| DB01039 | Fenofibrate | approved | yes | agonist | Details |
| DB01393 | Bezafibrate | approved, investigational | yes | agonist | Details |
| DB00636 | Clofibrate | approved, investigational | yes | agonist | Details |
| DB01241 | Gemfibrozil | approved | yes | agonist | Details |
| DB01890 | N,N-Bis(3-(D-gluconamido)propyl)deoxycholamide | experimental | unknown | | Details |
| DB04971 | Reglitazar | investigational | unknown | | Details |
| DB05187 | Elafibranor | investigational | unknown | | Details |
| DB06510 | Muraglitazar | investigational | unknown | | Details |
| DB06521 | Ertiprotafib | investigational | unknown | | Details |
| DB06533 | Ragaglitazar | investigational | unknown | | Details |
| DB06536 | Tesaglitazar | investigational | unknown | | Details |
| DB07215 | GW-590735 | investigational | unknown | | Details |
| DB07724 | Indeglitazar | experimental | unknown | | Details |
| DB08915 | Aleglitazar | investigational | yes | agonist | Details |
| DB00328 | Indomethacin | approved, investigational | unknown | agonist | Details |
| DB01708 | Prasterone | approved, investigational, nutraceutical | unknown | activator | Details |
| DB11133 | Omega-3 fatty acids | approved, nutraceutical | unknown | activator | Details |
| DB03756 | Doconexent | approved, investigational | yes | activator | Details |
| DB09422 | Soybean oil | approved | yes | activator | Details |
| DB11605 | Myrrh | approved | unknown | agonist | Details |
| DB00159 | Icosapent | approved, nutraceutical | unknown | | Details |
| DB03017 | Lauric acid | approved, experimental | unknown | | Details |
| DB08231 | Myristic acid | experimental | unknown | | Details |
| DB03796 | Palmitic Acid | approved | unknown | | Details |
| DB03193 | Stearic acid | approved, experimental | unknown | | Details |
| DB04557 | Arachidonic Acid | experimental | unknown | | Details |
| DB04224 | Oleic Acid | approved, investigational, vet_approved | unknown | | Details |
| DB00132 | alpha-Linolenic acid | approved, investigational, nutraceutical | unknown | | Details |
| DB09006 | Clinofibrate | experimental | unknown | | Details |
| DB00412 | Rosiglitazone | approved, investigational | unknown | | Details |
| DB00197 | Troglitazone | approved, investigational, withdrawn | unknown | | Details |
| DB12961 | Leukotriene B4 | investigational | unknown | activator | Details |
| DB09064 | Ciprofibrate | approved, investigational | unknown | | Details |
| DB04519 | Caprylic acid | investigational | unknown | | Details |
| DB05416 | Cardarine | investigational | unknown | agonist | Details |
| DB02746 | Phthalic Acid | experimental | unknown | | Details |
| DB02709 | Resveratrol | investigational | unknown | | Details |
| DB00313 | Valproic acid | approved, investigational | unknown | | Details |
| DB00573 | Fenoprofen | approved | unknown | activator | Details |
| DB02266 | Flufenamic acid | approved | unknown | activator | Details |
| DB01050 | Ibuprofen | approved | unknown | activator | Details |
| DB13873 | Fenofibric acid | approved | yes | agonist | Details |
| DB13961 | Fish oil | approved, nutraceutical | unknown | regulator | Details |
| DB12007 | Isoflavone | experimental | unknown | agonist | Details |
| DB09213 | Dexibuprofen | approved, investigational | unknown | | Details |
| DB01118 | Amiodarone | approved, investigational | unknown | agonist | Details |