| DB13179 | Troleandomycin | approved | unknown | inducer | Details |
| DB01234 | Dexamethasone | approved, investigational, vet_approved | unknown | inducer | Details |
| DB01058 | Praziquantel | approved, investigational, vet_approved | unknown | substrate | Details |
| DB01045 | Rifampicin | approved | unknown | inducer | Details |
| DB00624 | Testosterone | approved, investigational | unknown | substrate | Details |
| DB09048 | Netupitant | approved, investigational | no | substrate | Details |
| DB09102 | Daclatasvir | approved, investigational | unknown | substrate | Details |
| DB09054 | Idelalisib | approved | no | substrateinhibitor | Details |
| DB06412 | Oxymetholone | approved, illicit | unknown | inhibitor | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | inducer | Details |
| DB11574 | Elbasvir | approved | unknown | substrate | Details |
| DB12332 | Rucaparib | approved, investigational | no | inhibitor | Details |
| DB13943 | Testosterone cypionate | approved | unknown | substrate | Details |
| DB13944 | Testosterone enanthate | approved | unknown | substrate | Details |
| DB13946 | Testosterone undecanoate | approved, investigational | unknown | substrate | Details |
| DB14649 | Dexamethasone acetate | approved, investigational, vet_approved | unknown | inducer | Details |