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Thymectacin
go.drugbank.com/drugs/DB05116InvestigationalThymectacin is selectively active against tumor cells expressing high levels of thymidylate synthase (TS), a critical enzyme in DNA biosynthesis. … Thymectacin, a phosphoramidate derivative of (E)-5-(2-bromovinyl)-2'-deoxyuridine, is a novel small molecule anticancer agent.
Categories: Nucleic Acids, Nucleotides, and NucleosidesManaglinat dialanetil
go.drugbank.com/drugs/DB05518InvestigationalCS-917 is a novel inhibitor of fructose 1,6-bisphphosphatase (FBPase) which is one of the rate-limiting enzymes of gluconeogenesis.
Categories: Amino Acids, Peptides, and ProteinsGTI-2040
go.drugbank.com/drugs/DB15030ExperimentalGTI-2040 is under investigation in clinical trial NCT00084643 (GTI-2040, Oxaliplatin, and Capecitabine in Treating Patients With Locally Advanced or Metastatic Colorectal Cancer or Other Solid Tumors).
Categories: Nucleic Acids, Nucleotides, and NucleosidesAzadirachtin
go.drugbank.com/drugs/DB19419InvestigationalAzadirachtin is under investigation in clinical trial NCT06617026 (Short-term Outcome of Medical vs. Surgical Management of Chronic Anal Fissure).
Categories: Compounds used in a research, industrial, or household settingMarzeptacog alfa (activated)
go.drugbank.com/drugs/DB15278InvestigationalMarzeptacog alfa (activated) is under investigation in clinical trial NCT01439971 (Phase 1 Safety, Pharmacokinetics And Pharmacodynamics Study Of Recombinant Factor VIIa Variant (813d) In Adult Subjects
Categories: Enzymes and Coenzymes, Amino Acids, Peptides, and ProteinsRotigaptide
go.drugbank.com/drugs/DB13067InvestigationalRotigaptide is under investigation for the basic science of Heart Disease and Vascular Disease.
Categories: Amino Acids, Peptides, and ProteinsEsflurbiprofen
go.drugbank.com/drugs/DB16159InvestigationalEsflurbiprofen is under investigation in clinical trial NCT03434197 (Safety and Efficacy of SFPP in Knee Osteoarthritis).
Categories: Topical Products for Joint and Muscular PainProducts: LOCOA 40MG TRANSDERMAL PATCHPegbelfermin
go.drugbank.com/drugs/DB15365InvestigationalPegbelfermin is under investigation in clinical trial NCT03486899 (A Study of Experimental Medication BMS-986036 in Adults With Nonalcoholic Steatohepatitis (NASH) and Stage 3 Liver Fibrosis).
Categories: Amino Acids, Peptides, and Proteins, Intercellular Signaling Peptides and ProteinsAbelacimab
go.drugbank.com/drugs/DB16682InvestigationalAbelacimab is under investigation in clinical trial NCT04755283 (Safety and Tolerability of Abelacimab (MAA868) vs. Rivaroxaban in Patients With Atrial Fibrillation).
Categories: Amino Acids, Peptides, and ProteinsBimagrumab
go.drugbank.com/drugs/DB12584InvestigationalBimagrumab has been used in trials studying the treatment and supportive care of Sarcopenia, Skeletal Muscle, Mechanical Ventilation, Sporadic Inclusion Body Myositis, and Sporadic Inclusion Body Myositis
Categories: Amino Acids, Peptides, and Proteins