| DB00398 | Sorafenib | approved, investigational | yes | antagonist | Details |
| DB01268 | Sunitinib | approved, investigational | yes | inhibitor | Details |
| DB12874 | Quizartinib | investigational | unknown | | Details |
| DB12742 | Amuvatinib | investigational | unknown | | Details |
| DB05014 | XL999 | investigational | unknown | | Details |
| DB05465 | Tandutinib | investigational | unknown | | Details |
| DB06080 | Linifanib | investigational | unknown | | Details |
| DB06469 | Lestaurtinib | investigational | unknown | | Details |
| DB06595 | Midostaurin | approved, investigational | yes | antagonistinhibitor | Details |
| DB08901 | Ponatinib | approved, investigational | unknown | inhibitor | Details |
| DB09079 | Nintedanib | approved | unknown | inhibitor | Details |
| DB12267 | Brigatinib | approved, investigational | unknown | inhibitor | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | inhibitor | Details |
| DB12141 | Gilteritinib | approved, investigational | yes | inhibitor | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | inhibitor | Details |
| DB12500 | Fedratinib | approved, investigational | yes | inhibitor | Details |
| DB15822 | Pralsetinib | approved, investigational | unknown | inhibitor | Details |
| DB11800 | Tivozanib | approved, investigational | unknown | inhibitor | Details |