| DB00616 | Candoxatril | experimental | yes | inhibitor | Details |
| DB00886 | Omapatrilat | investigational | yes | | Details |
| DB02062 | N-[3-[(1-Aminoethyl)(Hydroxy)Phosphoryl]-2-(1,1'-Biphenyl-4-Ylmethyl)Propanoyl]Alanine | experimental | unknown | | Details |
| DB02557 | Phosphoramidon | experimental | unknown | inhibitor | Details |
| DB02558 | N-(3-Phenyl-2-Sulfanylpropanoyl)Phenylalanylalanine | experimental | unknown | | Details |
| DB02597 | [2(R,S)-2-Sulfanylheptanoyl]-Phe-Ala | experimental | unknown | | Details |
| DB05796 | Daglutril | investigational | unknown | | Details |
| DB08575 | 2-[(1S)-1-BENZYL-2-SULFANYLETHYL]-1H-IMIDAZO[4,5-C]PYRIDIN-5-IUM | experimental | unknown | | Details |
| DB08626 | Thiorphan | experimental | unknown | inhibitor | Details |
| DB06655 | Liraglutide | approved | unknown | substrate | Details |
| DB09292 | Sacubitril | approved | yes | antagonistinhibitor | Details |
| DB11623 | Candoxatrilat | experimental | yes | inhibitor | Details |
| DB13928 | Semaglutide | approved, investigational | no | substrate | Details |