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5-methoxy-N,N-dimethyltryptamine
go.drugbank.com/drugs/DB14010IllicitInvestigational5-methoxy-N,N-dimethyltryptamine (5-MeO-DMT) is a tryptamine with psychedelic properties. It is found in a wide variety of plant species, and a single psychoactive toad species, the Colorado River toad. This drug, as well as dimethyltryp...
Categories: Cytochrome P-450 Substrates, Cytochrome P-450 CYP2D6 SubstratesClinafloxacin
go.drugbank.com/drugs/DB14025ExperimentalClinafloxacin is a fluoroquinolone antibacterial currently under research. It has been proven to present good antibiotic properties. However, its approval and release have been halted due to the presence of serious side effects.
Categories: Cytochrome P-450 CYP1A2 Inhibitors, Cytochrome P-450 CYP2C19 InhibitorsMadecassic acid
go.drugbank.com/drugs/DB14037InvestigationalCategories: Cytochrome P-450 CYP2C9 Inhibitors, Cytochrome P-450 CYP2D6 InhibitorsValinomycin
go.drugbank.com/drugs/DB14057ExperimentalA cyclododecadepsipeptide ionophore antibiotic produced by Streptomyces fulvissimus and related to the enniatins. It is composed of 3 moles each of L-valine, D-alpha-hydroxyisovaleric acid, D-valine, and L-lactic acid linked alternately ...
Categories: P-glycoprotein inhibitors, P-glycoprotein substratesConcanamycin A
go.drugbank.com/drugs/DB14062ExperimentalConcanamycin A is an H+-ATPase (vacuolar) inhibitor.
Categories: P-glycoprotein inhibitorsTetrandrine
go.drugbank.com/drugs/DB14066InvestigationalCategories: P-glycoprotein inhibitors, Cytochrome P-450 SubstratesDofequidar
go.drugbank.com/drugs/DB14067InvestigationalDofequidar is an antineoplastic agent.
Categories: P-glycoprotein inhibitorsDesmethylsertraline
go.drugbank.com/drugs/DB14071ExperimentalDesmethylsertraline is a metabolite of sertraline.
Categories: P-glycoprotein inhibitorsReversin 121
go.drugbank.com/drugs/DB14072ExperimentalReversin 121 is a hydrophobic peptide chemosensitizer that can reverse P-glycoprotein-mediated multidrug resistance.
Categories: P-glycoprotein inhibitors