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Displaying results 1 - 10 of 8392 in total
  1. Drug

    Estradiol

    go.drugbank.com/drugs/DB00783
    ApprovedInvestigationalVet approved

    Ethinyl estradiol is different from estradiol due to its higher biovailability and increased resistance to metabolism, rendering it more suitable for oral administration. … Because it has a low oral bioavailability on its own, estradiol is commonly formulated with an ester side-chain.

    Synonyms: Estradiol, 17-β estradiolSalts: Estradiol hemihydrate
  2. Drug

    Estradiol valerate

    go.drugbank.com/drugs/DB13956
    ApprovedInvestigationalVet approved

    [DB00783] is commonly produced with an ester side-chain as endogenous estradiol has very low oral bioavailability on its own (2-10%). … Estradiol valerate is commercially available as an intramuscular injection as the product Delestrogen and is indicated for the treatment of moderate to severe vasomotor symptoms and vulvovaginal atrophy

    Synonyms: Estradiol valerateMixtures: Estradiol Valerate and Estradiol Valerate/Dienogest, Estradiol Valerate and Estradiol Valerate/Dienogest
  3. Drug

    Estradiol benzoate

    go.drugbank.com/drugs/DB13953
    ApprovedVet approvedWithdrawn

    [DB00783] is commonly produced with an ester side-chain as endogenous estradiol has very low oral bioavailability on its own (2-10%). … Following absorption, the esters are cleaved, resulting in the release of endogenous estradiol, or 17β-estradiol.

    Categories: Estradiol Congeners, P-glycoprotein substratesSynonyms: benzoato de estradiol, Estradiol benzoate
  4. Drug

    Estradiol cypionate

    go.drugbank.com/drugs/DB13954
    ApprovedVet approved

    [DB00783] is commonly produced with an ester side-chain as endogenous estradiol has very low oral bioavailability on its own (2-10%). … of hypoestrogenism due to hypogonadism [FDA Label].

    Categories: Estradiol Congeners, P-glycoprotein substratesSynonyms: Estradiol cypionate
  5. Drug

    Estradiol dienanthate

    go.drugbank.com/drugs/DB13955
    ApprovedVet approvedWithdrawn

    Estradiol is commonly produced with an ester side-chain as endogenous estradiol has very low oral bioavailability on its own (2-10%). … Following absorption, the esters are cleaved, resulting in the release of endogenous estradiol, or 17β-estradiol.

    Categories: Estradiol Congeners, Cytochrome P-450 CYP1A1 SubstratesSynonyms: Estradiol dienantate, Estradiol dienanthate
  6. Drug

    Estradiol acetate

    go.drugbank.com/drugs/DB13952
    ApprovedVet approved

    [DB00783] is commonly produced with an ester side-chain as endogenous estradiol has very low oral bioavailability on its own (2-10%). … Estradiol acetate is commercially available as Femring, a vaginal ring used for the treatment of moderate to severe vasomotor symptoms and vulvovaginal atrophy due to menopause.

    Categories: P-glycoprotein substrates, Cytochrome P-450 CYP1A1 SubstratesSynonyms: Estradiol acetate, Estradiol 3-acetate
  7. Drug

    Ethinylestradiol

    go.drugbank.com/drugs/DB00977
    ApprovedInvestigational

    [A191107] These properties were achieved by the substitution of an ethinyl group at carbon 17 of [estradiol].[A191107] Ethinylestradiol soon replaced [mestranol] in contraceptive pills. … [A191107] It was developed in an effort to create an estrogen with greater oral bioavailability.

    Mixtures: TRUST PILL, TRUST PILLCategories: Estradiol Congeners, P-glycoprotein substrates
  8. Drug

    Estramustine

    go.drugbank.com/drugs/DB01196
    ApprovedWithdrawn

    A nitrogen mustard linked to estradiol, usually as phosphate; used to treat prostatic neoplasms; also has radiation protective properties.

    Categories: Estradiol Congeners, Cytochrome P-450 SubstratesSynonyms: 17β-Estradiol 3-(bis(2-chloroethyl)carbamate), Estradiol 3-(N,N-bis(2-chloroethyl)carbamate)
  9. Drug

    Estradiol hemisuccinate

    go.drugbank.com/drugs/DB07891
    Experimental

    Synonyms: Estradiol hemisuccinate, 17beta-Estradiol hemisuccinate
  10. Drug

    Estradiol sulfamate

    go.drugbank.com/drugs/DB06597
    Investigational

    Categories: Estradiol CongenersSynonyms: Estradiol 3-sulfamate, Estradiol-3-O-Sulfamate