Carbamates

Name
Carbamates
Accession Number
DBCAT000800
Description

Derivatives of carbamic acid, H2NC(=O)OH. Included under this heading are N-substituted and O-substituted carbamic acids. In general carbamate esters are referred to as urethanes, and polymers that include repeating units of carbamate are referred to as POLYURETHANES. Note however that polyurethanes are derived from the polymerization of ISOCYANATES and the singular term URETHANE refers to the ethyl ester of carbamic acid.

Drugs
DrugDrug Description
AlbendazoleA benzimidazole anthelmintic used to treat parenchymal neurocysticercosis and other helminth infections.
Albendazole oxideNot Annotated
BethanecholA muscarinic agonist used to treat postoperative and postpartum nonobstructive functional urinary retention and neurogenic atony of the bladder with retention.
BuntanetapBuntanetap (previously known as Posiphen) is under investigation in clinical trial NCT02925650 (Safety, Tolerability, PK and PD of Posiphen® in Subjects With Early Alzheimer's Disease).
CarbarylA medication used in shampoo to remove lice.
CarisoprodolA centrally acting muscle relaxant used to relieve the discomfort associated with various musculoskeletal conditions.
CobicistatA CYP3A inhibitor used to increase the systemic exposure of atazanavir or darunavir in combination with other antiretroviral agents in the treatment of HIV-1 infection.
DarunavirA HIV protease inhibitor used in the treatment of human immunodeficiency virus (HIV) infection in patients with history of prior antiretroviral therapies.
DiethylcarbamazineAn anthelmintic used to treat filarial infections like Wuchereria bancrofti and Loa loa.
DisulfiramA carbamate derivative used to treat alcohol addiction.
DitiocarbA chelating agent that has been used to mobilize toxic metals from the tissues of man and experimental animals. It is the main metabolite of DISULFIRAM.
Ditiocarb zincDitiocarb Zinc is approved for use within allergenic epicutaneous patch tests which are indicated for use as an aid in the diagnosis of allergic contact dermatitis (ACD) in persons 6...
EmylcamateNot Annotated
Ethyl N-methylcarbamateNot Available
FelbamateAn anticonvulsant used to treat severe epilepsy.
FenbendazoleFenbendazole is a benzimidazole that presents a wide spectrum anthelmintic effect. It is used against a number of gastrointestinal parasites including giardia, roundworms, hookworms, whipworms, the Taenia genus of tapeworms,...
FlubendazoleFlubendazole is an anthelmintic that is used to treat worm infection in humans. It is available OTC in Europe.
GanstigmineInvestigated for use/treatment in alzheimer's disease.
LiranaftateLiranaftate is a small molecule drug. Liranaftate has a monoisotopic molecular weight of 328.12 Da.
MebendazoleA benzimidazole anthelmintic used to treat helminth infections.
MebutamateMebutamate is a sedative and anxiolytic drug with anti-hypertensive (blood pressure lowering) effects comparable to those of other barbiturates but is only around 1/3rd the potency of secobarbital as a...
MeprobamateAn anxiolytic drug used for the short-term management of anxiety symptoms.
MethocarbamolA CNS depressant indicated with rest, physical therapy and other treatments to control the discomfort associated with various acute musculoskeletal conditions.
NOX-700Investigated for use/treatment in diabetes mellitus (type 2).
PhencarbamidePhencarbamide is a small molecule drug. Phencarbamide has a monoisotopic molecular weight of 328.16 Da.
PhenserineFor the treatment of Alzheimer's disease (AD).
PhysostigmineA cholinesterase inhibitor used to treat glaucoma and anticholinergic toxicity.
PyricarbatePyricarbate is a small molecule drug. Pyricarbate has a monoisotopic molecular weight of 253.11 Da.
RivastigmineA cholinesterase inhibitor used to treat mild to moderate dementia in Alzheimer's and Parkinson's.
SulfiramSulfiram is a small molecule drug. Sulfiram has a monoisotopic molecular weight of 264.08 Da.
Tetramethylthiuram monosulfideNot Annotated
ThiramThiram may be used in dermatology as a scabicide . Thiram is mainly used as a fungicide for plants and treatment for seeds, however, this use is being investigated for...
TolciclateNot Annotated
TolnaftateAn antifungal agent used to treat various skin infections caused by fungi.
UrethaneUrethane, formerly marketed as an inactive ingredient in Profenil injection, was determined to be carcinogenic and was removed from the Canadian, US, and UK markets in 1963.
VelufenacinVelufenacin is a small molecule drug. The usage of the INN stem '-fenacin' in the name indicates that Velufenacin is a muscarinic receptor antagonist. Velufenacin is under investigation in clinical...
ZafirlukastA leukotriene receptor antagonist used for prophylaxis and chronic treatment of asthma.
Zinc dibutyldithiocarbamateZinc dibutyldithiocarbamate is approved for use within allergenic epicutaneous patch tests which are indicated for use as an aid in the diagnosis of allergic contact dermatitis (ACD) in persons 6...