Development of a high-affinity ligand that binds irreversibly to Mel1b melatonin receptors.

Article Details

Citation

Witt-Enderby PA, Chu GH, Gillen ML, Li PK

Development of a high-affinity ligand that binds irreversibly to Mel1b melatonin receptors.

J Med Chem. 1997 Dec 19;40(26):4195-8.

PubMed ID
9435890 [ View in PubMed
]
Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
MelatoninMelatonin receptor type 1AKi (nM)0.08N/AN/ADetails
MelatoninMelatonin receptor type 1BKi (nM)0.12N/AN/ADetails