Reverse Transcriptase Inhibitors

Name
Reverse Transcriptase Inhibitors
Accession Number
DBCAT000594
Description

Inhibitors of reverse transcriptase (RNA-DIRECTED DNA POLYMERASE), an enzyme that synthesizes DNA on an RNA template.

Drugs
DrugDrug Description
AbacavirAn antiviral nucleoside reverse transcriptase inhibitor used in combination with other antiretrovirals for the treatment of HIV.
AdefovirNot Annotated
Adefovir dipivoxilA nucleotide analog used to treat chronic hepatitis B.
Ammonium trichlorotellurateAmmonium trichlorotellurate is an investigational compound with anti-tumour and anti-inflammatory properties.
Arsanilic acidAn arsenical which has been used as a feed additive for enteric conditions in pigs and poultry. It causes blindness and is ototoxic and nephrotoxic in animals. [PubChem]
AtevirdineAtevirdine has been used in trials studying the treatment of HIV Infections.
CapravirineInvestigated for use/treatment in acquired immune deficiency syndrome (AIDS) and aids-related infections and HIV infection.
CensavudineCensavudine has been used in trials studying the treatment of HIV-1 Infection.
DelavirdineA non-nucleoside reverse transcriptase inhibitor used to treat HIV infection.
DexelvucitabineDexelvucitabine has been used in trials studying the treatment of HIV Infections and Human Immunodeficiency Virus.
DidanosineA reverse transcriptase inhibitor used to treat HIV.
EfavirenzA non-nucleoside reverse transcriptase inhibitor used to treat HIV infection or prevent the spread of HIV.
ElvucitabineInvestigated for use/treatment in hepatitis (viral, B) and HIV infection.
EmivirineEmivirine has been used in trials studying the treatment of HIV Infections.
EmtricitabineA nucleoside reverse transcriptase inhibitor used for the treatment and prophylaxis of HIV.
EtravirineA non-nucleoside reverse transcriptase inhibitor (NNRTI) used in the treatment of HIV-1 infections in combination with other antiretroviral agents.
FoscarnetAn antiviral used to treat CMV, HIV, and HSV infections.
IslatravirA nucleoside analog reverse transcriptase inhibitor (NRTI) indicated in combination with doravirine for the treatment of HIV-1 infection in virologically-suppressed adults on a stable antiretroviral regimen.
LamivudineA reverse transcriptase inhibitor used to treat HIV and hepatitis B infections.
LapachoneLapachone has been used in trials studying the treatment of Cancer, Carcinoma, Advanced Solid Tumors, Head and Neck Neoplasms, and Carcinoma, Squamous Cell.
LobucavirLobucavir has been used in trials studying the treatment of HIV Infections and Cytomegalovirus Infections.
NevirapineA non-nucleoside reverse transcriptase inhibitor used as part of a management regimen for HIV-1 virus infection.
OltiprazOltipraz has been used in trials studying the treatment and prevention of Lung Cancer, Liver Fibrosis, Liver Cirrhosis, and Non-alcoholic Fatty Liver Disease.
PenciclovirA topical nucleoside polymerase inhibitor used in the treatment of recurrent herpes labialis.
Phosphonoacetic AcidA simple organophosphorus compound that inhibits DNA polymerase, especially in viruses and is used as an antiviral agent. [PubChem]
R-82913Not Available
RilpivirineA non-nucleoside reverse transcriptase inhibitor (NNRTI) used in combination with other antiretrovirals to specifically treat human immunodeficiency virus type 1 (HIV-1).
Rovafovir etalafenamideRovafovir etalafenamide is under investigation in clinical trial NCT03472326 (Efficacy of GS-9131 Functional Monotherapy in HIV-1-Infected Adults Failing a Nucleos(t)Ide Reverse Transcriptase Inhibitor-Containing Regimen).
StavudineA dideoxynucleoside used in the treatment of HIV infection.
TenofovirA nucleotide analog indicated in the treatment of HIV infections.
Tenofovir disoproxilA nucleotide analog reverse transcriptase inhibitor used in the treatment of Hepatitis B infection and used in the management of HIV-1 infection.
UlonivirineNot Available
ZalcitabineA dideoxynucleoside used to treat HIV.
ZidovudineA dideoxynucleoside used in the treatment of HIV infection.
Drugs & Drug Targets
DrugTargetType
AbacavirAlcohol dehydrogenase 6enzyme
AbacavirUDP-glucuronosyltransferase 1A1enzyme
AbacavirReverse transcriptase/RNaseHtarget
AbacavirAdenosine kinaseenzyme
AbacavirGag-Pol polyproteintarget
AdefovirDNA polymerase catalytic subunittarget
AdefovirProtein Ptarget
Adefovir dipivoxilNucleoside diphosphate kinase Benzyme
Adefovir dipivoxilNucleoside diphosphate kinase Aenzyme
Adefovir dipivoxilAdenylate kinase 4, mitochondrialenzyme
Adefovir dipivoxilAdenylate kinase 2, mitochondrialenzyme
Adefovir dipivoxilSolute carrier family 22 member 3transporter
Adefovir dipivoxilATP-binding cassette sub-family C member 5transporter
Adefovir dipivoxilATP-binding cassette sub-family C member 4transporter
Adefovir dipivoxilSolute carrier family 22 member 6transporter
Adefovir dipivoxilProtein Ptarget
Ammonium trichlorotellurateCaspase-1target
Ammonium trichlorotellurateCaspase-3target
Ammonium trichlorotellurateGTPase HRastarget
Ammonium trichlorotellurateVLA-4 (very late antigen-4)target
Ammonium trichlorotellurateInterleukin-10target
Arsanilic acidLysozyme Ctarget
AtevirdineGag-Pol polyproteintarget
AtevirdineReverse transcriptase/RNaseHtarget
CapravirineCytochrome P450 3A4enzyme
CapravirineGag-Pol polyproteintarget
CapravirineCytochrome P450 2C8enzyme
CapravirineCytochrome P450 2C9enzyme
CapravirineCytochrome P450 2C19enzyme
CapravirineReverse transcriptase/RNaseHtarget
CapravirineGag-Pol polyproteintarget
CensavudineReverse transcriptase/RNaseHtarget
CensavudineGag-Pol polyproteintarget
DelavirdineGag-Pol polyproteintarget
DelavirdineCytochrome P450 3A4enzyme
DelavirdineCytochrome P450 2C9enzyme
DelavirdineCytochrome P450 2D6enzyme
DelavirdineCytochrome P450 3A5enzyme
DelavirdineCytochrome P450 3A7enzyme
DelavirdineReverse transcriptase/RNaseHtarget
DelavirdineCytochrome P450 2C19enzyme
DexelvucitabineReverse transcriptase/RNaseHtarget
DidanosineEquilibrative nucleoside transporter 2transporter
DidanosineEquilibrative nucleoside transporter 1transporter
DidanosineReverse transcriptase/RNaseHtarget
DidanosinePurine nucleoside phosphorylasetarget
DidanosineSolute carrier family 22 member 6transporter
DidanosineGag-Pol polyproteintarget
DidanosineAlbumincarrier
EfavirenzCytochrome P450 1A2enzyme
EfavirenzAlbumincarrier
EfavirenzGag-Pol polyproteintarget
EfavirenzSolute carrier family 22 member 1transporter
EfavirenzBile salt export pumptransporter
EfavirenzUDP-glucuronosyltransferase 1A1enzyme
EfavirenzCytochrome P450 2B6enzyme
EfavirenzCytochrome P450 3A4enzyme
EfavirenzCytochrome P450 2C19enzyme
EfavirenzCytochrome P450 2C9enzyme
EfavirenzCytochrome P450 3A7enzyme
EfavirenzCytochrome P450 2D6enzyme
EfavirenzReverse transcriptase/RNaseHtarget
EfavirenzCytochrome P450 2C8enzyme
EfavirenzCytochrome P450 3A5enzyme
ElvucitabineGag-Pol polyproteintarget
ElvucitabineReverse transcriptase/RNaseHtarget
EmivirineReverse transcriptase/RNaseHtarget
EmivirineGag-Pol polyproteintarget
EmivirineGag-Pol polyproteintarget
EmtricitabineDeoxycytidine kinaseenzyme
EmtricitabineAlbumincarrier
EmtricitabineGag-Pol polyproteintarget
EmtricitabineMultidrug and toxin extrusion protein 1transporter
EmtricitabineReverse transcriptase/RNaseHtarget
EtravirineCytochrome P450 3A4enzyme
EtravirineGag-Pol polyproteintarget
EtravirineGag-Pol polyproteintarget
EtravirineATP-dependent translocase ABCB1transporter
EtravirinePhosphatidylcholine translocator ABCB4transporter
EtravirineReverse transcriptase/RNaseHtarget
EtravirineCytochrome P450 2C9enzyme
EtravirineCytochrome P450 2C19enzyme
FoscarnetMonocarboxylate transporter 1transporter
FoscarnetDNA polymerase catalytic subunittarget
FoscarnetDNA polymerase catalytic subunittarget
FoscarnetSolute carrier family 22 member 6transporter
IslatravirReverse transcriptase/RNaseHtarget
IslatravirBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LamivudineATP-binding cassette sub-family C member 4transporter
LamivudineDNAtarget
LamivudineProtein Ptarget
LamivudineMultidrug resistance-associated protein 1transporter
LamivudineSolute carrier family 22 member 6transporter
LamivudineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
LamivudineReverse transcriptase/RNaseHtarget
LamivudineSolute carrier family 22 member 1transporter
LamivudineSolute carrier family 22 member 2transporter
LamivudineSolute carrier family 22 member 3transporter
LamivudineDeoxycytidine kinaseenzyme
LamivudineUMP-CMP kinaseenzyme
LamivudinePhosphoglycerate kinase 1enzyme
LamivudineNucleoside diphosphate kinase Aenzyme
LamivudineNucleoside diphosphate kinase Benzyme
LamivudineCholine-phosphate cytidylyltransferase Aenzyme
LamivudineEthanolamine-phosphate cytidylyltransferaseenzyme
LamivudineATP-dependent translocase ABCB1transporter
LamivudineGag-Pol polyproteintarget
LamivudineATP-binding cassette sub-family C member 3transporter
LamivudineATP-binding cassette sub-family C member 2transporter
Lamivudine5'(3')-deoxyribonucleotidase, cytosolic typeenzyme
LamivudineAlbumincarrier
LapachoneRetinol-binding protein 3target
LapachoneDNA topoisomerase 1target
LobucavirGag-Pol polyproteintarget
NevirapineCytochrome P450 3A4enzyme
NevirapineCytochrome P450 2B6enzyme
NevirapineCytochrome P450 3A5enzyme
NevirapineCytochrome P450 2C9enzyme
NevirapineCytochrome P450 2A6enzyme
NevirapineCytochrome P450 2D6enzyme
NevirapineReverse transcriptase/RNaseHtarget
NevirapineAlbumincarrier
NevirapineCytochrome P450 1A2enzyme
NevirapineSolute carrier family 22 member 1transporter
NevirapineCytochrome P450 3A7enzyme
NevirapineGag-Pol polyproteintarget
OltiprazProtein-glutamine gamma-glutamyltransferase 2target
PenciclovirDNA polymerase catalytic subunittarget
PenciclovirThymidine kinasetarget
PenciclovirThymidine kinase, cytosolictarget
Phosphonoacetic AcidAlkaline phosphatasetarget
R-82913Gag-Pol polyproteintarget
R-82913Gag-Pol polyproteintarget
RilpivirineCytochrome P450 2B6enzyme
RilpivirineCytochrome P450 2E1enzyme
RilpivirineSodium channel protein type 10 subunit alphatarget
RilpivirineGag-Pol polyproteintarget
RilpivirineCytochrome P450 2C8enzyme
RilpivirineCytochrome P450 2C9enzyme
RilpivirineCytochrome P450 2D6enzyme
RilpivirineAlbumincarrier
RilpivirineSolute carrier organic anion transporter family member 1B3transporter
RilpivirineSolute carrier organic anion transporter family member 1B1transporter
RilpivirineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RilpivirineATP-dependent translocase ABCB1transporter
RilpivirineCytochrome P450 2C19enzyme
RilpivirineNuclear receptor subfamily 1 group I member 2target
RilpivirineReverse transcriptase/RNaseHtarget
RilpivirineCytochrome P450 3A4enzyme
Rovafovir etalafenamideReverse transcriptase/RNaseHtarget
StavudineGag-Pol polyproteintarget
StavudineAlbumincarrier
StavudineSodium/nucleoside cotransporter 1transporter
StavudineReverse transcriptase/RNaseHtarget
StavudineSolute carrier family 22 member 6transporter
TenofovirNucleoside diphosphate kinase Benzyme
TenofovirNucleoside diphosphate kinase Aenzyme
TenofovirATP-binding cassette sub-family C member 4transporter
TenofovirOrganic anion transporter 3transporter
TenofovirSolute carrier family 22 member 6transporter
TenofovirATP-dependent translocase ABCB1transporter
TenofovirAdenylate kinase isoenzyme 1enzyme
TenofovirAdenylate kinase 2, mitochondrialenzyme
TenofovirReverse transcriptase/RNaseHtarget
TenofovirGag-Pol polyproteintarget
TenofovirReverse transcriptasetarget
TenofovirDNA polymerasetarget
TenofovirAlbumincarrier
Tenofovir disoproxilReverse transcriptase/RNaseHtarget
Tenofovir disoproxilATP-binding cassette sub-family C member 2transporter
Tenofovir disoproxilATP-binding cassette sub-family C member 4transporter
Tenofovir disoproxilATP-binding cassette sub-family C member 10transporter
Tenofovir disoproxilOrganic anion transporter 3transporter
Tenofovir disoproxilSolute carrier family 22 member 6transporter
Tenofovir disoproxilAdenylate kinase 2, mitochondrialenzyme
Tenofovir disoproxilAdenylate kinase 4, mitochondrialenzyme
Tenofovir disoproxilATP-dependent translocase ABCB1transporter
Tenofovir disoproxilNucleoside diphosphokinaseenzyme
Tenofovir disoproxilCreatine Kinasesenzyme
Tenofovir disoproxilProtein Ptarget
Tenofovir disoproxilGag-Pol polyproteintarget
UlonivirineReverse transcriptase/RNaseHtarget
ZalcitabineSolute carrier family 22 member 7transporter
ZalcitabineReverse transcriptase/RNaseHtarget
ZalcitabineDeoxycytidine kinaseenzyme
ZalcitabineEquilibrative nucleoside transporter 1transporter
ZalcitabineEquilibrative nucleoside transporter 2transporter
ZalcitabineAlbumincarrier
ZalcitabineGag-Pol polyproteintarget
ZalcitabineSolute carrier family 22 member 6transporter
ZidovudineEquilibrative nucleoside transporter 2transporter
ZidovudineCytochrome P450 2A6enzyme
ZidovudineOrganic anion transporter 3transporter
ZidovudineSolute carrier family 22 member 7transporter
ZidovudineCytochrome P450 2C9enzyme
ZidovudineSolute carrier family 22 member 6transporter
ZidovudineSodium/nucleoside cotransporter 1transporter
ZidovudineATP-dependent translocase ABCB1transporter
ZidovudineATP-binding cassette sub-family C member 4transporter
ZidovudineATP-binding cassette sub-family C member 5transporter
ZidovudineBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
ZidovudineTelomerase reverse transcriptasetarget
ZidovudineThymidine kinase, cytosolicenzyme
ZidovudineUDP-glucuronosyltransferase 2B7enzyme
ZidovudineUDP-glucuronosyltransferase 1A1enzyme
ZidovudineGag-Pol polyproteintarget
ZidovudineReceptor-type tyrosine-protein kinase FLT3target
ZidovudineSolute carrier family 22 member 2transporter
ZidovudineReverse transcriptase/RNaseHtarget
ZidovudineCytochrome P450 3A4enzyme
ZidovudineAlbumincarrier
ZidovudineSolute carrier family 22 member 11transporter