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Tricetin
go.drugbank.com/drugs/DB08230ExperimentalSynonyms: 5,7,3',4',5'-Pentahydroxyflavone, 3',4',5,5',7-pentahydroxyflavoneCategories: Compounds used in a research, industrial, or household setting, Heterocyclic Compounds, 1-RingNamodenoson
go.drugbank.com/drugs/DB12885InvestigationalNamodenoson has been used in trials studying the treatment of Chronic Hepatitis C and Hepatocellular Carcinoma.
Synonyms: 2-Chloro-N(6)-(3-iodobenzyl)adenosine-5'-N-methyluronamideCategories: Heterocyclic Compounds, 2-RingTaminadenant
go.drugbank.com/drugs/DB18811InvestigationalSynonyms: 4-pyrimidinamine, 5-bromo-2,6-di-1h-pyrazol-1-yl-Bimiralisib
go.drugbank.com/drugs/DB14846InvestigationalBimiralisib is under investigation in clinical trial NCT02723877 (PQR309 and Eribulin in Metastatic HER2 Negative and Triple-negative Breast Cancer (PIQHASSO)).
Synonyms: 2-Pyridinamine, 5-(4,6-di-4-morpholinyl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)-, 5-(4,6-Dimorpholino-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amineL-Saccharopine
go.drugbank.com/drugs/DB04207ExperimentalSynonyms: N-[(S)-5-Amino-5-carboxypentyl]-L-glutamic acid, epsilon-N-(L-Glutar-2-yl)-L-lysineFobrepodacin
go.drugbank.com/drugs/DB18409ExperimentalSynonyms: N-ethyl-n'-(6-fluoro-5-(2-(1-methyl-1-(phosphonooxy)ethyl)-5-pyrimidinyl)-7-((2r)-tetrahydro-2-furanyl)-1h-benzimidazol-2-yl)urea, Urea, n-ethyl-n'-(6-fluoro-5-(2-(1-methyl-1-(phosphonooxy)ethyl)-5-pyrimidinyl)-7-((2r)-tetrahydro-2-furanyl)-1h-benzimidazol-2-yl)-Isuzinaxib
go.drugbank.com/drugs/DB19109InvestigationalIsuzinaxib is under investigation in clinical trial NCT05758896 (Study of APX-115 in Contrast Induced Acute Kidney Injury in Subjects Undergoing PCI).
Categories: Heterocyclic Compounds, 1-RingSynonyms: 1-(pyridin-2-yl)-3-phenyl-4-propyl-1h-pyrazol-5-ol, 1h-pyrazol-5-ol, 3-phenyl-4-propyl-1-(2-pyridinyl)-Sonrotoclax
go.drugbank.com/drugs/DB18753ApprovedInvestigationallines of systemic therapy, including a BTK inhibitor. … Sonrotoclax is a selective, potent, small-molecule inhibitor of BCL-2, an antiapoptotic protein overexpressed in B-cell malignancies.
Categories: BCL-2 Inhibitor, P-glycoprotein substratesSynonyms: N-[4-({[(1r,4r)-4-hydroxy-4-methylcyclohexyl]methyl}amino)-3- nitrobenzene-1-sulfonyl]-4-(2-{(2S)-2-[2-(propan-2-yl)phenyl]pyrrolidin- 1-yl}-7-azaspiro[3.5]nonan-7-yl)-2-[(1H-pyrrolo[2,3-b]pyridin-5- ylCholesteryl Linoleate
go.drugbank.com/drugs/DB02092ExperimentalSynonyms: (3β)-cholest-5-en-3-ol, (Z,Z)-9,12-octadecadienoate, cholest-5-en-3β-yl (Z,Z)-octadeca-9,12-dienoateTemuterkib
go.drugbank.com/drugs/DB18806InvestigationalSynonyms: 4h-thieno(2,3-c)pyrrol-4-one, 5,6-dihydro-6,6-dimethyl-2-(2-((1-methyl-1h-pyrazol-5-yl)amino)-4-pyrimidinyl)-5-(2-(4-morpholinyl)ethyl)-, 5,6-dihydro-6,6-dimethyl-2-(2-((1-methyl-1h-pyrazol-5-yl)amino)-4-pyrimidinyl)-5-(2-(4-morpholinyl)ethyl)-4h-thieno(2,3-c)pyrrol-4-oneCategories: Heterocyclic Compounds, 1-Ring