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Suzetrigine
go.drugbank.com/drugs/DB18927
ApprovedInvestigational
Suzetrigine is a NaV1.8 voltage-gated sodium channel blocker with analgesic properties NaV1.8 is abundantly expressed in peripheral sensory nerves to play a role in pain signal transmission, making it a desirable therapeutic target for treatment of pain. On January 30, 2025, suzetrigine was approved by the FDA as a ...
Acute, moderate Pain
go.drugbank.com/conditions/DBCOND0112012Severe Acute Pain
go.drugbank.com/conditions/DBCOND0021329