Hypermenorrhea

Also known as: Menorrhagia / Excessive and frequent menstruation with regular cycle / Heavy menstrual bleeding / Menorrhagia (finding) / Menstrual flow excessive / Hypermenorrhoea / Heavy periods / Excessive menstruation / Bleeding menstrual heavy / Menses regular with excessive bleeding / Prolonged heavy periods / Menstruation increased

DrugDrug NameDrug Description
DB09123DienogestAn oral progestin used for the treatment of endometriosis as monotherapy or contraception in combination with ethinylestradiol.
DB00823Ethynodiol diacetateAn oral contraceptive used to prevent pregnancy.
DB00367LevonorgestrelA progestin found in oral and IUD contraceptives and at higher doses in emergency contraceptives.
DB12474LynestrenolA progestin used for contraception and in the treatment of menstrual disorders.
DB00939Meclofenamic acidAn NSAID used to treat mild to moderate pain, primary dysmenorrhea, heavy menstrual blood loss, rheumatoid arthritis, and osteoarthritis.
DB01357MestranolA synthetic estradiol found in oral contraceptive pills for contraception and the treatment of other conditions in the female reproductive system, such as dysmenorrhea and dysfunctional uterine bleeding.
DB00957NorgestimateA progesterone used as a contraceptive and to treat acne vulgaris.
DB09389NorgestrelA progestin used in combination with ethinyl estradiol for oral contraception and prevention of pregnancy in women.
DrugDrug NameTargetType
DB09123DienogestCytochrome P450 3A4enzyme
DB09123DienogestProgesterone receptortarget
DB09123DienogestAndrogen receptortarget
DB00823Ethynodiol diacetateEstrogen receptor alphatarget
DB00823Ethynodiol diacetateProgesterone receptortarget
DB00823Ethynodiol diacetateCytochrome P450 3A4enzyme
DB00367LevonorgestrelProgesterone receptortarget
DB00367LevonorgestrelEstrogen receptor alphatarget
DB00367Levonorgestrel3-oxo-5-alpha-steroid 4-dehydrogenase 1target
DB00367LevonorgestrelCytochrome P450 3A4enzyme
DB00367LevonorgestrelAndrogen receptortarget
DB00367LevonorgestrelSex hormone-binding globulintarget
DB00367LevonorgestrelGlucocorticoid receptortarget
DB00367LevonorgestrelCytochrome P450 3A5enzyme
DB12474LynestrenolCytochrome P450 3A4enzyme
DB12474LynestrenolCytochrome P450 2C9enzyme
DB12474LynestrenolCytochrome P450 2C19enzyme
DB00939Meclofenamic acidProstaglandin G/H synthase 1target
DB00939Meclofenamic acidProstaglandin G/H synthase 2target
DB00939Meclofenamic acidArachidonate 5-lipoxygenasetarget
DB00939Meclofenamic acidSolute carrier family 22 member 6transporter
DB00939Meclofenamic acidSolute carrier organic anion transporter family member 1C1transporter
DB00939Meclofenamic acidPotassium voltage-gated channel subfamily KQT member 2target
DB00939Meclofenamic acidPotassium voltage-gated channel subfamily KQT member 3target
DB00939Meclofenamic acidThyroxine-binding globulincarrier
DB01357MestranolEstrogen receptor alphatarget
DB01357MestranolCytochrome P450 2C9enzyme
DB01357MestranolCytochrome P450 3A4enzyme
DB01357MestranolCytochrome P450 2C8enzyme
DB00957NorgestimateProgesterone receptortarget
DB00957NorgestimateEstrogen receptor alphatarget
DB00957NorgestimateCanalicular multispecific organic anion transporter 1transporter
DB00957NorgestimateCytochrome P450 3A4enzyme
DB00957NorgestimateAndrogen receptortarget
DB00957NorgestimateCytochrome P450 2B6enzyme
DB00957NorgestimateCytochrome P450 2C9enzyme
DB00957NorgestimateUDP-glucuronosyltransferase 1-1enzyme
DB00957NorgestimateSerum albumincarrier
DB00957NorgestimateSex hormone-binding globulincarrier
DB00957NorgestimateP-glycoprotein 1transporter
DB09389NorgestrelProgesterone receptortarget
DB09389Norgestrel3-oxo-5-alpha-steroid 4-dehydrogenase 1target
DB09389NorgestrelAndrogen receptortarget
DB09389NorgestrelCytochrome P450 3A4enzyme
DB09389NorgestrelCytochrome P450 19A1enzyme
DrugDrug NamePhaseStatusCount
DB08995Diosmin1 / 2Unknown Status1
DB00302Tranexamic acid1 / 2Unknown Status1
DB06680Asoprisnil2Completed1
DB06680Asoprisnil3Completed6
DB13529Dobesilic acid3Unknown Status1
DB00367Levonorgestrel3Completed3
DB00603Medroxyprogesterone acetate3Completed1
DB00603Medroxyprogesterone acetate3Terminated1
DB00929Misoprostol3Withdrawn1
DB00302Tranexamic acid3Completed4
DB00302Tranexamic acid3Unknown Status1
DB04928XP12B3Completed4
DB00783Estradiol4Recruiting1
DB00783Estradiol4Unknown Status1
DB00977Ethinylestradiol4Completed1
DB00367Levonorgestrel4Completed3
DB00929Misoprostol4Completed1
DB00788Naproxen4Completed2
DB13981Nomegestrol acetate4Unknown Status1
DB00717Norethisterone4Recruiting1
DB00717Norethisterone4Unknown Status1
DB11853Relugolix4Recruiting1
DB00675Tamoxifen4Completed1
DB00302Tranexamic acid4Completed3
DB01281AbataceptNot AvailableRecruiting1
DB00945Acetylsalicylic acidNot AvailableRecruiting1
DB00513Aminocaproic acidNot AvailableRecruiting1
DB01118AmiodaroneNot AvailableRecruiting1
DB00182AmphetamineNot AvailableRecruiting1
DB00026AnakinraNot AvailableRecruiting1
DB00207AzithromycinNot AvailableRecruiting1
DB00559BosentanNot AvailableRecruiting1
DB01222BudesonideNot AvailableRecruiting1
DB06168CanakinumabNot AvailableRecruiting1
DB00535CefdinirNot AvailableRecruiting1
DB01413CefepimeNot AvailableRecruiting1
DB00438CeftazidimeNot AvailableRecruiting1
DB01190ClindamycinNot AvailableRecruiting1
DB00349ClobazamNot AvailableRecruiting1
DB01394ColchicineNot AvailableRecruiting1
DB00035DesmopressinNot AvailableCompleted1
DB01234DexamethasoneNot AvailableRecruiting1
DB00633DexmedetomidineNot AvailableRecruiting1
DB09123DienogestNot AvailableCompleted1
DB13956Estradiol valerateNot AvailableCompleted1
DB00977EthinylestradiolNot AvailableCompleted1
DB00294EtonogestrelNot AvailableCompleted1
DB00828FosfomycinNot AvailableRecruiting1
DB00695FurosemideNot AvailableRecruiting1
DB00996GabapentinNot AvailableRecruiting1
DB01018GuanfacineNot AvailableRecruiting1
DB00741HydrocortisoneNot AvailableRecruiting1
DB00065InfliximabNot AvailableRecruiting1
DB00598LabetalolNot AvailableRecruiting1
DB00367LevonorgestrelNot AvailableCompleted4
DB01601LopinavirNot AvailableRecruiting1
DB00603Medroxyprogesterone acetateNot AvailableCompleted2
DB00760MeropenemNot AvailableRecruiting1
DB00331MetforminNot AvailableRecruiting1
DB00235MilrinoneNot AvailableRecruiting1
DB00844NalbuphineNot AvailableRecruiting1
DB00622NicardipineNot AvailableRecruiting1
DB01115NifedipineNot AvailableRecruiting1
DB00717NorethisteroneNot AvailableCompleted1
DB00198OseltamivirNot AvailableRecruiting1
DB00497OxycodoneNot AvailableRecruiting1
DB14761RemdesivirNot AvailableRecruiting1
DB00811RibavirinNot AvailableRecruiting1
DB00734RisperidoneNot AvailableRecruiting1
DB00503RitonavirNot AvailableRecruiting1
DB08877RuxolitinibNot AvailableRecruiting1
DB11767SarilumabNot AvailableRecruiting1
DB01104SertralineNot AvailableRecruiting1
DB00658SevelamerNot AvailableRecruiting1
DB00421SpironolactoneNot AvailableRecruiting1
DB00871TerbutalineNot AvailableRecruiting1
DB06273TocilizumabNot AvailableRecruiting1
DB00302Tranexamic acidNot AvailableCompleted2
DB00302Tranexamic acidNot AvailableRecruiting1
DB00582VoriconazoleNot AvailableRecruiting1
DB00425ZolpidemNot AvailableRecruiting1