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Elraglusib
go.drugbank.com/drugs/DB16047InvestigationalElraglusib is under investigation in clinical trial NCT04218071 (Actuate 1901: 9-ING-41 in Myelofibrosis).
Synonyms: 1H-Pyrrole-2,5-dione, 3-(5-fluoro-3-benzofuranyl)-4-(5-methyl-5H-1,3-dioxolo(4,5-F)indol-7-yl)-, 3-(5-Fluoro-benzofuran-3-yl)-4-(5-methyl-5H-(1,3)dioxolo(4,5-F)indol-7-yl)-pyrrole-2,5-dioneBrivudine monophosphate
go.drugbank.com/drugs/DB04438ExperimentalSynonyms: Bvdu 5'-monophosphate, BVDU-MPAdenylate-3'-phosphate-[[2'-deoxy-uridine-5'-phosphate]-3'-phosphate]
go.drugbank.com/drugs/DB03186ExperimentalSynonyms: Adenylate-3'-phosphate-[[2'-deoxy-uridine-5'-phosphate]-3'-phosphate], U-PI-A-PIHonokiol
go.drugbank.com/drugs/DB19283InvestigationalHonokiol is under investigation in clinical trial NCT00966953 (Development of Clinical Method to Determination Triclosan Retention in Plaque Following Brushing.).
Synonyms: 3',5-diallyl-2,4'-biphenyldiol, (1,1'-biphenyl)-2,4'-diol, 3',5-di-2-propen-1-yl-Categories: Heterocyclic Compounds, 2-RingRisedronic acid
go.drugbank.com/drugs/DB00884ApprovedInvestigationalRisedronic acid is a third generation bisphosphonate that is used for the treatment of some forms of osteoperosis and Paget's disease[FDA Label][A959,A203111].
Mixtures: BONEPLUS D3 150 MG/2800 IU EFERVESAN TABLET, 3 ADET, RISEPLUS D3 150 MG/5600 IU EFERVESAN TABLET, 3 ADETCategories: Heterocyclic Compounds, 1-RingRiboflavin tetrabutyrate
go.drugbank.com/drugs/DB14727InvestigationalSynonyms: Riboflavin 2',3',4',5'-tetrabutyrate, Riboflavin, 2',3',4',5'-tetrabutanoateCategories: Heterocyclic Compounds, 3-Ring, Heterocyclic Compounds, 2-RingFurvina
go.drugbank.com/drugs/DB16547ExperimentalFurvina is marketed in Cuba as Dermofural®, an ointment containing G1 as the only active principle ingredient. It is used to treat dermatological infections.[A228063]
Categories: Heterocyclic Compounds, 1-RingSynonyms: 2-Bromo-5-(2-bromo-2-nitrovinyl)furan, 1-(5-Bromofur-2-yl)-2-bromo-2-nitroetheneAPL-030
go.drugbank.com/drugs/DB18735ExperimentalAPL-030 is a orally-active small molecule inhibitor of GCN2.
Synonyms: N-(4-((2-aminopyrimidin-5-yl)ethynyl)-3-fluoropyridin-2-yl)-5-chloro-2-methoxypyridine-3-sulfonamideHydroxychloroquine
go.drugbank.com/drugs/DB01611ApprovedInvestigational[A192132] **The FDA emergency use authorization for hydroxychloroquine and [chloroquine] in the treatment of COVID-19 was revoked on 15 June 2020. … Hydroxychloroquine is a racemic mixture consisting of an R and S enantiomer.[A183047] Hydroxychloroquine is an aminoquinoline like [chloroquine].
Categories: Cytochrome P-450 Substrates, Cytochrome P-450 CYP2C8 SubstratesSynonyms: 7-chloro-4-[5-(N-ethyl-N-2-hydroxyethylamino)-2-pentyl]aminoquinoline, 2-((4-((7-chloro-4-quinolyl)amino)pentyl)ethylamino)ethanolTricyclazole
go.drugbank.com/drugs/DB02891InvestigationalSynonyms: 5-methyl-1,2,4-triazolo(3,4-b)benzothiazole, 5-methyl-1,2,4-triazolo(3,4-b)(1,3)benzothiazoleCategories: Heterocyclic Compounds, 1-Ring