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Madecassic acid
go.drugbank.com/drugs/DB14037InvestigationalCategories: Cytochrome P-450 CYP2C9 Inhibitors, Cytochrome P-450 CYP2D6 InhibitorsValinomycin
go.drugbank.com/drugs/DB14057ExperimentalIt is composed of 3 moles each of L-valine, D-alpha-hydroxyisovaleric acid, D-valine, and L-lactic acid linked alternately to form a 36-membered ring.
Categories: P-glycoprotein inhibitors, P-glycoprotein substratesConcanamycin A
go.drugbank.com/drugs/DB14062ExperimentalConcanamycin A is an H+-ATPase (vacuolar) inhibitor.
Categories: P-glycoprotein inhibitorsTetrandrine
go.drugbank.com/drugs/DB14066InvestigationalSynonyms: D-TetrandrineCategories: P-glycoprotein inhibitors, Cytochrome P-450 SubstratesDofequidar
go.drugbank.com/drugs/DB14067InvestigationalDofequidar is an antineoplastic agent.
Categories: P-glycoprotein inhibitorsDesmethylsertraline
go.drugbank.com/drugs/DB14071ExperimentalDesmethylsertraline is a metabolite of sertraline.
Categories: P-glycoprotein inhibitorsReversin 121
go.drugbank.com/drugs/DB14072ExperimentalReversin 121 is a hydrophobic peptide chemosensitizer that can reverse P-glycoprotein-mediated multidrug resistance.
Categories: P-glycoprotein inhibitorsCloprostenol
go.drugbank.com/drugs/DB11507ExperimentalVet approvedProducts: GESTAVET PROST (d-cloprostenol 75 mcg/ml solution for injection)