Bexicaserin

This drug entry is a stub and has not been fully annotated. It is scheduled to be annotated soon.

Identification

Generic Name
Bexicaserin
DrugBank Accession Number
DB18885
Background

Bexicaserin is under investigation in clinical trial NCT05626634 (Open-label, Long-term Safety Study of LP352 in Subjects With Developmental and Epileptic Encephalopathy).

Type
Small Molecule
Groups
Investigational
Structure
Weight
Average: 295.334
Monoisotopic: 295.14961857
Chemical Formula
C15H19F2N3O
Synonyms
  • (7R)-N-(2,2-difluoroethyl)-7-methyl-1,2,3,4,6,7-hexahydro[1,4]diazepino[6,7,1-hi]indole-8-carboxamide
  • Bexicaserin
External IDs
  • LP352

Pharmacology

Indication

Not Available

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Contraindications & Blackbox Warnings
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Pharmacodynamics

Not Available

Mechanism of action
Not Available
Absorption

Not Available

Volume of distribution

Not Available

Protein binding

Not Available

Metabolism
Not Available
Route of elimination

Not Available

Half-life

Not Available

Clearance

Not Available

Adverse Effects
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Toxicity

Not Available

Pathways
Not Available
Pharmacogenomic Effects/ADRs
Not Available

Interactions

Drug Interactions
This information should not be interpreted without the help of a healthcare provider. If you believe you are experiencing an interaction, contact a healthcare provider immediately. The absence of an interaction does not necessarily mean no interactions exist.
Not Available
Food Interactions
Not Available

Categories

Drug Categories
Not Available
Classification
Not classified
Affected organisms
Not Available

Chemical Identifiers

UNII
R8XR1D6SCB
CAS number
2035818-24-5
InChI Key
KGOOOHQKLRUVSF-VIFPVBQESA-N
InChI
InChI=1S/C15H19F2N3O/c1-9-8-20-5-4-18-6-10-2-3-11(13(9)14(10)20)15(21)19-7-12(16)17/h2-3,9,12,18H,4-8H2,1H3,(H,19,21)/t9-/m0/s1
IUPAC Name
SMILES
C[C@H]1CN2CCNCC3=CC=C(C(=O)NCC(F)F)C1=C23

References

General References
Not Available
ChemSpider
129309383

Clinical Trials

Clinical Trials
Clinical Trial & Rare Diseases Add-on Data Package
Explore 4,000+ rare diseases, orphan drugs & condition pairs, clinical trial why stopped data, & more. Preview package
PhaseStatusPurposeConditionsCountStart DateWhy Stopped100+ additional columns
2Active Not RecruitingTreatmentDevelopmental and Epileptic Encephalopathy / Dravet Syndrome (DS) / Lennox-Gastaut Syndrome1somestatusstop reasonjust information to hide
1, 2CompletedTreatmentDevelopmental and Epileptic Encephalopathy / Dravet Syndrome (DS) / Lennox-Gastaut Syndrome1somestatusstop reasonjust information to hide
Not AvailableAvailableNot AvailableDevelopmental and Epileptic Encephalopathy / Dravet Syndrome (DS) / Lennox-Gastaut Syndrome1somestatusstop reasonjust information to hide

Pharmacoeconomics

Manufacturers
Not Available
Packagers
Not Available
Dosage Forms
Not Available
Prices
Not Available
Patents
Not Available

Properties

State
Not Available
Experimental Properties
Not Available
Predicted Properties
PropertyValueSource
Predicted ADMET Features
Not Available

Spectra

Mass Spec (NIST)
Not Available
Spectra
Not Available
Chromatographic Properties
Collision Cross Sections (CCS)
Not Available

Drug created at June 27, 2024 02:32 / Updated at June 28, 2024 04:46