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JBI-802
go.drugbank.com/drugs/DB17399InvestigationalSynonyms: N-hydroxy-4-((4-((((1R,2S)-2-phenylcyclopropyl) amino)methyl)-1H-pyrazol-1-yl)methyl)benzamide hydrogen bromideRU82197
go.drugbank.com/drugs/DB03268ExperimentalSynonyms: 4-[2-Acetylamino-2-(1-biphenyl-4-ylmethyl-2-oxo-azepan-3-ylcarbamoyl)-ethyl]-2-formyl-benzoic acidGlucoraphanin
go.drugbank.com/drugs/DB15436InvestigationalGlucoraphanin is under investigation in clinical trial NCT01879878 (Pilot Study Evaluating Broccoli Sprouts in Advanced Pancreatic Cancer [POUDER Trial]).
Synonyms: 4-methylsulfinylbutyl glucosinolatePyroquilon
go.drugbank.com/drugs/DB02756ExperimentalPyroquilon is a commercial blasticide which binds in the naphthol pocket of fungal trihydroxynaphthalene reductase active site.
Synonyms: 1,2,5,6-tetrahydropyrrolo[3,2,1-ij]quinolin-4-oneCategories: Heterocyclic Compounds, 1-Ring, Heterocyclic Compounds, 2-RingLomeguatrib
go.drugbank.com/drugs/DB21175ExperimentalLomeguatrib is a small molecule drug. Lomeguatrib has a monoisotopic molecular weight of 324.96 Da.
Synonyms: O6-(4-Bromothenyl)guanine, PaTrin-2Categories: Heterocyclic Compounds, 2-RingGlyburide
go.drugbank.com/drugs/DB01016ApprovedInvestigational[A183617] Glyburide was granted FDA approval on 1 May 1984.[L8117] A formulation with metformin was granted FDA approval on on 31 July 2000.[L8120] … Glyburide is a second generation sulfonylurea used to treat patients with diabetes mellitus type II.
Synonyms: 5-chloro-N-(2-(4-((((cyclohexylamino)carbonyl)amino)sulfonyl)phenyl)ethyl)-2-methoxybenzamide, 1-((p-(2-(5-chloro-o-anisamido)ethyl)phenyl)sulfonyl)-3-cyclohexylureaMixtures: SIL-NORBORAL ® 5/500 MG, SIL - NORBORAL ® 5 MG / 1000 MGOlafertinib
go.drugbank.com/drugs/DB17179InvestigationalSynonyms: N-(3-(2-(2,3-difluoro-4-(4-(2-hydroxyethyl)piperazin-1-yl)phenylamino)quinazolin-8-yl)phenyl)acrylamideAVL-3288
go.drugbank.com/drugs/DB18707InvestigationalSynonyms: (z)-3-(4-chloroanilino)-n-(4-chlorophenyl)-2-(3-methylisoxazol-5-yl)prop-2-enamide(R)-Rolipram
go.drugbank.com/drugs/DB04149InvestigationalThe (R)-enantiomer of rolipram, it is a phosphodiesterase inhibitor with antidepressant properties.
Synonyms: (R)-4-(3-Cyclopentyloxy-4-methoxy-phenyl)-pyrrolidin-2-one, R-rolipram