters

O95342ABCB11P08183ABCB1

What you can answer from here — as of September 20, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

2TransportersSubstrate / inhibitor direction, not just membership

Listed above

5+ReferencesStructured and connected to the statements they support

Which drugs share a target with Ditekiren, and which of those have an active Phase 3 trial?

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