| DB02378 | MMI-175 | experimental | unknown | | Details |
| DB06073 | CTS-21166 | investigational | yes | inhibitor | Details |
| DB06930 | N-[amino(imino)methyl]-2-(2,5-diphenyl-1H-pyrrol-1-yl)acetamide | experimental | unknown | | Details |
| DB07019 | N-[(5R,14R)-5-AMINO-5,14-DIMETHYL-4-OXO-3-OXA-18-AZATRICYCLO[15.3.1.1~7,11~]DOCOSA-1(21),7(22),8,10,17,19-HEXAEN-19-YL]-N-METHYLMETHANESULFONAMIDE | experimental | unknown | | Details |
| DB07089 | N-[amino(imino)methyl]-2-[2-(2-chlorophenyl)-4-(4-propoxyphenyl)-3-thienyl]acetamide | experimental | unknown | | Details |
| DB07110 | 4-(4-FLUOROBENZYL)PIPERIDINE | experimental | unknown | | Details |
| DB07175 | N-{2-methyl-5-[(6-phenylpyrimidin-4-yl)amino]phenyl}methanesulfonamide | experimental | unknown | | Details |
| DB07206 | 6-[2-(1H-INDOL-6-YL)ETHYL]PYRIDIN-2-AMINE | experimental | unknown | | Details |
| DB07245 | 6-[2-(3'-METHOXYBIPHENYL-3-YL)ETHYL]PYRIDIN-2-AMINE | experimental | unknown | | Details |
| DB07281 | N~3~-BENZYLPYRIDINE-2,3-DIAMINE | experimental | unknown | | Details |
| DB07284 | N~3~-(3-PYRIDIN-3-YLBENZYL)PYRIDINE-2,3-DIAMINE | experimental | unknown | | Details |
| DB07303 | N~3~-[3-(5-METHOXYPYRIDIN-3-YL)BENZYL]PYRIDINE-2,3-DIAMINE | experimental | unknown | | Details |
| DB07345 | 4-(2-aminoethyl)-2-cyclohexylphenol | experimental | unknown | | Details |
| DB07346 | 4-(2-aminoethyl)-2-ethylphenol | experimental | unknown | | Details |
| DB07415 | 4-[(1S)-1-(3-fluoro-4-methoxyphenyl)-2-(2-methoxy-5-nitrophenyl)ethyl]-1H-imidazol-2-amine | experimental | unknown | | Details |
| DB07519 | (6R)-2-amino-6-[2-(3'-methoxybiphenyl-3-yl)ethyl]-3,6-dimethyl-5,6-dihydropyrimidin-4(3H)-one | experimental | unknown | | Details |
| DB07535 | 2-amino-6-[2-(1H-indol-6-yl)ethyl]pyrimidin-4(3H)-one | experimental | unknown | | Details |
| DB07573 | (2S)-1-(2,5-dimethylphenoxy)-3-morpholin-4-ylpropan-2-ol | experimental | unknown | | Details |
| DB07734 | N-(1-benzylpiperidin-4-yl)-4-sulfanylbutanamide | experimental | unknown | | Details |
| DB07735 | N-[1-(2,6-dimethoxybenzyl)piperidin-4-yl]-4-sulfanylbutanamide | experimental | unknown | | Details |
| DB07736 | (2S)-4-(4-fluorobenzyl)-N-(2-sulfanylethyl)piperazine-2-carboxamide | experimental | unknown | | Details |
| DB07737 | (2S)-4-(4-fluorobenzyl)-N-(3-sulfanylpropyl)piperazine-2-carboxamide | experimental | unknown | | Details |
| DB07738 | N-[1-(5-bromo-2,3-dimethoxybenzyl)piperidin-4-yl]-4-sulfanylbutanamide | experimental | unknown | | Details |
| DB07874 | (6S)-2-amino-6-(3'-methoxybiphenyl-3-yl)-3,6-dimethyl-5,6-dihydropyrimidin-4(3H)-one | experimental | unknown | | Details |
| DB07993 | N~3~-[3-(1H-INDOL-6-YL)BENZYL]PYRIDINE-2,3-DIAMINE | experimental | unknown | | Details |
| DB07994 | N~3~-[5-(1H-INDOL-6-YL)-2-(PYRIDIN-2-YLMETHOXY)BENZYL]PYRIDINE-2,3-DIAMINE | experimental | unknown | | Details |
| DB08749 | 3-(2-AMINO-6-BENZOYLQUINAZOLIN-3(4H)-YL)-N-CYCLOHEXYL-N-METHYLPROPANAMIDE | experimental | unknown | | Details |
| DB12285 | Verubecestat | investigational | yes | inhibitor | Details |