Ergot-derivative Dopamine Receptor Agonists

Name
Ergot-derivative Dopamine Receptor Agonists
Accession Number
DBCAT003643
Description

Not Available

Drugs
DrugDrug Description
BromocriptineA dopamine D2 receptor agonist used for the treatment of galactorrhea due to hyperprolactinemia and other prolactin-related conditions, as well as in early Parkinsonian Syndrome.
CabergolineA dopamine receptor agonist used for the treatment of hyperprolactinemic conditions due to various causes.
DihydroergocornineA nootropic with an unknown mechanism of action indicated in individuals over sixty who manifest signs and symptoms of an idiopathic decline in mental capacity.
DihydroergocryptineA dopamine agonist indicated in the treatment of cerebrovascular diseases and atherosclerosis.
DihydroergotamineAn ergot alkaloid used in the acute treatment of migraine headache and cluster headache.
Ergoloid mesylateA nootropic with an unknown mechanism of action indicated in individuals over sixty who manifest signs and symptoms of an idiopathic decline in mental capacity.
LisurideFor the management of Parkinson's Disease
MetergolineAn ergot-derivative that acts as an antagonist at certain 5-HT receptor subtypes and as an agonist at dopamine receptors. It is often used in situations where inhibition of prolactin is desirable.
PergolideA long-acting dopamine agonist that is uncommonly used for the management of Parkinson's disease, due to the risk for cardiac valvulopathy.
Drugs & Drug Targets
DrugTargetType
BromocriptineD(1B) dopamine receptortarget
BromocriptineATP-dependent translocase ABCB1transporter
Bromocriptine5-hydroxytryptamine receptor 7target
BromocriptineAlpha-1D adrenergic receptortarget
BromocriptineAlpha-1B adrenergic receptortarget
BromocriptineAlpha-1A adrenergic receptortarget
BromocriptineD(1A) dopamine receptortarget
Bromocriptine5-hydroxytryptamine receptor 2Ctarget
Bromocriptine5-hydroxytryptamine receptor 1Btarget
Bromocriptine5-hydroxytryptamine receptor 2Atarget
BromocriptineD(4) dopamine receptortarget
Bromocriptine5-hydroxytryptamine receptor 2Btarget
BromocriptineAlpha-2B adrenergic receptortarget
BromocriptineAlpha-2C adrenergic receptortarget
Bromocriptine5-hydroxytryptamine receptor 1Atarget
BromocriptineD(3) dopamine receptortarget
BromocriptineAlpha-2A adrenergic receptortarget
Bromocriptine5-hydroxytryptamine receptor 1Dtarget
BromocriptineCytochrome P450 3A4enzyme
BromocriptineD(2) dopamine receptortarget
CabergolineBeta-2 adrenergic receptortarget
CabergolineD(1) dopamine receptortarget
CabergolineATP-dependent translocase ABCB1transporter
CabergolineBeta-1 adrenergic receptortarget
CabergolineAlpha-1D adrenergic receptortarget
CabergolineAlpha-1B adrenergic receptortarget
CabergolineAlpha-1A adrenergic receptortarget
Cabergoline5-hydroxytryptamine receptor 7target
CabergolineCytochrome P450 3A4enzyme
Cabergoline5-hydroxytryptamine receptor 2Ctarget
Cabergoline5-hydroxytryptamine receptor 1Btarget
CabergolineD(1A) dopamine receptortarget
CabergolineD(1B) dopamine receptortarget
CabergolineAlpha-2C adrenergic receptortarget
Cabergoline5-hydroxytryptamine receptor 1Atarget
CabergolineAlpha-2A adrenergic receptortarget
CabergolineD(2) dopamine receptortarget
CabergolineD(4) dopamine receptortarget
Cabergoline5-hydroxytryptamine receptor 1Dtarget
CabergolineAlpha-2B adrenergic receptortarget
Cabergoline5-hydroxytryptamine receptor 2Atarget
CabergolineD(3) dopamine receptortarget
Cabergoline5-hydroxytryptamine receptor 2Btarget
DihydroergocornineCytochrome P450 3A4enzyme
DihydroergocornineAlpha adrenergic receptortarget
DihydroergocornineBeta adrenergic receptortarget
DihydroergocornineSerotonin Receptorstarget
Dihydroergocryptine5-hydroxytryptamine receptor 2Btarget
Dihydroergocryptine5-hydroxytryptamine receptor 7target
DihydroergocryptineCytochrome P450 3A4enzyme
Dihydroergotamine5-hydroxytryptamine receptor 2Ctarget
DihydroergotamineBeta-3 adrenergic receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 4target
Dihydroergotamine5-hydroxytryptamine receptor 1Ftarget
DihydroergotamineD(4) dopamine receptortarget
DihydroergotamineD(3) dopamine receptortarget
DihydroergotamineD(2) dopamine receptortarget
DihydroergotamineAlpha-2 adrenergic receptorstarget
DihydroergotamineAlpha-1 adrenergic receptorstarget
Dihydroergotamine5-hydroxytryptamine receptor 1Dtarget
Dihydroergotamine5-hydroxytryptamine receptor 1Btarget
DihydroergotamineCytochrome P450 3A4enzyme
DihydroergotamineAlpha-2A adrenergic receptortarget
Dihydroergotamine5-hydroxytryptamine receptor 2Btarget
DihydroergotamineATP-dependent translocase ABCB1transporter
Dihydroergotamine5-hydroxytryptamine receptor 1Atarget
Dihydroergotamine5-hydroxytryptamine receptor 1Etarget
Dihydroergotamine5-hydroxytryptamine receptor 2Atarget
Ergoloid mesylateDopamine receptortarget
Ergoloid mesylateBeta adrenergic receptortarget
Ergoloid mesylateSerotonin Receptorstarget
Ergoloid mesylateAlpha adrenergic receptortarget
Ergoloid mesylateCytochrome P450 3A4enzyme
Lisuride5-hydroxytryptamine receptor 7target
LisurideCytochrome P450 3A4enzyme
Lisuride5-hydroxytryptamine receptor 1Btarget
LisurideD(1B) dopamine receptortarget
Lisuride5-hydroxytryptamine receptor 2Ctarget
LisurideD(4) dopamine receptortarget
Lisuride5-hydroxytryptamine receptor 2Atarget
Lisuride5-hydroxytryptamine receptor 2Btarget
Lisuride5-hydroxytryptamine receptor 1Dtarget
LisurideD(3) dopamine receptortarget
LisurideAlpha-2C adrenergic receptortarget
LisurideAlpha-2B adrenergic receptortarget
LisurideAlpha-2A adrenergic receptortarget
LisurideD(2) dopamine receptortarget
Lisuride5-hydroxytryptamine receptor 1Atarget
LisurideD(1A) dopamine receptortarget
Metergoline5-hydroxytryptamine receptor 1Ftarget
MetergolineSodium channel protein type 2 subunit alphatarget
Metergoline5-hydroxytryptamine receptor 2Ctarget
Metergoline5-hydroxytryptamine receptor 1Btarget
Metergoline5-hydroxytryptamine receptor 1Etarget
Metergoline5-hydroxytryptamine receptor 2Atarget
Metergoline5-hydroxytryptamine receptor 5Atarget
Metergoline5-hydroxytryptamine receptor 1Dtarget
Metergoline5-hydroxytryptamine receptor 2Btarget
PergolideCytochrome P450 3A4enzyme
PergolideD(2) dopamine receptortarget
PergolideD(1A) dopamine receptortarget
PergolideD(3) dopamine receptortarget
Pergolide5-hydroxytryptamine receptor 1Atarget
PergolideAlpha-1A adrenergic receptortarget
PergolideAlpha-2 adrenergic receptorstarget
PergolideAlpha-1B adrenergic receptortarget
PergolideAlpha-1D adrenergic receptortarget
PergolideD(4) dopamine receptortarget
PergolideD(1B) dopamine receptortarget
Pergolide5-hydroxytryptamine receptor 1Btarget
Pergolide5-hydroxytryptamine receptor 1Dtarget
Pergolide5-hydroxytryptamine receptor 2Atarget
Pergolide5-hydroxytryptamine receptor 2Btarget
PergolideDopamine receptortarget
Pergolide5-hydroxytryptamine receptor 2Ctarget