Name
Amides
Accession Number
DBCAT000494
Description

Organic compounds containing the -CO-NH2 radical. Amides are derived from acids by replacement of -OH by -NH2 or from ammonia by the replacement of H by an acyl group. (From Grant & Hackh's Chemical Dictionary, 5th ed)

Drugs
DrugDrug Description
1-(4-Amidinophenyl)-3-(4-Chlorophenyl)UreaNot Available
2-(4-(2-((3-(5-(PYRIDIN-2-YLTHIO)THIAZOL-2-YL)UREIDO)METHYL)-1H-IMIDAZOL-4-YL)PHENOXY)ACETIC ACIDNot Available
2-[3-(5-Mercapto-[1,3,4]thiadiazol-2-yl)-ureido]-N-methyl-3-phenyl-propionamideNot Available
2-[3-(5-Mercapto-[1,3,4]thiadiazol-2yl)-ureido]-N-methyl-3-pentafluorophenyl-propionamideNot Available
2-chloroethyl-3-sarcosinamide-1-nitrosourea2-chloroethyl-3-sarcosinamide-1-nitrosourea has been used in trials studying the treatment of Colorectal Cancer, Brain and Central Nervous System Tumors, and Unspecified Adult Solid Tumor, Protocol Specific.
3-MethoxybenzamideNot Available
4-(2-AMINOETHYL)BENZENESULFONAMIDENot Available
4-(dimethylamino)-N-[7-(hydroxyamino)-7-oxoheptyl]benzamideNot Available
4-FluorobenzylamineNot Available
7-Aminodesacetoxycephalosporanic acidNot Annotated
AbivertinibAbivertinib is a tyrosine kinase inhibitor targeted against mutant forms of both human epidermal growth factor receptor (EGFR) and Bruton's tyrosine kinase (BTK). It has been investigated for use in...
AbrocitinibA kinase inhibitor used to treat moderate-to-severe atopic dermatitis in adults.
ABSK-091Not Annotated
ABT-072ABT-072 is under investigation in clinical trial NCT00890318 (A Study in Healthy Adult Subjects to Evaluate the Safety, Tolerability, and Pharmacokinetic Profiles of Multiple Doses of ABT-072 Used to Treat...
ABT-102Not Annotated
ABT-639ABT-639 is under investigation in clinical trial NCT01345045 (A Multicenter Study Comparing the Analgesic Effects and Safety of ABT-639 Compared to Placebo in Subjects With Diabetic Neuropathic Pain).
ABT-737An inhibitor of members of the Bcl‑2 family of apoptosis regulators.
ABT-751ABT-751 has been investigated for the treatment of Lung Cancer, Non-Small Cell Lung Cancer, and Non-Small-Cell Lung Cancer.
ABX-196ABX-196 is under investigation in clinical trial NCT03897543 (ABX196 in Combination With Nivolumab in Patients With Hepatocellular Carcinoma).
AcalabrutinibA Bruton tyrosine kinase inhibitor used to treat mantle cell lymphoma, chronic lymphocytic leukemia, and small lymphocytic lymphoma.
AcecarbromalAcecarbromal is a small molecule drug. Acecarbromal has a monoisotopic molecular weight of 278.03 Da.
AcetamideNot Available
AcetaminophenAn analgesic drug used alone or in combination with opioids for pain management, and as an antipyretic agent.
AcetohexamideUsed in the management of diabetes mellitus type 2 (adult-onset).
Acetyl sulfisoxazoleAcute, recurrent or chronic urinary tract infections (primarily pyelonephritis, pyelitis and cystitis) due to susceptible organisms (usually Escherichia coli, Klebsiella-Enterobacter, staphylococcus, Proteus mirabilis and, less frequently, Proteus vulgaris) in the...
AcetyldinalineAcetyldinaline is under investigation in clinical trial NCT00005624 (CI-994 in Treating Patients With Advanced Myeloma).
AcoltremonAcoltremon is under investigation in clinical trial NCT05493111 (A Long-term Safety Study Evaluating the Safety and Systemic Exposure of AR-15512).
AcotiamideAcotiamide has been used in trials studying the treatment of Dyspepsia and Functional Dyspepsia.
AcoziboroleSCYX-7158 has been used in trials studying the treatment of Trypanosomiasis, Parasitic Diseases, Protozoan Infections, and Trypanosomiasis, African.
ACT-451840ACT-451840 has been used in trials studying Malaria.
Actelion-1Investigated for use/treatment in cardiovascular disorders, hypertension, and pulmonary hypertension.
AcumapimodAcumapimod is under investigation in clinical trial NCT02926326 (The Effect of Azithromycin on BCT197 Exposure in Healthy Male Volunteers).
ADL-5859ADL-5859 is under investigation in clinical trial NCT00626275 (Study Evaluating the Analgesic Efficacy and Safety of ADL5859 in Participants With Rheumatoid Arthritis).
AfatinibAn antineoplastic agent used for the treatment of locally advanced or metastatic non-small cell lung cancer (NSCLC) with non-resistant EGFR mutations or resistance to platinum-based chemotherapy.
AgerafenibAgerafenib is under investigation in clinical trial NCT03052569 (Expanded Access to RXDX-105 for Cancers With RET Alterations).
AgomelatineAgomelatine is indicated to treat major depressive episodes in adults.
AllantoinAn ingredient used in skin care products to relieve irritation and protect minor cuts, scrapes, and burns.
AllitinibAllitinib is under investigation in clinical trial NCT04671303 (To Evaluate the Efficacy and Safety of Anlotinib Combined With Allitinib in Lung Cancer).
AlloclamideAlloclamide is a small molecule drug. Alloclamide has a monoisotopic molecular weight of 310.14 Da.
AllylthioureaAllylthiourea is a small molecule drug. Allylthiourea has a monoisotopic molecular weight of 116.04 Da.
AlmonertinibA third-generation, irreversible epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI) indicated for the treatment of patients with metastatic EGFR T790M mutation-positive non-small cell lung cancer (NSCLC).
AlmorexantInvestigated for use/treatment in sleep disorders and insomnia.
AlofanibAlofanib is a small molecule drug. The usage of the INN stem '-anib' in the name indicates that Alofanib is a angiogenesis inhibitor. Alofanib is under investigation in clinical trial...
Alpha-galactosylceramideKRN7000 has been used in trials studying the treatment of Lung Cancer, Chronic Hepatitis C, Hepatitis B, Chronic, Unspecified Adult Solid Tumor, Protocol Specific, and Prevention of GvHD in Patients...
AltiratinibNot Annotated
AlvespimycinInvestigated for use as an antineoplastic agent for solid tumors, advanced solid tumours or acute myeloid leukaemia.
AM-211Not Annotated
AM-461Not Annotated
AmdinocillinUsed in the treatment of urinary tract infections caused by some strains of E. coli and klebsiella and enterobacter species. Used mainly against Gram negative organisms.
AmeltolideAmeltolide is a small molecule drug. Ameltolide has a monoisotopic molecular weight of 240.13 Da.
Aminohippuric acidA hippuric acid derivative injection utilized in the measurement of effective renal plasma flow (ERPF) and functional capacity of the renal excretory system.
AminoquinurideNot Available
AmisulprideA dopamine D2 receptor antagonist used in the treatment of acute and chronic schizophrenia, and in the prevention and treatment of postoperative nausea and vomiting in adults.
AmoxicillinA penicillin derivative used for the treatment of infections caused by gram-positive bacteria, in particular streptococcal bacteria causing upper respiratory tract infections.
AmpicillinA penicillin derivative used for the treatment of a variety of infections caused by gram-positive and gram-negative bacteria as well as some anaerobes.
AmprenavirA protease inhibitor used to treat HIV infection.
AmuvatinibAmuvatinib is a selective multi-targeted tyrosine kinase inhibitor that suppresses c-MET, c-RET and the mutant forms of c-KIT, PDGFR and FLT3. Amuvatinib also suppresses Rad51 protein, a critical component of...
ANC-501ANC-501 is under investigation in clinical trial NCT05439603 (ANC-501 in the Treatment of Adults With Major Depressive Disorder).
AndarineAndarine is a non-steroidal selective androgen receptor modulator.
AndolastAndolast is a small molecule drug. Andolast has a monoisotopic molecular weight of 333.11 Da.
Antineoplaston A10Antineoplaston A10 has been used in trials studying the treatment of Sarcoma, Lymphoma, Lung Cancer, Liver Cancer, and Kidney Cancer, among others.
AP5280Investigated for use/treatment in solid tumors.
ApalcillinApalcillin is a small molecule drug. The usage of the INN stem '-cillin' in the name indicates that Apalcillin is a antibiotic, 6-aminopenicillanic acid derivative. Apalcillin has a monoisotopic molecular...
ApararenoneApararenone is under investigation in clinical trial NCT02531568 (Drug Interaction Study of Warfarin and MT-3995).
APG-1387APG-1387 is under investigation in clinical trial NCT04568265 (A Clinical Study of APG-1387 in Combination With Entecavir in Patients With Chronic Hepatitis B).
ApinocaltamideApinocaltamide is under investigation in clinical trial NCT03239691 (A Study to Evaluate the Effect of ACT-709478 in Photosensitive Epilepsy Patients).
ApricoxibApricoxib has been used in trials studying the treatment and prevention of Lung Cancer, Breast Cancer, Pancreatic Cancer, Non Small Cell Lung Cancer, and Metastatic Pancreatic Cancer, among others.
AprocitentanAn endothelin receptor antagonist used for the treatment of uncontrolled hypertension in patients inadequately controlled on other treatments.
ApronalideApronalide is approved in Japan. Apronalide has been withdrawn from the market in many other countries due to patient development of thrombocytopenic purpura .
AR-12Not Annotated
AR-9281Investigated for use/treatment in hypertension.
AR-AO-14418Not Available
ArgatrobanA synthetic direct thrombin inhibitor used for the prevention and treatment of thrombosis related to heparin use.
ArhalofenateArhalofenate has been investigated for the treatment of Gout and Hyperuricemia.
ArticaineA local anesthetic used for inducing local, infiltrative, or conductive anesthesia in both simple and complex dental procedures.
AsapiprantAsapiprant is a small molecule drug. Asapiprant is under investigation in clinical trial NCT04705597 (Study to Evaluate the Safety, Tolerability, and Efficacy of BGE-175 in Hospitalized Adults With Coronavirus Disease...
AsimadolineInvestigated for use/treatment in irritable bowel syndrome (IBS).
AsivatrepPAC-14028 has been used in trials studying the treatment of Skin Pruritus, Papulopustular Rosacea, and Erythematotelangiectatic Rosacea.
AsnuciclibAsnuciclib is a small molecule drug. The usage of the INN stem '-ciclib' in the name indicates that Asnuciclib is a cyclin dependant kinase inhibitor. Asnuciclib has a monoisotopic molecular...
AspoxicillinNot Annotated
AST-487Not Annotated
AsunaprevirAn NS3 protease inhibitor used to treat hepatitis C genotype 1b.
AsundexianAsundexian is under investigation in clinical trial NCT05686070 (A Study to Test Asundexian for Preventing a Stroke Caused by a Clot in Participants After an Acute Ischemic Stroke or After...
AT9283Investigated for use/treatment in cancer/tumors (unspecified), leukemia (myeloid), and solid tumors.
AtaciguatAtaciguat has been investigated for the basic science of Aortic Valve Stenosis.
AticaprantAticaprant has been used in trials studying the health services research and basic science of Anxiety Disorders and Alcohol Dependence.
AtreleutonAtreleuton has been used in trials studying the treatment of Atherosclerosis and Coronary Artery Disease.
AtuveciclibAtuveciclib is a small molecule drug. The usage of the INN stem '-ciclib' in the name indicates that Atuveciclib is a cyclin dependant kinase inhibitor. Atuveciclib is under investigation in...
AvagacestatAvagacestat has been investigated for the basic science and treatment of Alzheimer Disease.
AvasimibeInvestigated for use/treatment in peripheral vascular disease.
AvitriptanAvitriptan is a small molecule drug. The usage of the INN stem '-triptan' in the name indicates that Avitriptan is a sumatriptan derivative serotonin (5HT1​) receptor agonist. Avitriptan has a...
AVN-944Investigated for use/treatment in cancer/tumors (unspecified), leukemia (unspecified), lymphoma (unspecified), multiple myeloma, and pancreatic cancer.
AvoralstatAvoralstat has been used in trials studying the prevention of HAE and Hereditary Angioedema.
AxelopranAxelopran has been used in trials studying the treatment of OIC and Opioid-induced Constipation.
AxitinibAn oral VEGFR and kinase inhibitor used for the treatment of advanced renal cell carcinoma after failure of one prior systemic therapy.
AZD-1236AZD1236 has been used in trials studying the basic science and treatment of Cystic Fibrosis and Chronic Obstructive Pulmonary Disease.
AZD-4877AZD4877 has been used in trials studying the treatment of NHL, Tumors, Cancer, Lymphoma, and Neoplasms, among others.
AZD-5069Not Annotated
AZD-5423AZD5423 has been used in trials studying the basic science and treatment of Asthma, Bioavailability and AUC, and Chronic Obstructive Pulmonary Disease (COPD).
AZD-5672Azd5672 has been used in trials studying the basic science and treatment of Pharmacokinetics, Renal Impairment, and Rheumatoid Arthritis.
AZD-6703Not Annotated
Azd-7624Not Annotated
AZD-7762AZD7762 has been investigated for the treatment of Cancer, Solid Tumors, and Advanced Solid Malignancies.
AZD-9056AZD9056 has been used in trials studying the basic science and treatment of Rheumatoid Arthritis.
AzidocillinFor treatment of infection (Respiratory, GI, UTI and meningitis) due to E. coli, P. mirabilis, enterococci, Shigella, S. typhosa and other Salmonella, nonpenicillinase-producing N. gononhoeae, H. influenzae, staphylococci, streptococci including...
AzlocillinFor the treatment of infections caused by Pseudomonas aeruginosa, Escherichia coli, and Haemophilus influenzae.
AzosemideAzosemide is a loop diuretic used to treat hypertension, edema, and ascites.
AztreonamA beta-lactam antibiotic used to treat select aztreonam sensitive gram negative bacteria.
BacampicillinAn ampicillin prodrug used to treat various susceptible bacterial infections in the body, such as respiratory infections and skin and subcutaneous tissue infections.
BalicatibBalicatib has been used in trials studying the treatment of Osteoporosis and Knee Osteoarthritis.
BaricitinibA Janus kinase inhibitor used to treat moderate to severe rheumatoid arthritis that has responded poorly to at least one TNF antagonist.
BatabulinBatabulin is under investigation in clinical trial NCT00057382 (T138067 Versus Doxorubicin in Chemotherapy-naive, Unresectable, Hepatocellular Carcinoma Patients).
BavisantBavisant has been used in trials studying the basic science and treatment of Alcoholism, Pharmacokinetics, Drug Interactions, Attention Deficit Hyperactivity Disorder, and Attention Deficit Disorders With Hyperactivity.
BedoradrineInvestigated for use/treatment in asthma and labor and delivery.
BefotertinibBefotertinib is under investigation in clinical trial NCT05007938 (Befotertinib and Icotinib in Treatment-naive Patients With Advanced Egfr-mutant Lung Cancer).
BegacestatBegacestat has been used in trials studying the treatment and basic science of Alzheimer Disease.
BelinostatA histone deacetylase (HDAC) inhibitor used for the treatment of patients with relapsed or refractory peripheral T-cell lymphoma (PTCL).
BelumosudilAn oral inhibitor of rho-associated coiled-coil-containing protein kinases (ROCK) used in the treatment of chronic graft-versus-host disease (GVHD).
BenapenemBenapenem is under investigation in clinical trial NCT04505683 (A Study to Assess Efficacy and Safety Intravenous Benapenem in Patients With Complicated Urinary Tract Infection (Cuti) or Acute Pyelonephritis (AP)).
BenorilateNot Annotated
BenzolamideNot Available
BenzotriptBenzotript is a small molecule drug. Benzotript has a monoisotopic molecular weight of 342.08 Da.
BenzylpenicillinA penicillin used for the treatment of infections caused by gram-positive cocci, in particular streptococcal infections. This form of penicillin is typically used in intravenous or long-acting injectable formulations due to poor oral absorption.
Benzylpenicilloyl polylysineA penicillin derivative used to determine penicillin allergies.
BetrixabanA Factor Xa inhibitor used for prophylaxis of venous thromboembolism in hospitalized patients.
BezafibrateA lipid-lowering fibrate used in the management of primary and secondary hyperlipidaemia, when there is a lack of clinical improvement following lifestyle modifications or correction of the underlying disorder.
BI-671800Bi 671800 has been used in trials studying the treatment of Asthma and Rhinitis, Allergic, Perennial.
BiapenemA carbapenem antibiotic indicated in the treatment of bacterial infections.
BicalutamideAn androgen receptor inhibitor used to treat Stage D2 metastatic carcinoma of the prostate.
BimatoprostA prostaglandin analog used to treat hypotrichosis of the eyelashes and intraocular pressure in open angle glaucoma or ocular hypertension.
BirabresibBirabresib is under investigation in clinical trial NCT02698176 (A Dose Exploration Study With MK-8628 in Participants With Selected Advanced Solid Tumors (MK-8628-006)).
BizelesinBizelesin has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.
BLU-9931Not Annotated
BMS-817399BMS-817399 is under investigation in clinical trial NCT01404585 (Proof-of-Concept Study With BMS-817399 to Treat Moderate to Severe Rheumatoid Arthritis).
BMS-833923Not Annotated
BMS-986141BMS-986141 is under investigation in clinical trial NCT02985632 (A Study to Evaluate the Pharmacokinetics of BMS-986141 in Participants With Hepatic Impairment Compared to Healthy Participants).
BomedemstatNot Annotated
BosentanA dual endothelin receptor antagonist used to treat pulmonary arterial hypertension.
BrinzolamideA carbonic anhydrase inhibitor used for the reduction of elevated intraocular pressure in patients with ocular hypertension or open-angle glaucoma.
BrobactamBrobactam is a small molecule drug. The usage of the INN stem '-bactam' in the name indicates that Brobactam is a ẞ-lactamase inhibitor. Brobactam has a monoisotopic molecular weight of...
BromisovalNot Annotated
BromoprideA substituted benzamide, closely related to metoclopramide, used as an antiemetic.
BrotianideBrotianide is a small molecule drug. Brotianide has a monoisotopic molecular weight of 460.85 Da.
BrovanexineNot Annotated
BuclosamideBuclosamide is a small molecule drug. Buclosamide has a monoisotopic molecular weight of 227.07 Da.
BufexamacAn NSAID used to treat skin conditions like atopic eczema and inflammatory dermatoses.
BuloxibutidNot Annotated
BumetanideA sulfamyl diuretic used to treat edema in congestive heart failure, hepatic and renal disease, and nephrotic syndrome.
BupivacaineA local anesthetic used in a wide variety of superficial and invasive procedures.
ButanilicaineNot Annotated
CabozantinibA tyrosine kinase inhibitor used to treat advanced renal cell carcinoma, hepatocellular carcinoma, and medullary thyroid cancer.
CapmatinibA kinase inhibitor targeting c-Met receptor tyrosine kinase in the treatment of non-small cell lung cancer with MET exon 14 skipping.
CapsaicinA topical analgesic agent used for the symptomatic relief of neuropathic pain associated with post-herpetic neuralgia, as well as other muscle and joint pain.
CaracemideCaracemide is a small molecule drug. Caracemide has a monoisotopic molecular weight of 189.07 Da.
Carbamide peroxideA medication used to loosen ear wax, whiten teeth, and clean oral wounds.
CarbapenemNot Annotated
Carbaspirin calciumAn NSAID indicated in the treatment of short term pain and fever.
CarbenicillinFor the treatment of acute and chronic infections of the upper and lower urinary tract and in asymptomatic bacteriuria due to susceptible strains of bacteria.
CarboxinA systemic agricultural fungicide and seed treatment agent.
CarbromalNot Annotated
CarbutamideNot Annotated
CarfecillinNot Annotated
CarindacillinA penicillin antibiotic used to treat a variety of infections, but is no longer marketed in the USA.
CarmustineAn alkylating agent used in the treatment of various malignancies, including brain tumours and multiple myeloma, among others.
CaroxazoneFor the treatment of depression.
CarumonamNot Annotated
CasopitantInvestigated for use/treatment in urinary incontinence and adverse effects (chemotherapy).
CE-224535CE-224535 has been used in trials studying the treatment of Osteoarthritis.
CefacetrileA broad-spectrum first-generation cephalosporin used for the treatment of susceptible bacterial infections.
CefaclorA second generation cephalosporin used to treat a wide variety of infections in the body.
CefadroxilA cephalosporin antibiotic used in the treatment of various bacterial infections, such as urinary tract infections, skin and skin structure infections, and tonsillitis.
CefaloniumNot Annotated
CefaloridineCephaloridine or cefaloridine is a first generation semisynthetic cephalosporin. It is derived from cephalosporin C and is a zwitterion at physiological pH.
CefalotinA broad-spectrum cephalosporin antibiotic used for the treatment of serious bacterial infections in various locations, such as the urinary tract, skin, bone, and lower respiratory tract.
CefamandoleA beta-lactam antibiotic used in the treatment of various infections caused by susceptible strains of bacteria, such as lower respiratory infections, urinary tract infections, skin infections, and bone and joint infections.
Cefamandole nafateA second generation cephalosporin indicated in the prevention of infections during surgery.
CefapirinA first generation cephalosporin indicated in the treatment of susceptible bacterial infections.
CefatrizineNot Annotated
CefazedoneNot Annotated
CefazolinA broad-spectrum cephalosporin antibiotic mainly used for the treatment of skin bacterial infections and other moderate to severe bacterial infections in the lung, bone, joint, stomach, blood, heart valve, and urinary tract.
CefbuperazoneNot Annotated
CefcanelCefcanel is a small molecule drug. Cefcanel has a monoisotopic molecular weight of 478.04 Da.
Cefcanel daloxateCefcanel daloxate is a small molecule drug. Cefcanel daloxate has a monoisotopic molecular weight of 661.1 Da.
CefclidinCefclidin is a small molecule drug. Cefclidin has a monoisotopic molecular weight of 550.14 Da.
CefditorenA broad-spectrum third-generation cephalosporin antibiotic typically used to treat bacterial infections of the skin and respiratory tract.
CefepimeA fourth-generation cephalosporin antibiotic used in the treatment of infections caused by susceptible bacteria, such as pneumonia, urinary tract infections, and skin infections.
CefetametNot Annotated
Cefetamet pivoxilCefetamet pivoxil is under investigation in clinical trial NCT04664803 (Safety and Efficacy of Cefecin Tab. in Patients With Acute Sinusitis).
CefiderocolA cephalosporin antibiotic used in complicated urinary tract infections.
CefilavancinInvestigated for use/treatment in bacterial infection, skin infections/disorders, and staph bacterial infections.
CefiximeA third generation cephalosporin used to treat susceptible Gram-negative and Gram-positive bacterial infections.
CefmatilenCefmatilen is a small molecule drug. Cefmatilen has a monoisotopic molecular weight of 514.0 Da.
CefmenoximeUsed to treat female gynecologic and obstetric infections caused by susceptible aerobic (including the gonococcus) and anaerobic bacteria.
CefmetazoleA cephalosporin antibiotic used to treat a variety of bacterial infections.
CefminoxCefminox (INN) is a second generation cephalosporin antibiotic. It is approved for use in Japan.
CefodizimeA broad-spectrum, third-generation cephalosporin used to treat serious infections caused by susceptible bacteria.
CefonicidFor the treatment of bacterial infections caused by susceptible microorganisms.
CefoperazoneA broad-spectrum cephalosporin antibiotic used for the treatment of bacterial infections in various locations, including the respiratory tract, abdomen, skin, and female genital tracts.
CeforanideFor the treatment of infections caused by susceptible organisms.
CefoselisCefoselis is a small molecule drug. Cefoselis has a monoisotopic molecular weight of 522.11 Da.
CefotaximeA third generation cephalosporin used to treat susceptible Gram negative and Gram positive bacterial infections.
CefotetanAn antibiotic medication used for the prophylaxis and treatment of various bacterial infections, including urinary tract infections, bone and joint infection, and lower respiratory tract infections.
CefotiamA cephalosporin antibiotic used to treat a variety of bacterial infections.
CefovecinCefovecin is a cephalosporin antibiotic used for the treatment of skin infections in cats and dogs. It is the first single-dose injectable antibiotic for dogs and cats that assures owner...
CefoxitinA semi-synthetic, broad-spectrum antibiotic for parenteral administration used for the treatment of serious bacterial infections, such as urinary tract infection, blood infection, bone and joint infection, and lower respiratory tract infection.
CefozopranNot Annotated
CefpimizoleCefpimizole is a small molecule drug. Cefpimizole has a monoisotopic molecular weight of 670.12 Da.
CefpiramideFor treatment of severe infections caused by susceptible bacteria such as P. aeruginosa.
CefpiromeAn antibiotic indicated in the treatment of a wide variety of infections in the body.
CefpodoximeA third-generation cephalosporin antibiotic used in the treatment of various bacterial infections, including gonorrhea, community acquired pneumonia, and sinusitis.
CefprozilA cephalosporin antibiotic used in the treatment of various bacterial infections, such as pharyngitis, tonsillitis, otitis media, and uncomplicated skin infections.
CefradineA first-generation cephalosporin antibiotic used in the treatment of bacterial infections of the respiratory and urinary tracts and of the skin and soft tissues.
CefroxadineWas used for the treatment of bacterial infections.
CefsulodinNot Annotated
CefsumideCefsumide is a small molecule drug. Cefsumide has a monoisotopic molecular weight of 440.08 Da.
Ceftaroline fosamilAn antibacterial agent used to treat various bacterial infections, such as acute bacterial skin and skin structure infections and community-acquired bacterial pneumonia.
CeftazidimeAn injected broad-spectrum third-generation cephalosporin beta-lactam antibiotic used to treat or prevent a variety of bacterial infections, including pneumonia, gynecological infections, bone and joint infections, and septicemia, among others.
CeftezoleNot Annotated
CeftibutenA third-generation cephalosporin antibiotic commonly used in the treatment of acute bacterial exacerbations of chronic bronchitis (ABECB), acute bacterial otitis media, pharyngitis, and tonsillitis.
CeftiofurCeftiofur is a third generation cephalosporin antibiotic, first described in 1987, and now used in veterinary medicine. It is marketed by pharmaceutical company Zoetis as Excenel, and is the active...
CeftizoximeA third-generation cephalosporin antibiotic used in the treatment of various bacterial infections, including lower respiratory tract infection, urinary tract infection, and gonorrhea.
CeftobiproleA broad spectrum 5th-generation cephalosporin antibacterial indicated for certain kinds of pneumonia, bacteremia, and skin and skin structure infections, including those caused by MRSA.
Ceftobiprole medocarilA broad spectrum 5th-generation cephalosporin antibacterial indicated for certain kinds of pneumonia, bacteremia, and skin and skin structure infections, including those caused by MRSA.
CeftolozaneA cephalosporin antibiotic used to treat complicated intra-abdominal infections in combination with metronidazole, complicated urinary tract infections, and hospital-acquired pneumonia.
CeftriaxoneA broad-spectrum cephalosporin antibiotic used for the treatment of bacterial infections in various locations, such as in the respiratory tract, skin, soft tissue, and urinary tract.
CefuroximeA cephalosporin indicated for the treatment of a variety of infections including acute bacterial otitis media, several upper respiratory tract infections, skin infections, urinary tract infections, gonorrhea, early Lyme disease, and impetigo.
CefuzonamCefuzonam is a small molecule drug. Cefuzonam has a monoisotopic molecular weight of 513.0 Da.
CelecoxibAn NSAID used to treat osteoarthritis, rheumatoid arthritis, acute pain, menstrual symptoms, and to reduce polyps is familial adenomatous polyposis.
CeliprololA beta-blocker for the management of hypertension and angina pectoris.
CEP-37440CEP-37440 has been used in trials studying the treatment of Solid Tumors.
CephalexinA first generation cephalosporin used to treat certain susceptible bacterial infections.
CephaloglycinFor treatment of severe infections caused by susceptible bacteria.
Cephalosporin CNot Available
CeralasertibCeralasertib is under investigation in clinical trial NCT03682289 (Phase II Trial of AZD6738 Alone and in Combination With Olaparib).
Ceramide APNot Annotated
Ceramide NGNot Annotated
CeruleninFor use as a biochemical tool, Cerulenin is shown to cause dramatic weight loss in animals
CGI-1842JI-101 has been used in trials studying the treatment of Cancer, Colon Cancer, Neuroendocrine, Ovarian Cancer, and Advanced Solid Tumors.
CGS-27023Not Available
CH-5132799CH5132799 has been used in trials studying the treatment of Solid Tumors.
ChlorpropamideA sulfonylurea used in the treatment of non insulin dependent diabetes mellitus.
ChlorsulfaquinoxalineChlorsulfaquinoxaline has been used in trials studying the treatment of Lung Cancer and Colorectal Cancer.
ChlorthalidoneA diuretic used to treat hypertension or edema caused by heart failure, renal failure, hepatic cirrhosis, estrogen therapy, and other conditions.
CI-1040CI-1040 has been used in trials studying the treatment of Lung Cancer, Breast Cancer, Breast Neoplasms, Pancreatic Cancer, and Colorectal Cancer, among others.
CimicoxibInvestigated for use/treatment in depression.
CinchocaineAn anesthetic used for local or regional anesthesia.
CinitaprideA benzamide with gastroprokinetic and antiemetic properties typically used for the treatment of gastrointestinal motility disorders such as gastroesophageal reflux disease (GERD), non-ulcer dyspepsia, and delayed gastric emptying.
CisaprideA medication used to treat heartburn associated with GERD.
Clamidoxic acidClamidoxic acid is a small molecule drug. Clamidoxic acid has a monoisotopic molecular weight of 339.01 Da.
ClamikalantClamikalant is a small molecule drug. The usage of the INN stem '-kalant' in the name indicates that Clamikalant is a potassium channel blocker. Clamikalant has a monoisotopic molecular weight...
ClanfenurClanfenur is a small molecule drug. Clanfenur has a monoisotopic molecular weight of 335.08 Da.
ClazosentanInvestigated for use/treatment in strokes.
CleboprideA dopamine antagonist used to treat symptoms associated with functional gastrointestinal disorders. Clebopride may also be used to treat nausea and vomiting associated with chemotherapy.
ClefamideNot Annotated
ClioxanideClioxanide is a small molecule drug. Clioxanide has a monoisotopic molecular weight of 540.84 Da.
CloflucarbanCloflucarban is a small molecule drug. Cloflucarban has a monoisotopic molecular weight of 348.0 Da.
ClofutribenClofutriben is a small molecule drug. Clofutriben is under investigation in clinical trial NCT05307328 (SPI-62 as a Treatment for Adrenocorticotropic Hormone-dependent Cushing's Syndrome). Clofutriben has a monoisotopic molecular weight of...
CloguanamilCloguanamil is a small molecule drug. Cloguanamil has a monoisotopic molecular weight of 237.04 Da.
ClopamideClopamide is an oral diuretic agent with antihypertensive activity. Like thiazide diuretics, it has an aromatic sulfonamide base but with no double-ring structure.
ClorexoloneNot Annotated
ClorsulonNot Annotated
CloxaceprideCloxacepride is a small molecule drug. The usage of the INN stem '-pride' in the name indicates that Cloxacepride is a sulpiride derivative and analogue. Cloxacepride has a monoisotopic molecular...
CloxacillinAn antibiotic agent used for the treatment of beta-hemolytic streptococcal and pneumococcal infections as well as staphylococcal infections.
CM4620CM4620 (Zegocractin), is under investigation in multiple clinical trials, including NCT04195347 (pancreatitis due to asparaginase), NCT03709342 (PK/PD study in acute pancreatitis), NCT03401190 and NCT04681066 (pancreatitis and SIRS), and NCT04661540 (critical...
CoelenteramideNot Available
ConteltinibConteltinib is a small molecule drug. The usage of the INN stem '-tinib' in the name indicates that Conteltinib is a tyrosine kinase inhibitor. Conteltinib is under investigation in clinical...
CP-547632CP-547632 has been used in trials studying the treatment of Ovarian Cancer, Lung Neoplasms, Ovarian Neoplasms, Peritoneal Neoplasms, and Fallopian Tube Cancer, among others.
CP-778875CP-778875 is under investigation in clinical trial NCT00326326 (Effect of CP-778,875 on HDL-C in Subjects With Abnormal Lipid Levels and Type 2 Diabetes.).
CresotamideCresotamide is a small molecule drug. Cresotamide has a monoisotopic molecular weight of 151.06 Da.
CyclacillinFor the treatment of bacterial infections caused by susceptible organisms.
CyclohexylformamideNot Available
DA-6886DA-6886 has been used in trials studying the treatment of Irritable Bowel Syndrome.
DabuzalgronDabuzalgron is a small molecule drug. Dabuzalgron has a monoisotopic molecular weight of 317.06 Da.
DagrocoratNot Annotated
DaltrobanDaltroban is a small molecule drug. Daltroban has a monoisotopic molecular weight of 353.05 Da.
DanavorextonNot Annotated
DanegaptideDanegaptide has been investigated for the treatment of Focus of Study is STEMI.
DanoprevirDanoprevir has been used in trials studying the treatment of Hepatitis C, Chronic.
DanusertibDanusertib has been used in trials studying the treatment of Leukemia.
DaporinadDaporinad has been used in trials studying the treatment of Melanoma, Cutaneous T-cell Lymphoma, and B-cell Chronic Lymphocytic Leukemia.
DarexabanDarexaban has been used in trials studying the prevention and basic science of Japanese, Caucasian, Thromboembolism, Pharmacodynamics, and Pharmacokinetics, among others.
DarunavirA HIV protease inhibitor used in the treatment of human immunodeficiency virus (HIV) infection in patients with history of prior antiretroviral therapies.
DasabuvirA direct-acting antiviral agent used to treat specific hepatitis C virus (HCV) infections in combination with other antiviral agents.
DazoprideDazopride is a small molecule drug. The usage of the INN stem '-pride' in the name indicates that Dazopride is a sulpiride derivative and analogue. Dazopride has a monoisotopic molecular...
Deacetoxycephalosporin CNot Available
DeclopramideInvestigated for use/treatment in colorectal cancer and inflammatory bowel disease.
DefactinibAn inhibitor of FAK used alongside a MEK1/RAF inhibitor for the treatment of recurrent low-grade serous ovarian cancer.
DeracoxibDeracoxib is a non-steroidal anti-inflammatory drug of the coxib class, used in veterinary medicine to treat osteoarthritis in dogs. It is sold in tablets, which have added beefy flavour to...
DiacetamateDiacetamate is a small molecule drug. Diacetamate has a monoisotopic molecular weight of 193.07 Da.
DiamfenetideDiamfenetide is a small molecule drug. Diamfenetide has a monoisotopic molecular weight of 372.17 Da.
DiapamideDiapamide is a small molecule drug. Diapamide has a monoisotopic molecular weight of 262.02 Da.
DiazolidinylureaAn ingredient used in hospitals for disinfection.
DibromsalanDibromsalan is a small molecule drug. Dibromsalan has a monoisotopic molecular weight of 368.9 Da.
DiclofenamideA carbonic anhydrase inhibitor used for the management of open-angle and secondary glaucoma, as well as acute angle-closure glaucoma in delayed pre-operative setting requiring a reduction in intraocular pressure.
DicloxacillinA penicillin used to treat penicillinase-producing bacterial infections that are susceptible to the drug.
DiethyltoluamideAn insect repellant, also known as DEET.
DiethyltryptamineDiethyltryptamine (DET) is an orally active hallucinogenic agent and a substituted form of tryptamine.
DifamilastA phosphodiesterase-4 inhibitor used for the treatment of atopic dermatitis.
DifenpiramideNot Annotated
DihydrocapsiateDihydrocapsiate is under investigation in clinical trial NCT00999297 (Effect of 4-week Dihydrocapsiate Ingestion on Resting Metabolic Rate).
DNK-333Not Annotated
DobuprideDobupride is a small molecule drug. The usage of the INN stem '-pride' in the name indicates that Dobupride is a sulpiride derivative and analogue. Dobupride has a monoisotopic molecular...
DofetilideA class III antiarrhythmic drug used for the maintenance of normal sinus rhythm and cardioversion in cases of atrial fibrillation and atrial flutter.
DomatinostatNot Annotated
DONUDonu has been used in trials studying the treatment of Psychosis.
DoramapimodDoramapimod is a P38 MAP kinase inhibitor.
DoripenemAn antibiotic of the penem class used to treat complicated intra-abdominal and urinary tract infections.
DorzolamideA carbonic anhydrase inhibitor used to treat high intraocular pressure in ocular hypertension and open angle glaucoma.
DrinabantInvestigated for use/treatment in alzheimer's disease, obesity, and schizophrenia and schizoaffective disorders.
DubermatinibDubermatinib is under investigation in clinical trial NCT03572634 (Phase 1/2 Study of TP-0903 (an Inhibitor of AXL Kinase) in Patients With Previously Treated CLL).
DulozafoneDulozafone is a small molecule drug. The usage of the INN stem '-zafone' in the name indicates that Dulozafone is a alozafone derivative. Dulozafone has a monoisotopic molecular weight of...
E-7820E7820 has been investigated for the treatment of Colon Cancer and Rectal Cancer.
EcabapideEcabapide is a small molecule drug. Ecabapide has a monoisotopic molecular weight of 371.18 Da.
EcomustineEcomustine is a small molecule drug. The usage of the INN stem '-mustine' in the name indicates that Ecomustine is a antineoplastic, alkylating agent, (β-chloroethyl) amine derivative. Ecomustine has a...
EcopladibEcopladib is a small molecule drug. The usage of the INN stem '-pladib' in the name indicates that Ecopladib is a phospholipase A2​ inhibitor. Ecopladib has a monoisotopic molecular weight...
EdasalonexentEdasalonexent is under investigation in clinical trial NCT01511900 (A Multiple Ascending Dose Study of CAT-1004 in Patients With Type 2 Diabetes).
Edonentan anhydrousEdonentan anhydrous is a small molecule drug. The usage of the INN stem '-entan' in the name indicates that Edonentan anhydrous is a endothelin receptor antagonist. Edonentan anhydrous has a...
EflucimibeEflucimibe is a small molecule drug. Eflucimibe has a monoisotopic molecular weight of 469.3 Da.
ElesclomolInvestigated for use/treatment in melanoma.
ElinogrelInvestigated for use/treatment in cardiovascular disorders and myocardial infarction.
ElmustineElmustine is a small molecule drug. The usage of the INN stem '-mustine' in the name indicates that Elmustine is a antineoplastic, alkylating agent, (β-chloroethyl) amine derivative. Elmustine has a...
ElsulfavirineElsulfavirine is under investigation in clinical trial NCT03706898 (Study to Evaluate the Safety and PK of Elpida® in Healthy Subjects and Patients With Hepatic Impairment and to Assess the Impact...
ElubrixinElubrixin has been used in trials studying the treatment of Cystic Fibrosis, Colitis, Ulcerative, and Chronic Obstructive Pulmonary Disease (COPD).
EncainideA voltage-gated sodium channel blocker used for management of atrial or ventricular fibrillation, atrial flutter, and ventricular tachycardia, that is no longer used due to proarrhythmic adverse effects.
EncorafenibA kinase inhibitor used to treat unresectable or metastatic melanoma with BRAF mutations.
EnobosarmEnobosarm has been used in trials studying the treatment of Stress Urinary Incontinence and Triple Negative Breast Cancer.
EntinostatEntinostat is under investigation for the treatment and other of Volunteers, Breast Cancer, Human Volunteers, and Normal Volunteers. Entinostat has been investigated for the treatment of Non-Small Lung Cancer, Epigenetic...
EntrectinibEntrectinib is indicated for the treatment of metastatic ROS1-positive non-small cell lung cancer in adults. Entrectinib is also indicated in adults and children over 12 years old for the treatment...
EnviroximeEnviroxime is a small molecule drug. Enviroxime has a monoisotopic molecular weight of 358.11 Da.
EnzalutamideA second-generation androgen receptor inhibitor used to treat castration-resistant prostate cancer and metastatic castration-sensitive prostate cancer.
Enzalutamide d3Enzalutamide d3 is under investigation in clinical trial NCT03850795 (HC-1119 Versus Enzalutamide in Metastatic Castration-resistant Prostate Cancer (Mcrpc)).
EpacadostatEpacadostat has been used in trials studying the treatment of HL, Melanoma, Glioblastoma, Mucosal Melanoma, and Ovarian Carcinoma, among others.
EpanololEpanolol is an beta blocker.
EperezolidEperezolid is a small molecule drug. The usage of the INN stem '-zolid' in the name indicates that Eperezolid is a oxazolidinone antibacterial. Eperezolid has a monoisotopic molecular weight of...
EpicillinNot Annotated
EprotiromeInvestigated for use/treatment in hyperlipidemia, metabolic disease, and obesity.
EragidomideEragidomide is under investigation in clinical trial NCT04297124 (A Study to Evaluate the Metabolism and Excretion of [14C]-CC-90009 in Healthy Male Subjects).
ErtapenemA carbapenem antibiotic used for the treatment of moderate to severe infections caused by susceptible bacteria.
Estradiol sulfamateInvestigated for use/treatment in endometriosis.
EtamivanEtamivan (INN) or ethamivan (USAN) is marketed under the name Analepticon. Etamvin is a respiratory stimulant drug similar to nikethamide. It is no longer used in the United States.
EtersalateEtersalate is a small molecule drug. Etersalate has a monoisotopic molecular weight of 357.12 Da.
EthenzamideNot Annotated
EthoxzolamideFor use in the treatment of duodenal ulcers, as a diuretic, and in the treatment of glaucoma, and may also be useful in the treatment of seizures associated with epilepsy.
EticloprideNot Annotated
EtidocaineEtidocaine is marketed under the name Duranest. It is an injectable local anesthetic during surgery, labor, and delivery. Etidocaine has a long duration of activity, but has the main disadvantage...
EtiracetamEtiracetam is under investigation in clinical trial NCT01137110 (Comparison of Short Duration Levetiracetam to Extended Course for Seizure Prophylaxis After Subarachnoid Hemorrhage (SAH)).
EtofamideEtofamide is used as an antiamoebic agent. Etofamide, under the brand name Kitnos, was marketed in Brazil by Pfizer but has been discontinued .
EVT 302Investigated for use/treatment in smoking cessation.
ExalamideExalamide is a small molecule drug. Exalamide has a monoisotopic molecular weight of 221.14 Da.
FallyprideFallypride is under investigation in clinical trial NCT02310360 (Striatal and Extra-striatal Dopamine Release in Response to Food in Healthy Humans).
FaropenemFaropenem has been used in trials studying the treatment of Tuberculosis, Pulmonary Tuberculosis, and Community Acquired Pneumonia.
Faropenem medoxomilInvestigated for use/treatment in bacterial infection, bronchitis, otitis media, and pediatric indications.
FasentinNot Annotated
FasitibantFasitibant is under investigation in clinical trial NCT02205814 (Fasitibant Intra-articular Injection in Patients With Symptomatic Osteoarthritis of the Knee).
FedratinibFedratinib is indicated for the treatment of adult patients with intermediate-2 or high-risk primary or secondary (post-polycythemia vera or post-essential thrombocythemia) myelofibrosis.
FigopitantFigopitant is under investigation in clinical trial NCT02209714 (Safety, Tolerability and Pharmacodynamics After Oral Administration of BIIF 1149 BS in Healthy Male Volunteers).
FipaxalparantNot Annotated
FiruglipelFiruglipel is a small molecule drug. Firuglipel is under investigation in clinical trial NCT02647320 (12-Week Study of DS-8500a in Subjects With Type 2 Diabetes Mellitus on Metformin). Firuglipel has a...
FK-960Investigated for use/treatment in dementia, alzheimer's disease, schizophrenia and schizoaffective disorders, and memory loss.
FlomoxefFlomoxef has been used in trials studying the treatment of Urinary Tract Infection.
FlorasulamFlorasulam is under investigation in clinical trial NCT01193465 (Temperature and Humidity Among Different Anesthesia Work-station).
Flotufolastat F-18A radiopharmaceutical diagnostic agent used in PET imaging to visualize PSMA-positive lesions in men with prostate cancer with suspected metastasis or recurrence.
FluazuronFluazuron is a benzoyl phenylurea compound.
FlucloxacillinA narrow spectrum penicillin antibiotic that exerts specific activity against Gram positive organisms in skin and soft tissue infections, except those caused by methicillin resistant staphylococcus aureus (MRSA).
FlufenoxuronFlufenoxuron is under investigation in clinical trial NCT00922870 (Evaluation of Hemodynamic Effects of Cascade Hemofiltration in Septic Shock).
FlumatinibFlumatinib has been used in trials studying the treatment of Myelogenous Leukemia, Chronic.
FlurofamideFlurofamide is a small molecule drug. Flurofamide has a monoisotopic molecular weight of 217.04 Da.
FlutamideAn antiandrogen used for locally confined stage B2-C and D-2 metastatic prostate carcinoma.
FomidacillinFomidacillin is a small molecule drug. The usage of the INN stem '-cillin' in the name indicates that Fomidacillin is a antibiotic, 6-aminopenicillanic acid derivative. Fomidacillin has a monoisotopic molecular...
ForetinibForetinib has been used in trials studying the treatment of Cancer, Breast Cancer, Carcinoma, Renal Cell, Recurrent Breast Cancer, and Neoplasms, Head and Neck, among others. Foretinib is an orally...
FosamprenavirAn antiretroviral agent used for the treatment and postexposure prophylaxis of human immunodeficiency virus (HIV-1) infection.
FosdagrocoratFosdagrocorat has been used in trials studying the treatment and basic science of Rheumatoid Arthritis.
FotemustineAn alkylating agent used in the treatment of metastatic melanoma.
FrentizoleFrentizole is a small molecule drug. Frentizole has a monoisotopic molecular weight of 299.07 Da.
FrunexianNot Available
FurosemideA loop diuretic used to treat hypertension and edema in congestive heart failure, liver cirrhosis, renal disease, and hypertension.
FuzlocillinFuzlocillin is a small molecule drug. The usage of the INN stem '-cillin' in the name indicates that Fuzlocillin is a antibiotic, 6-aminopenicillanic acid derivative. Fuzlocillin has a monoisotopic molecular...
GC-373GC-373 is a peptide aldehyde which is metabolized from the bisulfide adduct, GC-376 free acid . It is an inhibitor of Mpro (otherwise known as 3CLpro), a viral encoded protease...
GC-376 free acidGC-376 is a 3C-like protease (3CLpro or Mpro) inhibitor that stops the cleavage and activation of functional viral proteins required for replication and transcription in host cells . The compound...
GDC-0349GDC-0349 has been used in trials studying the treatment of Non-Hodgkin's Lymphoma, Solid Tumor.
GefapixantA P2X3 receptor antagonist that reduces the cough reflex in patients with refractory or unexplained chronic cough.
GeldanamycinNot Available
GiripladibGiripladib is under investigation in clinical trial NCT00396955 (A Study Comparing 4 Dose Regimens of PLA-695, Naproxen, and Placebo In Subjects With Osteoarthritis Of The Knee).
GisadenafilGisadenafil has been investigated for the treatment of Prostatic Hyperplasia.
GlasdegibA sonic hedgehog receptor inhibitor used to treat newly diagnosed acute myeloid leukemia in patients over 75 years who cannot receive intense chemotherapy.
GlecaprevirA Hepatitis C NS3/4A protease inhibitor used to treat Hepatitis C.
GlesatinibInvestigated for use/treatment in cancer/tumors (unspecified).
GlibornurideGlibornuride is a sulfonylurea-type anti-diabetic drug.
GlicaramideGlicaramide is a small molecule drug. Glicaramide has a monoisotopic molecular weight of 598.29 Da.
GliclazideA sulfonylurea used to treat hyperglycemia in patients with type 2 diabetes mellitus.
GliflumideGliflumide is a small molecule drug. Gliflumide has a monoisotopic molecular weight of 500.19 Da.
GlimepirideA sulfonylurea drug used to treat type 2 diabetes mellitus.
GliquidoneA sulfonylurea drug used in the management of diabetes mellitus type 2.
GlisentideGlisentide is a small molecule drug. Glisentide has a monoisotopic molecular weight of 445.17 Da.
GlisolamideGlisolamide is a small molecule drug. Glisolamide has a monoisotopic molecular weight of 434.16 Da.
GlisoxepideFor the treatment of diabetes mellitus type 2.
GLPG-0187GLPG0187 has been used in trials studying the treatment of Solid Tumors.
GlyburideA sulfonylurea used in the treatment of non insulin dependent diabetes mellitus.
GlybuzoleGlybuzole is a small molecule drug. Glybuzole has a monoisotopic molecular weight of 297.06 Da.
GlyclopyramideGlyclopyramide is a small molecule drug. Glyclopyramide has a monoisotopic molecular weight of 303.04 Da.
GlymidineGlycodiazine is used concomitantly with insulin for the treatment of noninsulin-dependent (type 2) diabetes mellitus.
GranotapideGranotapide has been used in trials studying the treatment of Type II Diabetes Mellitus.
GrapiprantThe effects of grapiprant have been investigated in the area of analgesia and anti-inflammation due to the effects that have been reported about this molecule. This molecule has been approved...
GrazoprevirAn antiviral and NS3/4A protease inhibitor used to treat hepatitis C infections.
GSK-2981278GSK-2981278 is under investigation in clinical trial NCT03004846 (A Study of GSK2981278 Ointment in Subjects With Plaque Psoriasis).
GSK-424887Gsk424887 has been used in trials studying the basic science and treatment of Depressive Disorder and Anxiety Disorder.
GTX-758GTX-758 is under investigation in clinical trial NCT01420861 (GTx-758 on Serum Prostate-specific Antigen (PSA) in Men With Castrate Resistant Prostate Cancer).
GW-813893Not Available
H-89Not Available
HetacillinHetacillin is a beta-lactam antibiotic prodrug used to treat bacterial infections. In the body it gets converted to ampicillin.
Hippuric acidNot Annotated
HMN-214Not Annotated
HQP1351HQP1351 is under investigation in clinical trial NCT03883100 (A Pivotal Study of HQP1351 in Patients of Chronic Myeloid Leukemia in Accelerated Phase With T315I Mutation).
HydrochlorothiazideA thiazide diuretic used to treat edema associated with a number of conditions, and hypertension.
HydroflumethiazideA thiazide diuretic used to treat hypertension as well as edema due to congestive heart failure and liver cirrhosis.
HydroxyureaAn antimetabolite used to treat sickle cell anemia crisis, resistant chronic myeloid leukemia, and Locally advanced squamous cell carcinomas of the head and neck (excluding the lip).
IbipinabantIbipinabant has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.
IbrigamparInvestigated for use/treatment in diabetes mellitus type 2.
IbrolipimIbrolipim is a small molecule drug. Ibrolipim has a monoisotopic molecular weight of 450.03 Da.
IbuproxamIbuproxam is a non steroidal anti-inflammatory drug (NSAID).
IbutilideA class III antiarrhythmic agent used to correct atrial fibrillation and atrial flutter, which can be considered as an alternative to cardioversion.
ICI-164384Not Available
IDD594Not Available
IguratimodIguratimod is under investigation in Rheumatoid Arthritis.
IlorasertibIlorasertib has been used in trials studying the treatment of Myelodysplasia, Solid Neoplasm, Advanced Cancers, Advanced Solid Tumors, and Acute Myelogenous Leukemia, among others.
ImatinibA tyrosine kinase inhibitor used to treat a number of leukemias, myelodysplastic/myeloproliferative disease, systemic mastocytosis, hypereosinophilic syndrome, dermatofibrosarcoma protuberans, and gastrointestinal stromal tumors.
IMD-0354Not Annotated
ImidocarbImidocarb is a urea derivative used in veterinary medicine as an antiprotozoal agent for the treatment of infection with Babesia and other parasites.
ImidureaImidurea is an antimicrobial preservative used in cosmetics. It acts as a formaldehyde releaser.
ImipenemA carbapenem antibiotic normally administered with cilastatin to treat a variety of infections.
INCB13739Investigated for use/treatment in diabetes mellitus type 2 and diabetes prevention.
INCB3284Investigated for use/treatment in inflammatory disorders (unspecified).
IndapamideA thiazide diuretic used to treat hypertension as well as edema due to congestive heart failure.
IndibulinInvestigated for use/treatment in solid tumors.
IndisulamInvestigated for use/treatment in lung cancer.
IndoraminIndoramin is a discontinued piperidine antiadrenergic drug with the trade names Baratol and Doralese. It is a selective alpha-1 adrenergic antagonist with no reflex tachycardia and direct myocardial depression action.
InfigratinibAn FGFR inhibitor used to treat locally advanced or metastatic cholangiocarcinoma in adults with a fibroblast growth factor receptor 2 (FGFR2) rearrangement.
IniparibNot Annotated
Inosine pranobexA medication used to treat subacute sclerosing panencephalitis.
Iobenzamic acidNot Annotated
Iodohippuric acidIodohippuric acid is under investigation in clinical trial NCT02599844 (Impact of Pediatric Acute Renal Injury in Severe Sepsis in Young Adults).
Iofolastat I-123Iofolastat I-123 is under investigation in clinical trial NCT00992745 (A Phase I Pilot Study Comparing 123I MIP 1072 Versus 111In Capromab Pendetide in Subjects With Metastatic Prostate Cancer).
IoforminolIoforminol has been used in trials studying the diagnostic of Cardio Renal Safety in High-risk Elderly Subjects Undergoing a Coronary CATH With or Without PCI.
Iolopride I-123Iolopride I-123 is a small molecule drug. The usage of the INN stem '-pride' in the name indicates that Iolopride I-123 is a sulpiride derivative and analogue. Iolopride I-123 has...
IPI-493IPI-493 has been used in trials studying the treatment of Advanced Malignancies.
Isoindolin-1,3-DithioneNot Annotated
Isopenicillin NNot Available
IspinesibInvestigated for use/treatment in breast cancer, lung cancer, solid tumors, renal cell carcinoma, pediatric indications, ovarian cancer, and head and neck cancer.
ItoprideAn acetylcholine esterase inhibitor and dopamine D2 receptor antagonist used to treat symptoms of functional dyspepsia such as nausea and vomiting.
JNJ-26489112JNJ-26489112 is under investigation in clinical trial NCT00579384 (A Study of the Effects of JNJ-26489112 on the Photic Induced Paroxysmal Electroencephalogram (EEG) Response in Patients With Photosensitive Epilepsy).
JNJ-41443532JNJ-41443532 has been used in trials studying the basic science and treatment of Diabetes Mellitus, Type 2.
JTC-801 free baseAn antagonist of nociceptin receptor and analgesic agent, evaluated for its use in cancer treatment.
K-134K-134 has been used in trials studying the treatment of Intermittent Claudication.
KD3010Investigated for use/treatment in metabolic disease and obesity.
KRN-633Not Annotated
KX-2361Not Annotated
LabetalolAn alpha and beta adrenergic antagonist used to treat hypertension, angina, and sympathetic overactivity syndrome.
LacosamideAn antiepileptic drug used to treat partial-onset seizures and primary generalized tonic-clonic seizures.
LadarixinLadarixin is under investigation in clinical trial NCT04628481 (A Study of Oral Ladarixin in New-onset Type 1 Diabetes and a Low Residual Β-Cell Function).
LafutidineLafutidine has been investigated in Peptic Ulcer, Community-acquired Pneumonia, and Gastroesophageal Reflux Disease (GERD).
LandiololA rapid-acting selective beta-blocker used to reduce ventricular rate in supraventricular tachycardia in adults.
LanifibranorLanifibranor is under investigation in clinical trial NCT03008070 (Phase 2b Study in NASH to Assess IVA337).
LaromustineInvestigated for use/treatment in brain cancer, cancer/tumors (unspecified), colorectal cancer, leukemia (lymphoid), leukemia (myeloid), lung cancer, myelodysplastic syndrome, pediatric indications, and solid tumors.
LasmiditanAn oral 5HT1F agonist used for the acute treatment of migraine headache with or without aura.
LatamoxefLatamoxef is an oxacephem antibiotic usually grouped with the cephalosporins. It is used to treat bacterial infections. Latamoxef is primarily indicated in conditions like Bone and joint infection, GI infections,...
LecimibideLecimibide is a small molecule drug. Lecimibide has a monoisotopic molecular weight of 590.29 Da.
LenacapavirA first-in-class capsid inhibitor being investigated for use in HIV-1 treatment.
LenampicillinLenampicillin is a small molecule drug. The usage of the INN stem '-cillin' in the name indicates that Lenampicillin is a antibiotic, 6-aminopenicillanic acid derivative. Lenampicillin has a monoisotopic molecular...
LenvatinibA receptor tyrosine kinase inhibitor used for the treatment of metastatic thyroid cancer, advanced renal cell carcinoma in combination with everolimus, and unresectable hepatocellular carcinoma.
LevetiracetamA novel anticonvulsant agent used as an adjunct medication to manage partial onset, myoclonic, and generalized tonic-clonic seizures in patients with epilepsy.
LevobupivacaineA drug used for nerve block and anesthesia.
Levosulpirideindicated to treat dyspepsia, symptoms of Meniere's syndrome, and second line in the treatment of drug-induced nausea and vomiting.
LGD-6972LGD-6972 is under investigation in clinical trial NCT01919684 (Study to Evaluate Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of LGD-6972 in Healthy Subjects and Subjects With Type 2 Diabetes Mellitus).
LidamidineLidamidine is a small molecule drug. Lidamidine has a monoisotopic molecular weight of 220.13 Da.
LidocaineA local anesthetic used in a wide variety of superficial and invasive procedures.
LinezolidAn oxazolidinone antibiotic used to treat infections by susceptible strains of aerobic Gram-positive bacteria.
LinifanibInvestigated for use/treatment in leukemia (myeloid), myelodysplastic syndrome, and solid tumors.
LinrodostatLinrodostat is under investigation in clinical trial NCT03247283 (Pharmacokinetics and Metabolism Study in Healthy Male Participants).
LitronesibLitronesib has been used in trials studying the treatment of Solid Tumors, Ovarian Cancer, Gastric Cancer, Prostate Cancer, and Acute Leukaemia, among others.
LixivaptanInvestigated for use/treatment in hyponatremia and congestive heart failure.
LomustineAn alkylating agent used as a part of chemotherapeutic regimens for the treatment of primary and metastatic brain tumors as well as refractory or relapsed Hodgkin's disease in addition to surgical and/or radiotherapeutic treatments.
LoracarbefUsed to treat upper respiratory tract bacterial infections, chronic bronchitis, pneumonia, sinusitis, pharyntitis and tonsillitis, skin absceses, urinary tract infections and pyelonephritis caused by E. coli, S. pyogenes, S. aureus,...
LorcainideNot Annotated
LorlatinibAn anaplastic lymphoma kinase inhibitor used to treat anaplastic lymphoma kinase positive metastatic non small cell lung cancer.
LozilureaLozilurea is a small molecule drug. Lozilurea has a monoisotopic molecular weight of 212.07 Da.
LufenuronLufenuron is used in veterinary for the control of flea.
LY-295501ILX-295501 has been used in trials studying the treatment of Ovarian Cancer, Metastatic Cancer, Fallopian Tube Cancer, and Primary Peritoneal Cavity Cancer.
LY-3009120Not Annotated
m-Hydroxyhippuric acidNot Available
MacitentanAn endothelin receptor antagonist used to manage pulmonary arterial hypertension to delay disease progression.
MafenideAn antimicrobial topical agent indicated for use as an adjunctive treatment to control bacterial infection when used under moist dressings over meshed autografts on excised burn wounds.
MasitinibMasitinib is a tyrosine-kinase inhibitor used in the treatment of mast cell tumors in dogs. It has been available in Europe since 2009, under the brand name Masivet. In the...
MebenilAn obsolete fungicide used to control various pathogens on cereals and seed potatoes.
MefrusideNot Annotated
MeglitinideMeglitinide is a small molecule drug. Meglitinide has a monoisotopic molecular weight of 333.08 Da.
MeloxicamAn NSAID used to treat osteoarthritis in adults, rheumatoid arthritis in adults, and juvenile rheumatoid arthritis in pediatrics.
MepivacaineA local anesthetic used for local or regional analgesia or anesthesia.
MerimepodibFor the treatment of hepatitis C virus (HCV) infection.
MeropenemA carbapenem antibiotic used to treat a wide variety of infections in the body.
Mesosulfuron-methylMesosulfuron-methyl is under investigation in clinical trial NCT01118117 (A Multi-center Clinical Trial of the Misago™ Self-Expanding Stent System for Superficial Femoral Artery).
MetabromsalanNot Annotated
MetahexamideNot Annotated
MetampicillinMetampicillin is a penicillin antibiotic prepared by the reaction of ampicillin with formaldehyde. It is hydrolysed in aqueous solution to form ampicillin. Hydrolysis is rapid under acid conditions like the...
MethenamineA urinary tract antiseptic and antibacterial drug used for the prophylaxis and treatment of frequently recurring urinary tract infections requiring a long-term therapy.
MethfuroxamMethfuroxam is under investigation in clinical trial NCT01213407 (Dendritic Cell Cancer Vaccine for High-grade Glioma).
MetiamidePotential in the treatment and the management of acid-reflux disorders (GERD), peptic ulcer disease, heartburn, and acid indigestion.
MeticillinUsed to treat infections caused by susceptible Gram-positive bacteria, particularly beta-lactamase-producing organisms such as Staphylococcus aureus that would otherwise be resistant to most penicillins.
MetoclopramideAn antiemetic agent and dopamine D2 antagonist used in the treatment of gastroesophageal reflux disease, prevention of nausea and vomiting, and to stimulate gastric emptying.
MetolazoneA thiazide-like diuretic used to treat hypertension.
MezlocillinUsed to treat serious gram–negative infections of the lungs, urinary tract, and skin.
MibampatorMibampator has been used in trials studying the treatment of Alzheimer's Disease.
MilacemideMilacemide is a small molecule drug. Milacemide has a monoisotopic molecular weight of 144.13 Da.
MirabegronA beta-3 adrenergic agonist used to treat overactive bladder and neurogenic detrusor overactivity.
MirdametinibA kinase inhibitor used to treat neurofibromatosis type 1 in children and adults.
MirodenafilMirodenafil has been used in trials studying the treatment and supportive care of Kidney Diseases, Urologic Diseases, Renal Insufficiency, Erectile Dysfunction, and Male Erectile Dysfunction.
MivebresibMivebresib is a small molecule drug. The usage of the INN stem '-bresib' in the name indicates that Mivebresib is a inhibitor of the bromodomain and extra-terminal motif (BET) family...
MK-0686MK0686 has been used in trials studying the treatment of Osteoarthritis, Pain, Postoperative, and Neuralgia, Postherpetic.
MK-8033Not Annotated
MocetinostatMocetinostat has been used in trials studying the treatment of Lymphoma, Urothelial Carcinoma, Relapsed and Refractory, Myelodysplastic Syndrome, and Metastatic Leiomyosarcoma, among others.
MoclobemideA monoamine oxidase inhibitor used in the treatment of major depressive disorder and bipolar disorder.
MomelotinibA Janus Kinase inhibitor used to treat intermediate or high-risk myelofibrosis.
MosaprideA prokinetic 5-HT4 receptor agonist used to stimulate gastric motility.
MozenavirNot Available
N-(6-Aminohexyl)-5-Chloro-1-NaphthalenesulfonamideNot Available
N-(Benzoylcarbamoyl)-beta-D-glucopyranosylamineNot Available
N-6022N6022 has been used in trials studying the treatment of Asthma and Cystic Fibrosis.
N-acetyl-N'-beta-D-glucopyranosyl ureaNot Available
N-BenzylformamideNot Available
N-phenylthioureaNot Available
N,N-dimethylformamideNot Available
NacubactamNacubactam is under investigation in clinical trial NCT03174795 (A Study to Investigate the Pharmacokinetics of RO7079901 and Meropenem in Participants With a Complicated Urinary Tract Infection).
NafcillinA penicillin derivative antibiotic used to treat susceptible staphylococcal infections.
NaluzotanInvestigated for use/treatment in anxiety disorders and depression.
NarlaprevirNot Annotated
NaronaprideInvestigated for use/treatment in gastroesophageal reflux disease (GERD) and gastroparesis.
NavarixinNavarixin has been investigated for the treatment of Asthma.
NavitoclaxNavitoclax has been used in trials studying the treatment and basic science of Solid Tumors, Non-Hodgkin's Lymphoma, EGFR Activating Mutation, Chronic Lymphoid Leukemia, and Hematological Malignancies, among others. Navitoclax is...
NCX 701Investigated for use/treatment in pain (acute or chronic).
NebentanNebentan is a small molecule drug. The usage of the INN stem '-entan' in the name indicates that Nebentan is a endothelin receptor antagonist. Nebentan has a monoisotopic molecular weight...
NelotanserinNelotanserin has been used in trials studying the treatment of Lewy Body Dementia, Visual Hallucinations, Dementia With Lewy Bodies, and REM Sleep Behavior Disorder. It is a highly selective antagonist...
NemonaprideNot Annotated
NepafenacAn ophthalmic NSAID used for the symptomatic treatment of pain and inflammation associated with cataract surgery.
NesbuvirNesbuvir has been investigated for the treatment of Hepatitis C.
NetazepideNetazepide has been used in trials studying the prevention and treatment of Dyspepsia, Hypergastrinaemia, Barrett's Esophagus, ECL-cell Hyperplasia, and Rebound Hyperacidity, among others.
NetupitantAn antiemetic agent used in combination with palonosetron to prevent acute and delayed vomiting and nausea caused by chemotherapy.
NevanimibeNevanimibe is under investigation in clinical trial NCT03053271 (A Study of ATR-101 for the Treatment of Endogenous Cushing's Syndrome).
NicarbazinNot Annotated
NiclosamideAn anthelmintic indicated in the treatment of beef, pork, fish, and dwarf tapeworm infections in adults and children.
NimesulideA cyclooxygenase 2 inhibitor used to treat acute pain and primary dysmenorrhea.
NimustineNimustine has been used in trials studying the treatment of Glioblastoma.
NiravolineNiravoline is a small molecule drug. Niravoline has a monoisotopic molecular weight of 379.19 Da.
NirmatrelvirAn oral protease inhibitor with emergency use authorization for the treatment of mild-to-moderate COVID-19.
NitrocefinNitrocefin is a chromogenic cephalosporin substrate used to detect the presence of beta-lactamase enzymes, an important mediator of bacterial antibiotic resistance. While other detection methods exist, such as PCR, nitrocefin...
NonivamideNonivamide is used as a topical analgesic and is also used as a flavoring ingredient , , .
NoxytiolinLocal antibacterial that probably acts by releasing formaldehyde in aqueous solutions. It is used for THERAPEUTIC IRRIGATION of infected body cavities - bladder, peritoneum, etc. and as a spray for...
NRC-AN-019Not Annotated
NS-3728Investigated for use/treatment in anemia (sickle cell) and cancer/tumors (unspecified).
NS-398NS-398 is a COX-2 inhibitor. It was developed as part of the mechanistic study of the cyclooxygenases.
NupafantNupafant is a small molecule drug. The usage of the INN stem '-pafant' in the name indicates that Nupafant is a platelet-activating factor antagonist. Nupafant has a monoisotopic molecular weight...
OclacitinibNot Annotated
OlorofimOlorofim is under investigation in clinical trial NCT03340597 (Assessment of Varying Oral Dosing Regimens for F901318 in Healthy Subjects).
OmbitasvirA direct acting antiviral agent used in combination with other antiviral agents for the treatment of Hepatitis C Virus (HCV) infections.
Omecamtiv MecarbilOmecamtiv Mecarbil has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic Heart Failure, and History of Chronic Heart Failure, among others.
OmipalisibOmipalisib has been used in trials studying the treatment of CANCER, Solid Tumours, and Idiopathic Pulmonary Fibrosis.
OnalespibInvestigated for use/treatment in cancer/tumors (unspecified).
ORC-13661ORC-13661 is under investigation in clinical trial NCT05730283 (Prevention of Ototoxicity in NTM Patients Treated With IV Amikacin).
OrludodstatOrludodstat is a small molecule drug. The usage of the INN stem '-dodstat' in the name indicates that Orludodstat is a dihydro-orotate dehydrogenase (DHODH) inhibitor. Orludodstat is under investigation in...
OseltamivirA neuraminidase inhibitor used in the prophylaxis and treatment of influenza.
Oseltamivir acidNot Available
OsimertinibA tyrosine kinase inhibitor used in the treatment of certain types of non-small cell lung carcinoma.
OxacillinA penicillin antibiotic used to treat a number of susceptible bacterial infections.
OximonamOximonam is a small molecule drug. The usage of the INN stem '-monam' in the name indicates that Oximonam is a monobactam antibiotic. Oximonam has a monoisotopic molecular weight of...
OxyclozanideOxyclozanide is a small molecule drug. Oxyclozanide has a monoisotopic molecular weight of 398.88 Da.
p-ToluenesulfonamideNot Available
PadnarsertibNot Annotated
PalosuranPalosuran is a small molecule drug. The usage of the INN stem '-osuran' in the name indicates that Palosuran is a urotensin receptor antagonist. Palosuran has a monoisotopic molecular weight...
PamufetinibPamufetinib is a small molecule drug. The usage of the INN stem '-tinib' in the name indicates that Pamufetinib is a tyrosine kinase inhibitor. Pamufetinib is under investigation in clinical...
ParapropamolParapropamol is a small molecule drug. Parapropamol has a monoisotopic molecular weight of 165.08 Da.
Paratoulene phosphateNot Available
ParitaprevirA direct acting antiviral agent used in combination with other antiviral agents for the treatment of Hepatitis C Virus (HCV) infections.
ParsalmideParsalmide is a small molecule drug. Parsalmide has a monoisotopic molecular weight of 246.14 Da.
PavinetantPavinetant has been used in trials studying the basic science and treatment of Safety and Schizophrenia.
PazopanibAn antineoplastic agent used in the treatment of advanced renal cell cancer and advanced soft tissue sarcoma in patients with prior chemotherapy.
PC-786Not Annotated
PCI-27483PCI-27483 has been used in trials studying the treatment of Pancreatic Cancer, Ductal Adrenocarcinoma, and Exocrine Pancreatic Cancer.
PenamecillinNot Annotated
PenimepicyclinePenimepicycline is a tetracycline-class antibiotic. It is mentioned on List A produced by the Government of Canada, which is a list of antimicrobial active pharmaceutical ingredients . In the classification...
PesampatorPF-04958242 has been used in trials studying the basic science and treatment of Schizophrenia and Hearing Loss, Sensorineural.
PexmetinibPexmetinib is under investigation in clinical trial NCT04074967 (Study of ARRY-614 Plus Either Nivolumab or Ipilimumab).
PF-00489791PF-00489791 has been used in trials studying the treatment of Hypertension, Raynaud's Disease, Diabetic Nephropathies, Hypertension, Pulmonary, and Peripheral Vascular Disease.
PF-00610355PF-00610355 has been used in trials studying the treatment of Lung Disease, Moxifloxacin, Pulmonary Disease, Asthma, Bronchial, and Bronchial Diseases, among others.
PF-03715455PF-03715455 has been used in trials studying the treatment of Asthma, Pulmonary Disease, Chronic Obstructive, and Chronic Obstructive Pulmonary Disease (COPD).
PF-04457845PF-04457845 is under investigation in Fear Conditioning. PF-04457845 has been investigated for the treatment of Tourette Syndrome and Cannabis Dependence.
PF-05089771PF-05089771 is under investigation in clinical trial NCT01529671 (A Safety And Tolerability Study Of PF-05089771 In Healthy Subjects And In Subjects With Otseoarthritis Of The Knee).
PF-06282999Pf 06282999 is under investigation in clinical trial NCT01626976 (A Study To Assess The Safety, Tolerability And Pharmacokinetics Of PF-06282999 Administered Orally In Healthy Adult Subjects).
PF-5212372PF-5212372 is under investigation in clinical trial NCT02795832 (A Study to Determine the Safety & Efficacy of ZPL-5212372 in Healthy Subjects and in Subjects With Atopic Dermatitis).
PF-562271Not Annotated
PH-797804PH-797804 has been investigated for the treatment of Osteoarthritis.
PhenacemideUsed to control certain seizures in the treatment of epilepsy.
PhenacetinUsed principally as an analgesic.
PheneturideNot Annotated
PhenoxymethylpenicillinA penicillin antibiotic used to prevent and treat mild to moderately severe infections in the respiratory tract, skin, and soft tissues.
PhthalylsulfathiazoleA sulfonamide antibacterial indicated in the treatment of gastrointestinal infections.
PiclamilastPiclamilast (RP-73,401), is a selective PDE4 inhibitor comparable to other PDE4 inhibitors for its anti-inflammatory effects. It has been investigated for its applications to the treatment of conditions such as...
PicobenzidePicobenzide is a small molecule drug. Picobenzide has a monoisotopic molecular weight of 240.13 Da.
PictilisibPictilisib has been used in trials studying the treatment of Solid Cancers, Breast Cancer, Advanced Solid Tumours, Metastatic Breast Cancer, and Non-Hodgkin's Lymphoma, Solid Cancers, among others.
Piflufolastat F 18A radiopharmaceutical diagnostic agent used with PET to image PSMA-positive lesions for the diagnosis of metastatic or recurrent prostate cancer.
PIK-75PIK-75 is a preferential p110 alpha/gamma PI3K inhibitor.
PilaralisibPilaralisib is an orally available small molecule that selectively inhibits the activity of phosphoinositide-3 kinase (PI3K). Pilaralisib has been used in trials studying the treatment of Cancer, Lymphoma, Solid Tumors,...
PilsicainidePilsicainide has been investigated for the treatment of Paroxysmal Atrial Fibrillation.
PimavanserinA second generation atypical antipsychotic used for the treatment of hallucinations and delusions caused by Parkinson's Disease.
PimitespibTAS-116 is under investigation in clinical trial NCT02965885 (A Study of TAS-116 in Patients With Solid Tumors).
PincainidePincainide is a small molecule drug. The usage of the INN stem '-cain-' in the name indicates that Pincainide is a class I antiarrhythmic, procainamide and lidocaine derivative. Pincainide has...
PiperacillinA penicillin antibiotic combined with tazobactam to treat piperacillin-resistant, piperacillin/tazobactam­ susceptible, β-lactamase generating strains of several bacteria.
PiperineBioperine has been used in trials studying the treatment of Multiple Myeloma and Deglutition Disorders.
PiracetamA nootropic cyclic GABA derivative used in myoclonus, sickle cell disease, alcohol dependence, and as a general cognitive enhancer.
PiragliatinPiragliatin is a small molecule drug. The usage of the INN stem '-gliatin' in the name indicates that Piragliatin is a glucokinase activator. Piragliatin has a monoisotopic molecular weight of...
PirbenicillinPirbenicillin is a small molecule drug. The usage of the INN stem '-cillin' in the name indicates that Pirbenicillin is a antibiotic, 6-aminopenicillanic acid derivative. Pirbenicillin has a monoisotopic molecular...
PiretanideA loop diuretic used to manage essential arterial hypertension and edema cardiac, hepatic, and renal origin.
PivampicillinAn ampicillin prodrug used to treat a variety of infections.
PivmecillinamA prodrug of the beta lactam antibiotic mecillinam, indicated for the treatment of uncomplicated urinary tract infections (UTIs).
PKI-179PKI-179 has been used in trials studying the treatment of Advanced Malignant Solid Tumors.
PlatensimycinNot Available
PlixorafenibPLX8394 is under investigation in clinical trial NCT02428712 (A Study of PLX8394 as a Single Agent in Patients With Advanced Unresectable Solid Tumors).
PLX-4720Not Available
PolmacoxibPolmacoxib has been used in trials studying the treatment of Osteoarthritis, Osteoarthritis, Hip, Osteoarthritis, Knee, Localized Primary Osteoarthritis of Hip, and Localized Primary Osteoarthritis of Knee.
PolythiazideA thiazide diuretic used in the management of hypertension and treatment of edema.
PractololUsed in the emergency treatment of cardiac arrhythmias.
PrazocillinPrazocillin is a small molecule drug. The usage of the INN stem '-cillin' in the name indicates that Prazocillin is a antibiotic, 6-aminopenicillanic acid derivative. Prazocillin has a monoisotopic molecular...
PresatovirPresatovir has been used in trials studying the treatment of RSV Infection, Respiratory Syncytial Virus (RSV), Respiratory Syncytial Virus Infections, and Respiratory Syncytial Virus (RSV) Infections.
PrilocaineA local anesthetic used in dental procedures.
PritelivirPritelivir has been used in trials studying the prevention of HSV-2 and Genital Herpes.
ProbenecidA medication used to treat gouty arthritis, tophaceous gout, and hyperuricemia.
ProcainamideA medication used to treat life threatening ventricular arrhythmias.
Procaine benzylpenicillinA local anesthetic and antibiotic combination for intramuscular injection to treat a variety of bacterial infections while reducing pain from a deep intramuscular injection.
ProcarbazineAn antineoplastic agent indicated for the treatment of stage III and stage IV Hodgkin's disease in combination with other chemotherapeutic agents.
PropacetamolPropacetamol is a paracetamol prodrug of intravenous administration used to control fever and pain of perioperative period in multimodal analgesia therapy.
PropicillinNot Annotated
PXS-4728A free basePXS-4728A free base is under investigation in clinical trial NCT05904717 (Effect of PXS-4728A on Microglia Activation in Participants With Isolated Rapid Eye Movement Sleep Behaviour Disorder).
PyrotinibPyrotinib is under investigation in clinical trial NCT03756064 (Neoadjuvant Study of Pyrotinib in Patients With HER2 Positive Breast Cancer).
PyrrocainePyrrocaine is a small molecule drug. The usage of the INN stem '-caine' in the name indicates that Pyrrocaine is a local anaesthetic. Pyrrocaine has a monoisotopic molecular weight of...
QuinacillinQuinacillin is a small molecule drug. The usage of the INN stem '-cillin' in the name indicates that Quinacillin is a antibiotic, 6-aminopenicillanic acid derivative. Quinacillin has a monoisotopic molecular...
QuinethazoneUsed to treat hypertension.
QuizartinibA FLT3 inhibitor used in combination with cytarabine and anthracycline to treat acute myeloid leukemia with FLT3 internal tandem duplication
R-95845R-95845 is an inhibitor of HIV-1 reverse transcriptase.
RabusertibRabusertib has been used in trials studying the treatment of Cancer, Solid Tumors, Advanced Cancer, Pancreatic Neoplasms, and Non Small Cell Lung Cancer.
RacloprideRaclopride has been used in trials studying Parkinson Disease.
RadiprodilRadiprodil has been used in trials studying the treatment of Infantile Spasms (IS) and Diabetic Peripheral Neuropathic Pain.
RadotinibRadotinib is indicated for the treatment of different types of cancer, most notably Philadelphia chromosome-positive (Ph+) chronic myeloid leukemia (CML) with resistance or intolerance of other Bcr-Abl tyrosine-kinase inhibitors, such...
RafoxanideRafoxanide is a small molecule drug. Rafoxanide has a monoisotopic molecular weight of 624.82 Da.
RamatrobanRamatroban has been used in trials studying the treatment of Asthma.
RanimustineNot Annotated
RazupenemRazupenem has been used in trials studying the treatment of Skin Infections.
RecainamRecainam is a small molecule drug. The usage of the INN stem '-cain-' in the name indicates that Recainam is a class I antiarrhythmic, procainamide and lidocaine derivative. Recainam has...
RedaporfinNot Available
RefametinibInvestigated for use/treatment in cancer/tumors (unspecified).
RegorafenibA kinase inhibitor used to treat patients with metastatic colorectal cancer, unresectable, locally advanced, or metastatic gastrointestinal stromal tumors, and hepatocellular carcinoma.
RelenoprideRelenopride has been used in trials studying the treatment of Chronic Idiopathic Constipation.
RelugolixAn oral GnRH receptor antagonist for androgen deprivation therapy in the treatment of advanced prostate cancer.
RemacemideInvestigated for use/treatment in epilepsy, huntington's disease, and parkinson's disease.
RemoxiprideAn discontinued atypical antipsychotic selective for dopamine D2 receptors.
RenzaprideFor the treatment of constipation-predominant irritable bowel syndrome (IBS-C).
ReparixinReparixin has been used in trials studying the treatment and prevention of Breast Cancer, Metastatic Breast Cancer, Pancreatectomy for Chronic Pancreatitis, Islet Transplantation in Diabetes Mellitus Type 1, and Pancreatic...
ResatorvidInvestigated for use/treatment in sepsis and septicemia.
ResminostatResminostat has been used in trials studying the treatment of Sezary Syndrome, Mycosis fungoides, Hodgkin's Lymphoma, Hepatocellular Carcinoma, and Lymphoma, T-Cell, Cutaneous, among others.
ResorantelResorantel is a small molecule drug. The usage of the INN stem '-antel' in the name indicates that Resorantel is a anthelminthic. Resorantel has a monoisotopic molecular weight of 306.98...
RetaspimycinInvestigated for use/treatment in gastric cancer, lung cancer, and multiple myeloma.
RevefenacinAn anticholinergic agent used to treat COPD.
RevumenibA small molecule menin inhibitor for the treatment of relapsed/refractory leukemia with KMT2A translocation.
RG-2833Not Annotated
Rgb-286638 free baseNot Annotated
RifampinAn antibiotic used alone or in combination with other antimicrobial drugs to treat tuberculosis and asymptomatic carriers of Neisseria meningitidis.
RilapladibInvestigated for use/treatment in atherosclerosis and cardiovascular disorders.
RipasudilA rho kinase inhibitor indicated to treat ocular hypertension and open-angle glaucoma.
RipretinibA kinase inhibitor used to treat advanced gastrointestinal stromal tumor (GIST).
RisotilideRisotilide is a small molecule drug. The usage of the INN stem '-ilide' in the name indicates that Risotilide is a sematilide derivative class III antiarrhythmic. Risotilide has a monoisotopic...
RitipenemRitipenem is a small molecule drug. Ritipenem has a monoisotopic molecular weight of 288.04 Da.
RO-4987655RO4987655 has been used in trials studying the treatment of Neoplasms.
RociletinibRociletinib has been used in trials studying the treatment and prevention of Nonsmall Cell Lung Cancer, Non-small Cell Lung Cancer, and Locally Advanced or Metastatic Non-small Cell Lung Cancer.
RoflumilastA selective phosphodiesterase-4 inhibitor indicated to decrease the risk of exacerbations in patients with severe chronic obstructive pulmonary disease (COPD) and to treat skin conditions such as plaque psoriasis and atopic dermatitis.
RopivacaineAn amide-type local anesthetic used for local or regional anesthesia during surgery and for short-term management of acute pain.
RosuvastatinAn HMG-CoA reductase inhibitor used to lower lipid levels and reduce the risk of cardiovascular disease including myocardial infarction and stroke.
RSV-604RSV-604 is under investigation in clinical trial NCT00416442 (Safety, Tolerability and Pharmacokinetic Study of Single and Multiple Intravenous Doses of RSV604 in Healthy Subjects.).
S-23An androgen receptor modulator.
S-38093Not Annotated
S-EthylisothioureaS-Ethylisothiourea is a nitric oxide synthase inhibitor.
SafotibantSafotibant is a small molecule drug. The usage of the INN stem '-tibant' in the name indicates that Safotibant is a bradykinin receptor antagonist. Safotibant has a monoisotopic molecular weight...
SalicylamideSalicylamide is the common name for the substance o-hydroxybenzamide, or amide of salicyl. Salicylamide is a non-prescription drug with analgesic and antipyretic properties. It has similar medicinal uses to aspirin....
Salicylamide O-acetic acidA salicylate indicated in combination with local anesthetics and corticosteroids for short term treatment of inflammation.
SalicylanilideNot Annotated
Salicylhydroxamic AcidNot Available
SanfetrinemSanfetrinem is a small molecule drug. Sanfetrinem has a monoisotopic molecular weight of 281.13 Da.
Sanfetrinem cilexetilSanfetrinem cilexetil is under investigation in clinical trial NCT05388448 (EBA, Safety and Tolerability of Sanfetrinem Cilexetil).
SAR-125844SAR-125844 is under investigation in clinical trial NCT01391533 (Study of SAR125844 Single Agent Administered as Slow Intravenous Infusion in Adult Patients With Advanced Malignant Solid Tumors).
SaredutantInvestigated for use/treatment in depression and anxiety disorders.
SB-269970SB-269970 is an experimental drug developed by GlaxoSmithKline. In the studies performed with this agent, it has been suggested that SB-269970 acts either as a selective antagonist or inverse agonist...
SB-705498SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.
SB-743921Investigated for use/treatment in cancer/tumors (unspecified) and lymphoma (non-hodgkin's).
SC-236SC-236 is a potent, selective, orally active inhibitor of cyclooxygenase-2 (COX-2) that has been studied in cancer therapy , lower back pain , and inflammation , , , .
SC-74020Not Available
SeclidemstatNot Annotated
SelexipagA non prostanoid IP prostacyclin receptor agonist used to treat pulmonary arterial hypertension.
SelonsertibSelonsertib is under investigation in clinical trial NCT03053050 (Safety and Efficacy of Selonsertib in Adults With Nonalcoholic Steatohepatitis (NASH) and Bridging (F3) Fibrosis).
SemapimodSemapimod has been used in trials studying the treatment of Crohn Disease.
SematilideSematilide is a small molecule drug. The usage of the INN stem '-ilide' in the name indicates that Sematilide is a sematilide derivative class III antiarrhythmic. Sematilide has a monoisotopic...
SembragilineSembragiline is a small molecule drug. The usage of the INN stem '-giline' in the name indicates that Sembragiline is a monoamine oxydase (MAO)-inhibitor type B. Sembragiline has a monoisotopic...
SemustineNot Annotated
SenicapocInvestigated for use/treatment in anemia (sickle cell) and asthma.
SildenafilA phosphodiesterase inhibitor used for the treatment of erectile dysfunction.
Silver sulfadiazineA topical sulfonamide antibiotic that acts on the bacterial cell wall and cell membrane; approved for the treatment of burns.
SirpiglenastatSirpiglenastat, also known as DRP-104, is a prodrug of 6-diazo-5-oxo-L-norleucine (DON), which is a broad-acting glutamine antagonist. It is under investigation in clinical trial NCT04471415 (Study to Investigate DRP-104 in...
SitravatinibSitravatinib is under investigation in clinical trial NCT03680521 (Neoadjuvant Sitravatinib in Combination With Nivolumab in Patients With Clear Cell Renal Cell Carcinoma).
SivelestatSivelestat has been used in trials studying the treatment of Acute Lung Injury and Respiratory Distress Syndrome, Adult.
SKF-91488Not Available
SLC-0111Not Available
SLV319Investigated for use/treatment in obesity.
SLx-4090Investigated for use/treatment in hyperlipidemia.
SNS-314Investigated for use/treatment in solid tumors.
SNX-5422Investigated for use/treatment in cancer/tumors (unspecified).
SonepiprazoleSonepiprazole is a small molecule drug. The usage of the INN stem '-prazole' in the name indicates that Sonepiprazole is a benzimidazole derivative antiulcer medication. Sonepiprazole has a monoisotopic molecular...
SorafenibA kinase inhibitor used to treat unresectable liver carcinoma, advanced renal carcinoma, and differentiated thyroid carcinoma.
SP-8203SP-8203 has been used in trials studying the treatment of Ischemic Stroke.
SparsentanAn endothelin and angiotensin II receptor antagonist indicated to reduce proteinuria in adults with primary immunoglobulin A nephropathy at risk of rapid disease progression.
SpebrutinibSpebrutinib has been used in trials studying the treatment of Rheumatoid Arthritis, Lymphoma, Large B-Cell, Diffuse, and Leukemia Lymphocytic Chronic B-Cell.
StreptozocinA nitrosourea antineoplastic agent used in the treatment of metastatic pancreatic islet cell carcinoma.
SuccinylsulfathiazoleNot Annotated
SulbactamAn beta-lactamase inhibitor antibiotic combined with other antibiotics to treat a variety of susceptible bacterial infections.
Sulbactam pivoxilA prodrug of a beta-lactamase inhibitor used to improve the efficacy of beta lactam antibiotics
SulbenicillinNot Annotated
SulfabenzamideA sulfonamide antibacterial used as an ingredient in various topical and vaginal preparations to treat certain infections, but has been discontinued by the FDA.
SulfacarbamideSulfacarbamide is a small molecule drug. Sulfacarbamide has a monoisotopic molecular weight of 215.04 Da.
SulfacetamideA sulfonamide used to treat inflammatory ocular conditions and acne vulgaris.
SulfachlorpyridazineA sulfonamide antimicrobial used for urinary tract infections and in veterinary medicine.
SulfaclomideSulfaclomide is a small molecule drug. Sulfaclomide has a monoisotopic molecular weight of 312.04 Da.
SulfaclozineSulfaclozine is a small molecule drug. Sulfaclozine has a monoisotopic molecular weight of 284.01 Da.
SulfacytineUsed orally in the treatment of acute urinary tract infections.
SulfadiazineA sulfonamide antibiotic used in a variety of infections, such as urinary tract infections, trachoma, and chancroid.
SulfadimethoxineFor use in the treatment of infections.
SulfadoxineA long acting sulfonamide used for the treatment or prevention of malaria.
SulfaethoxypyridazineNot Annotated
SulfaguanidineSulfaguanidine is a sulfonamide antibiotic with antimicrobial and antibacterial activities.
SulfaisodimidineSulfaisodimidine also called sulfisomidine is an antibacterial product that has been studied for the treatment of urinary tract infections in the 1950s, however, it is unclear whether this drug has...
SulfamerazineAn antibacterial agent used in the treatment of various bacterial infections, such as bronchitis, prostatitis, and urinary tract infections.
SulfameterLong acting sulfonamide used in leprosy, urinary, and respiratory tract infections.
SulfamethazineAn antibacterial agent used in the treatment of various bacterial infections, such as bronchitis, prostatitis, and urinary tract infections.
SulfamethizoleA sulfonamide antibiotic used to treat a wide variety of susceptible bacterial infections.
SulfamethoxypyridazineA sulphonamide antibiotic indicated in the treatment of gonorrhea, inflammation, urinary tract ulcers, and bronchitis.
SulfametopyrazineAn antibiotic used in the treatment or prevention of bacterial infections and malaria.
SulfametroleAn antibiotic indicated in combination intravenous products for various bacterial infections.
SulfamoxoleFor the treatment of bacterial infection.
SulfanilamideA sulfonamide anti-infective used to treat vulvovaginal candidiasis caused by Candida albicans.
SulfanitranNot Annotated
SulfaphenazoleFor the treatment bacterial infections.
SulfaproxylineSulfaproxyline is a small molecule drug. Sulfaproxyline has a monoisotopic molecular weight of 334.1 Da.
SulfapyridineA sulfonamide antibiotic used to treat dermatitis herpetiformis, benign mucous membrane pemphigoid and pyoderma gangrenosum.
SulfaquinoxalineSulfaquinoxaline is a veterinary medicine which can be given to cattle and sheep to treat coccidiosis.It is available in Pakistan with Sanna Laboratories in combination with Amprolium and Vitamin K...
SulfasalazineA salicylate used to treat Crohn's disease, ulcerative colitis, and rheumatoid arthritis.
SulfasymazineSulfasymazine is a small molecule drug. Sulfasymazine has a monoisotopic molecular weight of 307.11 Da.
SulfathiazoleSulfathiazole is effective against a wide range of gram positive and gram negative pathogenic microorganisms. Although no longer used in humans, it is used in cattle.
SulfathioureaNot Annotated
SulfatolamideNot Annotated
SulfatroxazoleSulfatroxazole is a small molecule drug. Sulfatroxazole has a monoisotopic molecular weight of 267.07 Da.
SulfisoxazoleA sulfonamide antibiotic used with other antibiotics to prevent and treat a variety of bacterial infections.
SulofenurSulofenur is a small molecule drug. Sulofenur has a monoisotopic molecular weight of 350.05 Da.
SulopenemSulopenem is a penem antibacterial. It is marketed as the prodrug sulopenem etzadroxil in combination with probenecid.
SulotrobanSulotroban is a small molecule drug. Sulotroban has a monoisotopic molecular weight of 335.08 Da.
SulpirideA selective D2 dopamine receptor antagonist indicated to treat chronic and acute schizophrenia.
SultamicillinA mutual prodrug of ampicillin and sulbactam useful in the treatment of infections caused by beta-lactamase-producing bacteria.
SulthiameA carbonic anhydrase inhibitor used primarily in benign focal epilepsies of childhood that may be useful as an adjunct therapy in a variety of other refractory epilepsies.
SultoprideSultopride is used in Japan, Hong Kong, and Europe to treat schizophrenia. It is of the drug class atypical antipsychotics .
SumatriptanA serotonin receptor agonist used to treat migraines and cluster headaches.
SuncillinSuncillin is a small molecule drug. The usage of the INN stem '-cillin' in the name indicates that Suncillin is a antibiotic, 6-aminopenicillanic acid derivative. Suncillin has a monoisotopic molecular...
SunvozertinibA tyrosine kinase inhibitor used to treat adults with locally advanced or metastatic non-small cell lung cancer (NSCLC) with epidermal growth factor receptor (EGFR) exon 20 insertion mutations.
SurufatinibSurufatinib is under investigation in clinical trial NCT02588170 (Phase III Study of Surufatinib in Treating Advanced Extrapancreatic Neuroendocrine Tumors).
SusalimodSusalimod is a small molecule drug. The usage of the INN stem '-imod' in the name indicates that Susalimod is a immunomodulator, both stimulant/suppressive and stimulant. Susalimod has a monoisotopic...
SutezolidSutezolid has been used in trials studying the treatment of Tuberculosis.
T-900607T900607 has been used in trials studying the treatment of Liver Cancer and Gastric Cancer.
TacedinalineTacedinaline has been used in trials studying the treatment of Lung Cancer, Multiple Myeloma, and Pancreatic Cancer.
TagorizineTagorizine is a small molecule drug. The usage of the INN stem '-rizine' in the name indicates that Tagorizine is a antihistaminic/cerebral (or peripheral) vasodilator. Tagorizine has a monoisotopic molecular...
TAK-243TAK-243 is under investigation in clinical trial NCT03816319 (TAK-243 in Treating Patients With Relapsed or Refractory Acute Myeloid Leukemia or Refractory Myelodysplastic Syndrome or Chronic Myelomonocytic Leukemia).
TAK-715TAK-715 is under investigation in clinical trial NCT00760864 (Safety and Efficacy of TAK-715 in Subjects With Rheumatoid Arthritis).
TalampicillinNot Annotated
TamsulosinAn alpha-1A and alpha-1B adrenergic receptor antagonist used to treat benign prostatic hyperplasia, ureteral stones, prostatitis, and female voiding dysfunction.
TanespimycinInvestigated for use/treatment in leukemia (myeloid) and solid tumors.
TanimilastCHF6001 has been used in trials studying the treatment of Asthma and Chronic Obstructive Pulmonary Disease.
TaprenepagTaprenepag has been used in trials studying the treatment of Ocular Hypertension and Glaucoma, Open-Angle.
TaprizosinTaprizosin is a small molecule drug. Taprizosin has a monoisotopic molecular weight of 506.17 Da.
TasisulamTasisulam has been used in trials studying the treatment and basic science of Melanoma, Lymphoma, Solid Tumors, Breast Cancer, and Ovarian Cancer, among others.
TauromustineTauromustine is a small molecule drug. The usage of the INN stem '-mustine' in the name indicates that Tauromustine is a antineoplastic, alkylating agent, (β-chloroethyl) amine derivative. Tauromustine has a...
TazemetostatA methyltransferase inhibitor indicated to treat patients 16 years and older with metastatic or locally advanced epithelioid sarcoma not eligible for complete resection.
TazobactamA beta lactamase inhibitor administered with antibiotics such as piperacillin and ceftolozane to prevent their degradation, resulting in increased efficacy.
Tebipenem pivoxilAn oral carbapenem antibacterial indicated for complicated urinary tract infections, including pyelonephritis, caused by susceptible Enterobacterales and Enterococcus faecalis in adults with limited or no alternative oral treatment options.
TecovirimatAn antiviral medication used to treat smallpox, monkeypox, and cowpox.
TefinostatTefinostat is under investigation in clinical trial NCT02759601 (Dose Escalation Trial of Tefinostat for Cancer Associated Inflamation in Hepatocellular Carcinoma (HCC)).
TelaglenastatTelaglenastat is under investigation in clinical trial NCT02071862 (Study of the Glutaminase Inhibitor CB-839 in Solid Tumors).
TemanogrelFor the treatment and prophylaxis of arterial thrombosis.
TemgicolurilNot Annotated
TemocillinTemocillin has been investigated in Infection, Liver Dysfunction, and Urinary Tract Infection.
TersolisibSTX-478 is under investigation in clinical trail NCT05768139 (First-in-Human Study of STX-478 as Monotherapy and in Combination With Other Antineoplastic Agents in Participants With Advanced Solid Tumors).
ThiambutosineThiambutosine is a small molecule drug. Thiambutosine has a monoisotopic molecular weight of 343.17 Da.
ThiocitrullineNot Available
TicaloprideInvestigated for use/treatment in gastroesophageal reflux disease (GERD) and gastroparesis.
TicarcillinA beta lactam antibiotic used to treat a variety of infections in the body.
TigemonamTigemonam is a small molecule drug. The usage of the INN stem '-monam' in the name indicates that Tigemonam is a monobactam antibiotic. Tigemonam has a monoisotopic molecular weight of...
TilmacoxibTilmacoxib is a small molecule drug. The usage of the INN stem '-coxib' in the name indicates that Tilmacoxib is a selective cyclo-oxygenase inhibitor. Tilmacoxib has a monoisotopic molecular weight...
TipranavirA protease inhibitor used to treat HIV-1 resistant to more than 1 protease inhibitor.
Tipranavir C-14Tipranavir C-14 is under investigation in clinical trial NCT02253797 (Pharmacokinetics of Tipranavir/Ritonavir and Its Metabolites in Healthy Male Subjects).
TirbanibulinA tyrosine kinase and tubulin inhibitor used to treat actinic keratosis on the face or scalp.
TivozanibA kinase inhibitor to treat adult patients with renal cell carcinoma (RCC) who have failed prior systemic therapies or experienced relapsed disease.
TMC-310911TMC-310911 (also known as ASC-09) is a novel investigational protease inhibitor (PI) that is structurally similar to the currently available darunavir. It is being investigated for use in HIV-1 infections....
TMC-647055TMC647055 has been used in trials studying the treatment of Hepatitis C, Chronic Hepatitis C, Hepatitis C, Chronic, and Chronic Hepatitis C Virus.
TO-901317TO-901317 is an LXRalpha and LXRbeta agonist.
TocainideAn orally active class 1b antiarrhythmic agent that interferes with cardiac sodium channels and typically used to treat ventricular arrhythmias.
TolazamideA sulfonylurea used in the treatment of non insulin dependent diabetes mellitus.
TolbutamideA sulfonylurea used to treat hyperglycemia in patients with type 2 diabetes mellitus.
TonabersatInvestigated for use/treatment in migraine and cluster headaches.
TosifenTosifen is a small molecule drug. Tosifen has a monoisotopic molecular weight of 332.12 Da.
TrametinibA kinase inhibitor used alone or in combination with dabrafenib to treat patients with cancers with specific BRAF mutations, such as melanoma and non-small cell lung cancer.
TrecetilideTrecetilide is a small molecule drug. The usage of the INN stem '-ilide' in the name indicates that Trecetilide is a sematilide derivative class III antiarrhythmic. Trecetilide has a monoisotopic...
TribromsalanTribromsalan is a small molecule drug. Tribromsalan has a monoisotopic molecular weight of 446.81 Da.
TriclocarbanAn antibacterial agent used in liquid soaps and body washes.
TriflumidateTriflumidate is a small molecule drug. Triflumidate has a monoisotopic molecular weight of 401.05 Da.
TrimethobenzamideAn antiemetic used to treat postoperative nausea and vomiting and nausea associated with gastroenteritis.
TTI-101Not Annotated
TucidinostatInvestigated for use/treatment in cancer/tumors (unspecified).
UC-781Investigated for use/treatment in HIV infection.
UdenafilA PDE5 inhibitor used to treat erectile dysfunction.
UpamostatUpamostat has been used in trials studying the treatment of Pancreatic Cancer.
UreaA keratolytic emollient used to treat hyperkeratotic lesions and moisturize the skin.
ValdecoxibA COX-2 inhibitor used to treat osteoarthritis and dysmenorrhoea.
VaniprevirVaniprevir has been used in trials studying the treatment and diagnostic of Hepatitis C, Chronic Hepatitis C, Hepatitis C, Chronic, Chronic Hepatitis C Infection, and Chronic Genotype 1 Hepatitis C...
VemurafenibA kinase inhibitor used to treat patients with Erdheim-Chester Disease who have the BRAF V600 mutation, and melanoma in patients who have the BRAF V600E mutation.
VenetoclaxA BCL-2 inhibitor used to treat chronic lymphocytic leukemia, small lymphocytic lymphoma, or acute myeloid leukemia.
VeraliprideNot Annotated
VercirnonVercirnon is a novel, orally active anti-inflammatory agent that targets a chemokine receptor protein implicated in both Crohn's disease and ulcerative colitis, the two principal forms of IBD. It is...
VerdinexorKpt 335 is under investigation in clinical trial NCT02431364 (Trial of Safety and Tolerability of Oral Verdinexor (Verdinexor) in Healthy Adults).
VidupiprantVidupiprant has been used in trials studying the treatment and basic science of Asthma.
VismodegibA hedgehog pathway inhibitor used to treat patients with locally advanced or metastatic basal cell carcinoma.
VistusertibVistusertib is under investigation for the treatment of Advanced Gastric Adenocarcinoma.
VLX-1005Not Annotated
VM4-037VM4-037 is under investigation in clinical trial NCT00884520 (An Exploratory, Open Label, Multi-Center, Non-Randomized Study of [F-18]VM4-037).
VonoprazanA potassium-competitive acid blocker used in the treatment of acid-related disorders and as an adjunct to Helicobacter pylori eradication.
VorinostatA histone deacetylase (HDAC) inhibitor used for the treatment of cutaneous manifestations in patients with progressive, persistent, or recurrent cutaneous T- cell lymphoma (CTCL) following prior systemic therapies.
VoxilaprevirA nonstructural protein 3 and 4a protease inhibitor used to treat Hepatitis C infections.
VoxtalisibVoxtalisib has been used in trials studying the treatment of Cancer, Melanoma, Lymphoma, Glioblastoma, and Breast Cancer, among others.
VX-148Investigated for use/treatment in autoimmune diseases, psoriasis and psoriatic disorders, and viral infection.
VX-702Investigated for use/treatment in coronary artery disease, inflammatory disorders (unspecified), and rheumatoid arthritis.
WAY-151693Not Available
XipamideA diuretic indicated in the treatment of edema.
XL765For the treatment of various forms of cancer.
Y-33075Not Annotated
ZafirlukastA leukotriene receptor antagonist used for prophylaxis and chronic treatment of asthma.
ZaleplonA sedative used for short term treatment of insomnia in adults.
ZidebactamA diazabicyclooctane beta-lactamase inhibitor and PBP2-binding antibacterial, used only with cefepime, indicated for complicated urinary tract infections including pyelonephritis caused by susceptible Gram-negative pathogens.
ZileutonA leukotriene synthesis inhibitor used in the prophylaxis and treatment of chronic asthma.
ZimlovisertibPF-06650833 is under investigation in clinical trial NCT02609139 (Study to Evaluate Pharmacokinetics of A Modified Release Formulation of PF-06650833 in Healthy Subjects).
ZinviroximeZinviroxime is a small molecule drug. Zinviroxime has a monoisotopic molecular weight of 358.11 Da.
ZoaleneDinitolmide is a fodder additive for prophylaxis against coccidiosis infections in poultry.
ZongertinibZongertinib is an orally bioavailable, selective tyrosine kinase inhibitor that irreversibly targets activating HER2 mutations, including exon 20 insertions, used to inhibit downstream oncogenic signaling in patients with HER2-mutant non-small cell lung cancer.
ZonisamideA sulfonamide anticonvulsant used to treat partial seizures.
ZucapsaicinA topical analgesic used as an adjunct to relieve severe pain of osteoarthritis of the knee in selected adult patients.