Nootropic Agents

Name
Nootropic Agents
Accession Number
DBCAT000278
Description

Drugs used to specifically facilitate learning or memory, particularly to prevent the cognitive deficits associated with dementias. These drugs act by a variety of mechanisms. While no potent nootropic drugs have yet been accepted for general use, several are being actively investigated.

Drugs
DrugDrug Description
AcetylcarnitineAn acetylated form of the amino acid derivative L-carnitine that assists in mitochondrial fatty acid metabolism. It is under investigation as a treatment for numerous conditions, including neuropathy, depression, and dementia.
AniracetamA nootropic drug used to ameliorate memory and attention disturbances accompanying cerebrovascular diseases and degenerative brain disorders.
CerebrolysinA proteolytic protein indicated in the treatment of cerebrovascular disorders.
CholineA nutrient found in a wide variety of vitamins including pre-natal formulations.
CiticolineAn endogenous intermediate in the formation of phosphatidylcholine from choline which is thought to have neuroprotective effects.
CutamesineInvestigated for use/treatment in strokes and depression.
DonepezilAn acetylcholinesterase inhibitor used to treat the behavioral and cognitive effects of Alzheimer's Disease and other types of dementia.
Ergoloid mesylateA nootropic with an unknown mechanism of action indicated in individuals over sixty who manifest signs and symptoms of an idiopathic decline in mental capacity.
EtiracetamEtiracetam is under investigation in clinical trial NCT01137110 (Comparison of Short Duration Levetiracetam to Extended Course for Seizure Prophylaxis After Subarachnoid Hemorrhage (SAH)).
GalantamineA cholinesterase inhibitor used to manage mild to moderate dementia associated with Alzheimer's Disease.
Hopantenic acidHopantenic acid (Pantogam) is a central nervous system depressant. Hopantenic acid has a unique spectrum of pharmacological effects (nootropic, anticonvulsant, mild activating) in the absence of addiction, hyperstimulation or withdrawal...
MeclofenoxateNot Annotated
NefiracetamNefiracetam has been used in trials studying the treatment of Alzheimer's Disease.
NicergolineAn ergot derivative use for the treatment of symptoms associated with cerebrovascular abnormalities.
Omega-3-acid ethyl estersA mixture of fatty acids used as an adjunct to diet to reduce triglyceride (TG) levels in adult patients with severe hypertriglyceridemia.
OxiracetamNot Annotated
PiracetamA nootropic cyclic GABA derivative used in myoclonus, sickle cell disease, alcohol dependence, and as a general cognitive enhancer.
TacrineAn anticholinesterase drug used for the management of Alzheimer's disease symptoms.
TaltirelinTaltirelin is a small molecule drug. The usage of the INN stem '-tirelin' in the name indicates that Taltirelin is a thyrotropin releasing hormone analogue. Taltirelin has a monoisotopic molecular...
TilavonemabNot Annotated
VinpocetineA synthetic derivative of a vinca alkaloid used to treat neurological symptoms of cerebrovascular disease.
Drugs & Drug Targets
DrugTargetType
AcetylcarnitineOrganic cation/carnitine transporter 2transporter
AcetylcarnitineSolute carrier family 22 member 21transporter
AcetylcarnitineCarnitine O-acetyltransferaseenzyme
AcetylcarnitineCarnitine O-acetyltransferasetarget
Aniracetam5-hydroxytryptamine receptor 2Atarget
AniracetamD(2) dopamine receptortarget
AniracetamGlutamate receptor 2target
AniracetamGlutamate receptor 3target
CerebrolysinGlycogen synthase kinase-3 betatarget
CerebrolysinCyclin-dependent kinase 5target
CholineCholine transporter-like protein 3transporter
CholineCholine/ethanolamine kinaseenzyme
CholineCholine O-acetyltransferaseenzyme
CholineCholine kinase alphaenzyme
CholineCholine dehydrogenase, mitochondrialenzyme
CholineHigh affinity choline transporter 1transporter
CholineNeuronal acetylcholine receptor subunit alpha-7target
CholineNeuronal acetylcholine receptor subunit alpha-2target
CholineCholine-phosphate cytidylyltransferase Btarget
CholineCholine-phosphate cytidylyltransferase Aenzyme
CholinePhospholipase D1enzyme
CholinePhospholipase D2enzyme
CholineCholinesteraseenzyme
CholinePhosphoethanolamine/phosphocholine phosphataseenzyme
CholineCholine transporter-like protein 2transporter
CholineCholine transporter-like protein 4transporter
CholineCholine transporter-like protein 1transporter
CholineCholine/ethanolaminephosphotransferase 1enzyme
CholineSolute carrier family 22 member 4transporter
CholineOrganic cation/carnitine transporter 2transporter
CholineSolute carrier family 22 member 3transporter
CholineSolute carrier family 22 member 1transporter
CholineSolute carrier family 22 member 2transporter
CholineAcetylcholinesteraseenzyme
CiticolineLicC proteintarget
CutamesineSigma non-opioid intracellular receptor 1target
DonepezilCytochrome P450 2D6enzyme
DonepezilCytochrome P450 2C9enzyme
DonepezilCholinesterasetarget
DonepezilNitric oxide synthase 1target
DonepezilTumor necrosis factor-inducible gene 6 proteintarget
DonepezilInterleukin-1 betatarget
DonepezilNuclear factor NF-kappa-Btarget
DonepezilBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DonepezilNMDA receptortarget
DonepezilCytochrome P450 3A4enzyme
Donepezil5-hydroxytryptamine receptor 2Atarget
DonepezilAcetylcholinesterasetarget
Ergoloid mesylateCytochrome P450 3A4enzyme
Ergoloid mesylateSerotonin Receptorstarget
Ergoloid mesylateBeta adrenergic receptortarget
Ergoloid mesylateAlpha adrenergic receptortarget
Ergoloid mesylateDopamine receptortarget
GalantamineAcetylcholinesterasetarget
GalantamineCytochrome P450 3A4enzyme
GalantamineCytochrome P450 2D6enzyme
GalantamineCholinesterasetarget
GalantamineATP-dependent translocase ABCB1transporter
GalantamineNeuronal acetylcholine receptor subunit alpha-7target
GalantamineMuscle nicotinic acetylcholine receptortarget
Hopantenic acidGABA(A) Receptortarget
NefiracetamProtein kinase Ctarget
NefiracetamNMDA receptortarget
NefiracetamMetabotropic glutamate receptor 5target
NicergolineAlpha-1A adrenergic receptortarget
NicergolineCytochrome P450 2D6enzyme
Omega-3-acid ethyl estersSterol regulatory element-binding protein 1target
Omega-3-acid ethyl estersSterol O-acyltransferase 1enzyme
OxiracetamCholine O-acetyltransferasetarget
TacrineAcetylcholinesterasetarget
TacrineCytochrome P450 1A2enzyme
TacrineCholinesterasetarget
TacrineATP-dependent translocase ABCB1transporter
TacrineLiver carboxylesterase 1target
TaltirelinThyrotropin-releasing hormone receptortarget
TilavonemabMicrotubule-associated protein tautarget
VinpocetineVoltage-dependent calcium channeltarget
VinpocetineSodium channel proteintarget
VinpocetineTranslocator proteintarget
VinpocetineCytochrome P450 3A4enzyme