| DB01011 | Metyrapone | approved, investigational | unknown | inhibitor | Details |
| DB04630 | Aldosterone | experimental, investigational | unknown | substrate | Details |
| DB00700 | Eplerenone | approved | unknown | inhibitor | Details |
| DB00292 | Etomidate | approved | unknown | inhibitor | Details |
| DB00741 | Hydrocortisone | approved, vet_approved | unknown | substrate | Details |
| DB01388 | Mibefradil | investigational, withdrawn | unknown | inhibitor | Details |
| DB06281 | Torcetrapib | investigational | unknown | inducer | Details |
| DB00421 | Spironolactone | approved | unknown | antagonist | Details |
| DB14539 | Hydrocortisone acetate | approved, vet_approved | unknown | substrate | Details |
| DB14540 | Hydrocortisone butyrate | approved, vet_approved | unknown | substrate | Details |
| DB14543 | Hydrocortisone probutate | approved, vet_approved | unknown | substrate | Details |
| DB14544 | Hydrocortisone valerate | approved, vet_approved | unknown | substrate | Details |
| DB14545 | Hydrocortisone succinate | approved | no | substrate | Details |
| DB11837 | Osilodrostat | approved, investigational | no | inhibitor | Details |
| DB05667 | Levoketoconazole | approved, investigational | yes | inhibitor | Details |