| DB00216 | Eletriptan | approved, investigational | yes | agonist | Details |
| DB00669 | Sumatriptan | approved, investigational | yes | agonist | Details |
| DB00952 | Naratriptan | approved, investigational | yes | agonist | Details |
| DB00953 | Rizatriptan | approved | yes | agonist | Details |
| DB00315 | Zolmitriptan | approved, investigational | yes | agonist | Details |
| DB00247 | Methysergide | approved | unknown | binder | Details |
| DB00696 | Ergotamine | approved | unknown | agonist | Details |
| DB06148 | Mianserin | approved, investigational | unknown | binder | Details |
| DB11732 | Lasmiditan | approved, investigational | yes | agonist | Details |
| DB00320 | Dihydroergotamine | approved, investigational | yes | agonist | Details |