Cholinergic Receptor Agonist

Name
Cholinergic Receptor Agonist
Accession Number
DBCAT003290
Description

Not Available

Drugs
DrugDrug Description
CevimelineA muscarinic agonist with parasympathomimetic activities that is used for the symptomatic treatment of dry mouth in patients with Sjögren's Syndrome.
CarbamoylcholineA direct acting miotic agent administered ophthalmically to decrease intraocular pressure after cataract surgery, and to induce miosis during surgery.
PilocarpineA muscarinic agonist used to treat dry mouth and various ophthalmic conditions, such as presbyopia, increased intraocular pressure, and angle-closure glaucoma.
AcetylcholineA parasympathomimetic neurotransmitter used to induce miosis of the iris in seconds after delivery of the lens in cataract surgery, in penetrating keratoplasty, iridectomy and other anterior segment surgery where rapid miosis may be required.
MethacholineA parasympathomimetic bronchoconstrictor used to diagnose bronchial hyperreactivity in subjects who do not have clinically apparent asthma.
VareniclineA partial agonist at nicotinic acetylcholine receptors used as an aid in smoking cessation.
Drugs & Drug Targets
DrugTargetType
CevimelineMuscarinic acetylcholine receptor M1target
CevimelineMuscarinic acetylcholine receptor M3target
CevimelineCytochrome P450 3A4enzyme
CevimelineCytochrome P450 2D6enzyme
CevimelineDimethylaniline monooxygenase [N-oxide-forming] 1enzyme
CarbamoylcholineMuscarinic acetylcholine receptor M1target
CarbamoylcholineMuscarinic acetylcholine receptor M2target
CarbamoylcholineNeuronal acetylcholine receptor subunit alpha-2target
CarbamoylcholineCytosolic phospholipase A2enzyme
CarbamoylcholineMuscarinic acetylcholine receptor M3target
CarbamoylcholineMuscarinic acetylcholine receptor M4target
CarbamoylcholineAcetylcholinesteraseenzyme
PilocarpineMuscarinic acetylcholine receptor M1target
PilocarpineMuscarinic acetylcholine receptor M2target
PilocarpineCytochrome P450 2A6enzyme
PilocarpineMuscarinic acetylcholine receptor M3target
PilocarpineCytochrome P450 3A4enzyme
PilocarpineMuscarinic acetylcholine receptor M4target
PilocarpineMuscarinic acetylcholine receptor M5target
PilocarpineSerum paraoxonase/arylesterase 1enzyme
AcetylcholineSolute carrier family 22 member 5transporter
AcetylcholineSolute carrier family 22 member 1transporter
AcetylcholineMuscarinic acetylcholine receptor M1target
AcetylcholineMuscarinic acetylcholine receptor M2target
AcetylcholineMuscarinic acetylcholine receptor M3target
AcetylcholineMuscarinic acetylcholine receptor M4target
AcetylcholineNeuronal acetylcholine receptor subunit alpha-7target
AcetylcholineAcetylcholinesteraseenzyme
AcetylcholineCholinesteraseenzyme
MethacholineMuscarinic acetylcholine receptor M3target
MethacholineMuscarinic acetylcholine receptor M2target
MethacholineMuscarinic acetylcholine receptor M1target
MethacholineMuscarinic acetylcholine receptor M4target
MethacholineMuscarinic acetylcholine receptor M5target
MethacholineSolute carrier family 22 member 5transporter
VareniclineNeuronal acetylcholine receptor subunit alpha-4target
VareniclineNeuronal acetylcholine receptor subunit alpha-7target
VareniclineNeuronal acetylcholine receptor subunit alpha-3target
VareniclineNeuronal acetylcholine receptor subunit alpha-6target
VareniclineNeuronal acetylcholine receptor subunit beta-2target
VareniclineSolute carrier family 22 member 2transporter