Targeting peroxisome proliferator-activated receptors (PPARs): development of modulators.

Article Details

Citation

Pirat C, Farce A, Lebegue N, Renault N, Furman C, Millet R, Yous S, Speca S, Berthelot P, Desreumaux P, Chavatte P

Targeting peroxisome proliferator-activated receptors (PPARs): development of modulators.

J Med Chem. 2012 May 10;55(9):4027-61. doi: 10.1021/jm101360s. Epub 2012 Feb 27.

PubMed ID
22260081 [ View in PubMed
]
Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
alpha-Linolenic acidPeroxisome proliferator-activated receptor gammaKd (nM)2000N/AN/ADetails
ClofibratePeroxisome proliferator-activated receptor alphaEC 50 (nM)55000N/AN/ADetails
GW-590735Peroxisome proliferator-activated receptor alphaEC 50 (nM)4N/AN/ADetails
IcosapentPeroxisome proliferator-activated receptor gammaKd (nM)2000N/AN/ADetails