| DB00800 | Fenoldopam | approved | unknown | antagonist | Details |
| DB01392 | Yohimbine | approved, investigational, vet_approved | yes | antagonist | Details |
| DB00484 | Brimonidine | approved | yes | agonist | Details |
| DB00368 | Norepinephrine | approved | yes | agonist | Details |
| DB04855 | Dronedarone | approved | yes | antagonist | Details |
| DB05461 | OPC-28326 | investigational | unknown | | Details |
| DB05492 | Epicept NP-1 | investigational | unknown | | Details |
| DB06262 | Droxidopa | approved, investigational | yes | agonist | Details |
| DB06216 | Asenapine | approved | unknown | antagonist | Details |
| DB06229 | Ocaperidone | investigational | unknown | | Details |
| DB00575 | Clonidine | approved | yes | agonist | Details |
| DB01200 | Bromocriptine | approved, investigational, withdrawn | unknown | agonist | Details |
| DB00589 | Lisuride | approved, investigational | unknown | other/unknown | Details |
| DB00248 | Cabergoline | approved | unknown | antagonist | Details |
| DB00714 | Apomorphine | approved, investigational | unknown | agonist | Details |
| DB01267 | Paliperidone | approved | unknown | agonist | Details |
| DB01224 | Quetiapine | approved | unknown | antagonist | Details |
| DB00246 | Ziprasidone | approved | unknown | antagonist | Details |
| DB00363 | Clozapine | approved | no | antagonist | Details |
| DB01238 | Aripiprazole | approved, investigational | no | antagonistother/unknown | Details |
| DB01403 | Methotrimeprazine | approved, investigational | unknown | antagonist | Details |
| DB00925 | Phenoxybenzamine | approved | unknown | antagonist | Details |
| DB01363 | Ephedra sinica root | nutraceutical | yes | agonist | Details |
| DB01577 | Metamfetamine | approved, illicit, withdrawn | yes | agonist | Details |
| DB06694 | Xylometazoline | approved, investigational | unknown | agonist | Details |
| DB08815 | Lurasidone | approved, investigational | unknown | antagonist | Details |
| DB04946 | Iloperidone | approved | unknown | antagonist | Details |
| DB08838 | Agmatine | experimental | yes | agonist | Details |
| DB00408 | Loxapine | approved | unknown | binder | Details |
| DB01136 | Carvedilol | approved, investigational | unknown | antagonist | Details |
| DB00797 | Tolazoline | approved, vet_approved | unknown | binder | Details |
| DB00935 | Oxymetazoline | approved, investigational | unknown | agonist | Details |
| DB06148 | Mianserin | approved, investigational | unknown | antagonist | Details |
| DB09128 | Brexpiprazole | approved, investigational | unknown | antagonist | Details |
| DB11124 | Racepinephrine | approved | yes | agonist | Details |
| DB06153 | Pizotifen | approved | unknown | antagonist | Details |
| DB04846 | Celiprolol | approved, investigational | unknown | antagonist | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | no | | Details |
| DB00502 | Haloperidol | approved | unknown | | Details |
| DB00734 | Risperidone | approved, investigational | unknown | antagonist | Details |
| DB00696 | Ergotamine | approved | unknown | | Details |