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Displaying results 1 - 10 of 10000 in total
  1. Drug

    Estradiol

    go.drugbank.com/drugs/DB00783
    ApprovedInvestigationalVet approved

    Because it has a low oral bioavailability on its own, estradiol is commonly formulated with an ester side-chain. … Estradiol is a naturally occurring hormone circulating endogenously in females.

    Synonyms: Estradiol, 17-β estradiolSalts: Estradiol hemihydrate
  2. Drug

    Estradiol valerate

    go.drugbank.com/drugs/DB13956
    ApprovedInvestigationalVet approved

    [DB00783] is commonly produced with an ester side-chain as endogenous estradiol has very low oral bioavailability on its own (2-10%). … Estradiol valerate is commercially available as an intramuscular injection as the product Delestrogen and is indicated for the treatment of moderate to severe vasomotor symptoms and vulvovaginal atrophy

    Synonyms: Estradiol valerateMixtures: Estradiol Valerate and Estradiol Valerate/Dienogest, Estradiol Valerate and Estradiol Valerate/Dienogest
  3. Drug

    Estradiol benzoate

    go.drugbank.com/drugs/DB13953
    ApprovedVet approvedWithdrawn

    Ester pro-drugs of estradiol are therefore considered to be bioidentical forms of estrogen [T84]. Estradiol benzoate is not currently available in Canada or the US. … [DB00783] is commonly produced with an ester side-chain as endogenous estradiol has very low oral bioavailability on its own (2-10%).

    Categories: Estradiol CongenersSynonyms: Estradiol benzoate, benzoato de estradiol
  4. Drug

    Estradiol cypionate

    go.drugbank.com/drugs/DB13954
    ApprovedVet approved

    [DB00783] is commonly produced with an ester side-chain as endogenous estradiol has very low oral bioavailability on its own (2-10%). … Estradiol cypionate is commercially available as Depo-Estradiol, an intramuscular depot injection used for the treatment of moderate to severe vasomotor symptoms associated with menopause and for the treatment

    Synonyms: Estradiol cypionateMixtures: OBAT SUNTIK KB II
  5. Drug

    Estradiol dienanthate

    go.drugbank.com/drugs/DB13955
    ApprovedVet approvedWithdrawn

    Estradiol dienanthate is not currently available in any commercially available products in Canada or the US. … Estradiol is commonly produced with an ester side-chain as endogenous estradiol has very low oral bioavailability on its own (2-10%).

    Synonyms: Estradiol dienantate, Estradiol dienanthateCategories: Estradiol Congeners
  6. Drug

    Estradiol acetate

    go.drugbank.com/drugs/DB13952
    ApprovedVet approved

    [DB00783] is commonly produced with an ester side-chain as endogenous estradiol has very low oral bioavailability on its own (2-10%). … As a pro-drug of estradiol, estradiol acetate therefore has the same downstream effects within the body through binding to the Estrogen Receptor (ER) including ERα and ERβ subtypes, which are located in

    Synonyms: Estradiol acetate, Estradiol 3-acetate
  7. Drug

    Ethinylestradiol

    go.drugbank.com/drugs/DB00977
    ApprovedInvestigational

    [A191107] These properties were achieved by the substitution of an ethinyl group at carbon 17 of [estradiol].[A191107] Ethinylestradiol soon replaced [mestranol] in contraceptive pills. … Ethinylestradiol was first synthesized in 1938 by Hans Herloff Inhoffen and Walter Hohlweg at Schering.[A191107] It was developed in an effort to create an estrogen with greater oral bioavailability.

    Synonyms: Ethinyl estradiol, 17-ethinyl-3,17-estradiolMixtures: Drospirenone and Ethinyl Estradiol Tablets USP, Drospirenone and Ethinyl Estradiol Tablets USP 21
  8. Drug

    Estramustine

    go.drugbank.com/drugs/DB01196
    ApprovedWithdrawn

    A nitrogen mustard linked to estradiol, usually as phosphate; used to treat prostatic neoplasms; also has radiation protective properties.

    Categories: Estradiol CongenersSynonyms: 17β-Estradiol 3-(bis(2-chloroethyl)carbamate), Estradiol 3-(N,N-bis(2-chloroethyl)carbamate)
  9. Drug

    Estradiol hemisuccinate

    go.drugbank.com/drugs/DB07891
    Experimental

    Synonyms: Estradiol hemisuccinate, 17beta-Estradiol hemisuccinate
  10. Drug

    Estradiol sulfamate

    go.drugbank.com/drugs/DB06597
    Investigational

    Synonyms: Estradiol 3-sulfamate, Estradiol-3-O-SulfamateCategories: Estradiol Congeners