R107474
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Explore a selection of our essential drug information below, or:
Identification
- Generic Name
- R107474
- DrugBank Accession Number
- DB06553
- Background
Not Available
- Type
- Small Molecule
- Groups
- Investigational
- Structure
- Weight
- Average: 359.429
Monoisotopic: 359.163376928 - Chemical Formula
- C22H21N3O2
- Synonyms
- 3-(2-(3,4-Dihydrobenzofuro(3,2-c)pyridin-2(1H)-yl)ethyl)-2-methyl-4H-pyrido(1,2-a)pyrimidin-4-one
- 3-[2-(3,4-dihydro-1H-[1]benzofuro[3,2-c]pyridin-2-yl)ethyl]-2-methylpyrido[1,2-a]pyrimidin-4-one
- Lusaperidone
- External IDs
- CS-7154
- DA-75161
- G13590
- HY-U00117
- MS-25665
- R107474
Pharmacology
- Indication
Investigated for use/treatment in depression.
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- Pharmacodynamics
Not Available
- Mechanism of action
- Not Available
- Absorption
Not Available
- Volume of distribution
Not Available
- Protein binding
Not Available
- Metabolism
- Not Available
- Route of elimination
Not Available
- Half-life
Not Available
- Clearance
Not Available
- Adverse Effects
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- Toxicity
Not Available
- Pathways
- Not Available
- Pharmacogenomic Effects/ADRs
- Not Available
Interactions
- Drug Interactions
- This information should not be interpreted without the help of a healthcare provider. If you believe you are experiencing an interaction, contact a healthcare provider immediately. The absence of an interaction does not necessarily mean no interactions exist.Not Available
- Food Interactions
- Not Available
Categories
- Drug Categories
- Not Available
- Classification
- Not classified
- Affected organisms
- Not Available
Chemical Identifiers
- UNII
- 5KTD2O86CB
- CAS number
- 214548-46-6
- InChI Key
- ZYXHQIPQIKTEDI-UHFFFAOYSA-N
- InChI
- InChI=1S/C22H21N3O2/c1-15-16(22(26)25-11-5-4-8-21(25)23-15)9-12-24-13-10-20-18(14-24)17-6-2-3-7-19(17)27-20/h2-8,11H,9-10,12-14H2,1H3
- IUPAC Name
- SMILES
- CC1=C(CCN2CCC3=C(C2)C2=C(O3)C=CC=C2)C(=O)N2C=CC=CC2=N1
References
- General References
- Not Available
- External Links
- ChemSpider
- 2308142
- BindingDB
- 50403744
- ChEMBL
- CHEMBL162501
- ZINC
- ZINC000001903948
Clinical Trials
- Clinical Trials
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Pharmacoeconomics
- Manufacturers
- Not Available
- Packagers
- Not Available
- Dosage Forms
- Not Available
- Prices
- Not Available
- Patents
- Not Available
Properties
- State
- Solid
- Experimental Properties
- Not Available
- Predicted Properties
Property Value Source - Predicted ADMET Features
- Not Available
Spectra
- Mass Spec (NIST)
- Not Available
- Spectra
- Not Available
- Chromatographic Properties
Collision Cross Sections (CCS)
Not Available
Drug created at March 19, 2008 16:36 / Updated at July 31, 2024 09:44