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Polyestradiol phosphate
go.drugbank.com/drugs/DB09369ApprovedPolymeric phosphoric acid ester of estradiol.
Synonyms: Estradiol phosphate polymer, Poly(estradiol phosphate)Categories: Estradiol CongenersFluoroestradiol F-18
go.drugbank.com/drugs/DB15690ApprovedInvestigationalFluoroestradiol F-18 is an imaging agent used with positron emission tomography (PET) to detect estrogen receptor-positive breast cancer lesions. … [L14117] It is expected to be available in late 2020/early 2021.[L14117]
Synonyms: 16-alpha-(18F)Fluoro-17beta-estradiol, 16alpha-(18F)Fluoro-17beta-estradiolCategories: Estradiol CongenersQuinestrol
go.drugbank.com/drugs/DB04575ApprovedThe 3-cyclopentyl ether of ethinyl estradiol.
Categories: Estradiol Congeners, Ethinyl EstradiolSynonyms: Estradiol-17-beta 3-cyclopentyl ether2-Hydroxyestradiol
go.drugbank.com/drugs/DB07706Experimental2-Hydroxyestradiol is classified as an endogenous steroid, catechol estrogen, and metabolite of estradiol. It is also a positional isomer of estriol. [A31630]
Categories: Estradiol CongenersSynonyms: 2-OH-Estradiol, 2-hydroxy-17β-estradiolAtrimustine
go.drugbank.com/drugs/DB21376ExperimentalAtrimustine is a small molecule drug. The usage of the INN stem '-mustine' in the name indicates that Atrimustine is a antineoplastic, alkylating agent, (β-chloroethyl) amine derivative.
Synonyms: Estradiol benzoate butyrateIK-930
go.drugbank.com/drugs/DB18149InvestigationalIK-930 is an oral, paralog-selective TEAD inhibitor.
2-Methoxyestradiol
go.drugbank.com/drugs/DB02342Investigational2-Methoxyestradiol (2ME2) is a drug that prevents the formation of new blood vessels that tumors need in order to grow (angiogenesis). … It has undergone Phase 1 clinical trials against breast cancers and preclinical studies suggest that 2ME2 could also be effective against inflammatory diseases such as rheumatoid arthritis.
Categories: Estradiol CongenersSynonyms: 2-methoxy-17β-estradiolEstradiol acetate Predicted Metabolism Pathway
smpdb.ca/view/SMP0174628MetabolicMetabolites of Estradiol acetate are predicted with biotransformer.
Estradiol benzoate Predicted Metabolism Pathway
smpdb.ca/view/SMP0174629MetabolicMetabolites of Estradiol benzoate are predicted with biotransformer.
Estriol
go.drugbank.com/drugs/DB04573ApprovedInvestigationalVet approvedA hydroxylated metabolite of estradiol or estrone that has a hydroxyl group at C3-beta, 16-alpha, and 17-beta position. Estriol is a major urinary estrogen. … Though estriol is used as part of the primarily North American phenomenon of bioidentical hormone replacement therapy, it is not approved for use by the FDA or Health Canada.
Synonyms: Estriol, 16α,17β-estriolCategories: Estradiol Congeners, estriol