Ankyrin repeat and protein kinase domain-containing protein 1
Details
- Name
- Ankyrin repeat and protein kinase domain-containing protein 1
- Synonyms
- 2.7.11.1
- PKK2
- Protein kinase PKK2
- SGK288
- Sugen kinase 288
- X-kinase
- Gene Name
- ANKK1
- UniProtKB Entry
- Q8NFD2Swiss-Prot
- Organism
- Humans
- NCBI Taxonomy ID
- 9606
- Amino acid sequence
>lcl|BSEQ0051700|Ankyrin repeat and protein kinase domain-containing protein 1 MAADPTELRLGSLPVFTRDDFEGDWRLVASGGFSQVFQARHRRWRTEYAIKCAPCLPPDA ASSDVNYLIEEAAKMKKIKFQHIVSIYGVCKQPLGIVMEFMANGSLEKVLSTHSLCWKLR FRIIHETSLAMNFLHSIKPPLLHLDLKPGNILLDSNMHVKISDFGLSKWMEQSTRMQYIE RSALRGMLSYIPPEMFLESNKAPGPKYDVYSFAIVIWELLTQKKPYSGFNMMMIIIRVAA GMRPSLQPVSDQWPSEAQQMVDLMKRCWDQDPKKRPCFLDITIETDILLSLLQSRVAVPE SKALARKVSCKLSLRQPGEVNEDISQELMDSDSGNYLKRALQLSDRKNLVPRDEELCIYE NKVTPLHFLVAQGSVEQVRLLLAHEVDVDCQTASGYTPLLIAAQDQQPDLCALLLAHGAD ANRVDEDGWAPLHFAAQNGDDGTARLLLDHGACVDAQEREGWTPLHLAAQNNFENVARLL VSRQADPNLHEAEGKTPLHVAAYFGHVSLVKLLTSQGAELDAQQRNLRTPLHLAVERGKV RAIQHLLKSGAVPDALDQSGYGPLHTAAARGKYLICKMLLRYGASLELPTHQGWTPLHLA AYKGHLEIIHLLAESHANMGALGAVNWTPLHLAARHGEEAVVSALLQCGADPNAAEQSGW TPLHLAVQRSTFLSVINLLEHHANVHARNKVGWTPAHLAALKGNTAILKVLVEAGAQLDV QDGVSCTPLQLALRSRKQGIMSFLEGKEPSVATLGGSKPGAEMEI
- Number of residues
- 765
- Molecular Weight
- 84631.68
- Theoretical pI
- Not Available
- GO Classification
- Functionsprotein serine kinase activityProcessesregulation of cell cycle processComponentscell projection / cytoplasm / nucleus
- General Function
- Not Available
- Specific Function
- ATP binding
- Pfam Domain Function
- Signal Regions
- Not Available
- Transmembrane Regions
- Not Available
- Cellular Location
- Not Available
- Gene sequence
>lcl|BSEQ0051701|Ankyrin repeat and protein kinase domain-containing protein 1 (ANKK1) ATGGCTGCCGACCCCACCGAGCTGCGGCTGGGCAGCCTCCCCGTCTTCACCCGCGACGAC TTCGAGGGCGACTGGCGCCTAGTGGCCAGCGGCGGCTTCAGCCAGGTGTTCCAGGCGCGG CACAGGCGCTGGCGGACGGAGTACGCCATCAAGTGCGCCCCCTGCCTTCCACCCGACGCC GCCAGCTCTGATGTGAATTACCTCATTGAAGAAGCTGCCAAAATGAAGAAGATCAAGTTT CAGCACATCGTGTCTATCTACGGGGTGTGCAAGCAGCCCCTGGGTATTGTGATGGAGTTT ATGGCCAACGGCTCCCTGGAGAAGGTGCTGTCCACCCACAGCCTCTGCTGGAAGCTCAGG TTCCGCATCATCCATGAGACCAGCTTGGCCATGAACTTCCTGCACAGCATTAAGCCGCCT CTGCTCCACCTGGACCTCAAGCCGGGCAACATACTCCTGGACAGCAACATGCATGTCAAA ATTTCAGACTTCGGCCTGTCCAAGTGGATGGAACAGTCCACCCGGATGCAGTACATCGAG AGGTCGGCTCTGCGGGGCATGCTCAGCTACATCCCCCCTGAGATGTTCCTGGAGAGTAAC AAGGCCCCAGGACCTAAATATGATGTGTACAGCTTTGCAATTGTCATCTGGGAGCTACTC ACTCAGAAGAAACCATACTCAGGGTTCAACATGATGATGATTATTATCCGAGTGGCGGCA GGCATGCGGCCCTCCCTACAGCCTGTCTCTGACCAATGGCCAAGCGAGGCCCAGCAGATG GTGGACCTGATGAAACGCTGCTGGGACCAGGACCCCAAGAAGAGGCCATGCTTTCTAGAC ATTACCATCGAGACAGACATACTGCTGTCACTGCTGCAGAGTCGTGTGGCAGTCCCAGAG AGCAAGGCCCTGGCCAGGAAGGTGTCCTGCAAGCTGTCGCTGCGCCAGCCCGGGGAGGTT AATGAGGACATCAGCCAGGAACTGATGGACAGTGACTCAGGAAACTACCTGAAGCGGGCC CTTCAGCTCTCCGACCGTAAGAATTTGGTCCCGAGAGATGAGGAACTGTGTATCTATGAG AACAAGGTCACCCCCCTCCACTTCCTGGTGGCCCAGGGCAGTGTGGAGCAGGTGAGGTTG CTGCTGGCCCACGAGGTAGACGTGGACTGCCAGACGGCCTCTGGATACACGCCCCTCCTG ATCGCCGCCCAGGACCAGCAACCCGACCTCTGTGCCCTGCTTTTGGCACATGGTGCTGAT GCCAACCGAGTGGATGAGGATGGCTGGGCCCCACTGCACTTTGCAGCCCAGAATGGGGAT GACGGCACTGCGCGCCTGCTCCTGGACCACGGGGCCTGTGTGGATGCCCAGGAACGTGAA GGGTGGACCCCTCTTCACCTGGCTGCACAGAATAACTTTGAGAATGTGGCACGGCTTCTG GTCTCCCGTCAGGCTGACCCCAACCTGCATGAGGCTGAGGGCAAGACCCCCCTCCATGTG GCCGCCTACTTTGGCCATGTTAGCCTGGTCAAGCTGCTGACCAGCCAGGGGGCTGAGTTG GATGCTCAGCAGAGAAACCTGAGAACACCACTGCACCTGGCAGTAGAGCGGGGCAAAGTG AGGGCCATCCAACACCTGCTGAAGAGTGGAGCGGTCCCTGATGCCCTTGACCAGAGCGGC TACGGCCCACTGCACACTGCAGCTGCCAGGGGCAAATACCTGATCTGCAAGATGCTGCTC AGGTACGGAGCCAGCCTTGAGCTGCCCACCCACCAGGGCTGGACACCCCTGCATCTAGCA GCCTACAAGGGCCACCTGGAGATCATCCATCTGCTGGCAGAGAGCCACGCAAACATGGGT GCTCTTGGAGCTGTGAACTGGACTCCCCTGCACCTAGCTGCACGCCACGGGGAGGAGGCG GTGGTGTCAGCACTGCTGCAGTGTGGGGCTGACCCCAATGCTGCAGAGCAGTCAGGCTGG ACACCCCTCCACCTGGCGGTCCAGAGGAGCACCTTCCTGAGTGTCATCAACCTCCTAGAA CATCACGCAAATGTCCACGCCCGCAACAAGGTGGGCTGGACACCCGCCCACCTGGCCGCC CTCAAGGGCAACACAGCCATCCTCAAAGTGCTGGTCGAGGCAGGCGCCCAGCTGGACGTC CAGGATGGAGTGAGCTGCACACCCCTGCAACTGGCCCTCCGCAGCCGAAAGCAGGGCATC ATGTCCTTCCTAGAGGGCAAGGAGCCGTCAGTGGCCACTCTGGGTGGTTCTAAGCCAGGA GCCGAGATGGAAATTTAG
- Chromosome Location
- 11
- Locus
- 11q23.2
- External Identifiers
Resource Link UniProtKB ID Q8NFD2 UniProtKB Entry Name ANKK1_HUMAN GeneCard ID ANKK1 HGNC ID HGNC:21027 KEGG ID hsa:255239 NCBI Gene ID 255239 - General References
- Neville MJ, Johnstone EC, Walton RT: Identification and characterization of ANKK1: a novel kinase gene closely linked to DRD2 on chromosome band 11q23.1. Hum Mutat. 2004 Jun;23(6):540-5. [Article]
- Dubertret C, Gouya L, Hanoun N, Deybach JC, Ades J, Hamon M, Gorwood P: The 3' region of the DRD2 gene is involved in genetic susceptibility to schizophrenia. Schizophr Res. 2004 Mar 1;67(1):75-85. [Article]
- Manning G, Whyte DB, Martinez R, Hunter T, Sudarsanam S: The protein kinase complement of the human genome. Science. 2002 Dec 6;298(5600):1912-34. [Article]
- Greenman C, Stephens P, Smith R, Dalgliesh GL, Hunter C, Bignell G, Davies H, Teague J, Butler A, Stevens C, Edkins S, O'Meara S, Vastrik I, Schmidt EE, Avis T, Barthorpe S, Bhamra G, Buck G, Choudhury B, Clements J, Cole J, Dicks E, Forbes S, Gray K, Halliday K, Harrison R, Hills K, Hinton J, Jenkinson A, Jones D, Menzies A, Mironenko T, Perry J, Raine K, Richardson D, Shepherd R, Small A, Tofts C, Varian J, Webb T, West S, Widaa S, Yates A, Cahill DP, Louis DN, Goldstraw P, Nicholson AG, Brasseur F, Looijenga L, Weber BL, Chiew YE, DeFazio A, Greaves MF, Green AR, Campbell P, Birney E, Easton DF, Chenevix-Trench G, Tan MH, Khoo SK, Teh BT, Yuen ST, Leung SY, Wooster R, Futreal PA, Stratton MR: Patterns of somatic mutation in human cancer genomes. Nature. 2007 Mar 8;446(7132):153-8. [Article]
Associated Data
- Bio-Entities
Bio-Entity Type Ankyrin repeat and protein kinase domain-containing protein 1 (Humans) protein primary- Drug Relations
Drug Drug group Pharmacological action? Type Actions Details Fostamatinib approved, investigational unknown target inhibitor Details