| DB02482 | Phosphonothreonine | experimental | unknown | | Details |
| DB05220 | Alisertib | investigational | unknown | inhibitorregulator | Details |
| DB05198 | CYC116 | investigational | unknown | | Details |
| DB05169 | AT9283 | investigational | unknown | | Details |
| DB06134 | SNS-314 | investigational | unknown | | Details |
| DB13061 | MLN8054 | investigational | unknown | | Details |
| DB06347 | Cenisertib | investigational | unknown | | Details |
| DB06486 | Enzastaurin | investigational | unknown | | Details |
| DB07186 | 4-(4-METHYLPIPERAZIN-1-YL)-N-[5-(2-THIENYLACETYL)-1,5-DIHYDROPYRROLO[3,4-C]PYRAZOL-3-YL]BENZAMIDE | experimental | unknown | | Details |
| DB07266 | AKI-001 | experimental | unknown | | Details |
| DB07360 | 1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]urea | experimental | unknown | | Details |
| DB07362 | 1-(5-{2-[(1-methyl-1H-pyrazolo[4,3-d]pyrimidin-7-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]urea | experimental | unknown | | Details |
| DB07545 | N-{3-[(4-{[3-(TRIFLUOROMETHYL)PHENYL]AMINO}PYRIMIDIN-2-YL)AMINO]PHENYL}CYCLOPROPANECARBOXAMIDE | experimental | unknown | | Details |
| DB07801 | N-butyl-3-{[6-(9H-purin-6-ylamino)hexanoyl]amino}benzamide | experimental | unknown | | Details |
| DB08065 | 2-(1H-pyrazol-3-yl)-1H-benzimidazole | experimental | unknown | | Details |
| DB08066 | N-[3-(1H-BENZIMIDAZOL-2-YL)-1H-PYRAZOL-4-YL]BENZAMIDE | experimental | unknown | | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | inhibitor | Details |
| DB12556 | MK-5108 | investigational | unknown | regulator | Details |