| DB00334 | Olanzapine | approved, investigational | unknown | substrate | Details |
| DB00250 | Dapsone | approved, investigational | unknown | substrate | Details |
| DB00675 | Tamoxifen | approved | unknown | substrate | Details |
| DB00582 | Voriconazole | approved | unknown | substrate | Details |
| DB00363 | Clozapine | approved | no | substrate | Details |
| DB01254 | Dasatinib | approved, investigational | unknown | substrate | Details |
| DB00918 | Almotriptan | approved, investigational | unknown | substrate | Details |
| DB00501 | Cimetidine | approved, investigational | unknown | substrate | Details |
| DB05294 | Vandetanib | approved | unknown | substrate | Details |
| DB11828 | Neratinib | approved, investigational | unknown | substrate | Details |
| DB12278 | Propiverine | approved, investigational | unknown | substrate | Details |
| DB00768 | Olopatadine | approved | no | substrate | Details |
| DB12500 | Fedratinib | approved, investigational | unknown | substrate | Details |
| DB00763 | Methimazole | approved | unknown | substrate | Details |
| DB13609 | Umifenovir | investigational | unknown | substrate | Details |
| DB15305 | Risdiplam | approved, investigational | unknown | substrate | Details |
| DB11886 | Infigratinib | approved, investigational | no | substrate | Details |
| DB12265 | Fexinidazole | approved, investigational | unknown | substrate | Details |