| DB00246 | Ziprasidone | approved | unknown | antagonist | Details |
| DB00247 | Methysergide | approved | yes | antagonist | Details |
| DB06216 | Asenapine | approved | unknown | antagonist | Details |
| DB01200 | Bromocriptine | approved, investigational, withdrawn | unknown | antagonist | Details |
| DB00751 | Epinastine | approved, investigational | unknown | antagonist | Details |
| DB00363 | Clozapine | approved | unknown | antagonist | Details |
| DB01238 | Aripiprazole | approved, investigational | unknown | antagonistpartial agonist | Details |
| DB01224 | Quetiapine | approved | unknown | ligand | Details |
| DB00248 | Cabergoline | approved | unknown | antagonist | Details |
| DB06288 | Amisulpride | approved, investigational | yes | antagonist | Details |
| DB04946 | Iloperidone | approved | unknown | antagonist | Details |
| DB08815 | Lurasidone | approved, investigational | unknown | antagonist | Details |
| DB00477 | Chlorpromazine | approved, investigational, vet_approved | unknown | binder | Details |
| DB00408 | Loxapine | approved | unknown | binder | Details |
| DB00458 | Imipramine | approved | unknown | antagonist | Details |
| DB00543 | Amoxapine | approved | unknown | antagonist | Details |
| DB00988 | Dopamine | approved | unknown | binder | Details |
| DB00321 | Amitriptyline | approved | unknown | antagonist | Details |
| DB00934 | Maprotiline | approved, investigational | unknown | antagonist | Details |
| DB06148 | Mianserin | approved, investigational | unknown | antagonist | Details |
| DB09068 | Vortioxetine | approved, investigational | yes | antagonist | Details |
| DB00589 | Lisuride | approved, investigational | unknown | | Details |
| DB01267 | Paliperidone | approved | unknown | | Details |
| DB00434 | Cyproheptadine | approved | unknown | antagonist | Details |
| DB13988 | SB-269970 | investigational | unknown | antagonist | Details |
| DB09225 | Zotepine | approved, investigational, withdrawn | yes | antagonist | Details |
| DB04948 | Lofexidine | approved, investigational | no | agonist | Details |
| DB14185 | Aripiprazole lauroxil | approved, investigational | unknown | | Details |
| DB00502 | Haloperidol | approved | unknown | | Details |
| DB00924 | Cyclobenzaprine | approved | unknown | antagonist | Details |
| DB00734 | Risperidone | approved, investigational | unknown | antagonist | Details |
| DB00315 | Zolmitriptan | approved, investigational | no | agonist | Details |
| DB00953 | Rizatriptan | approved | unknown | agonist | Details |
| DB09128 | Brexpiprazole | approved, investigational | unknown | antagonist | Details |