Quercetin | Tyrosine-protein kinase HCK | target |
Quercetin | Cytochrome P450 2C8 | enzyme |
Quercetin | Multidrug resistance-associated protein 1 | transporter |
Quercetin | Canalicular multispecific organic anion transporter 1 | transporter |
Quercetin | Monocarboxylate transporter 2 | transporter |
Quercetin | Solute carrier organic anion transporter family member 2B1 | transporter |
Quercetin | P-glycoprotein 1 | transporter |
Quercetin | Monocarboxylate transporter 1 | transporter |
Quercetin | ATP-binding cassette sub-family G member 2 | transporter |
Quercetin | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | target |
Quercetin | UDP-glucuronosyltransferase 3A1 | target |
Quercetin | ATP synthase subunit alpha, mitochondrial | target |
Quercetin | ATP synthase subunit beta, mitochondrial | target |
Quercetin | ATP synthase subunit gamma, mitochondrial | target |
Quercetin | Serine/threonine-protein kinase pim-1 | target |
Quercetin | HTH-type transcriptional regulator TtgR | target |
Quercetin | 3-hydroxyisobutyryl-CoA hydrolase, mitochondrial | target |
Quercetin | 3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ | target |
Quercetin | Serine/threonine-protein kinase 17B | target |
Quercetin | Estrogen receptor alpha | target |
Quercetin | Estrogen receptor beta | target |
Quercetin | Ribosyldihydronicotinamide dehydrogenase [quinone] | target |
Quercetin | Serum albumin | carrier |
Quercetin | Aryl hydrocarbon receptor | target |
Quercetin | Cytochrome P450 1B1 | target |
Quercetin | Actin, cytoplasmic 1 | target |
Quercetin | Casein kinase II subunit alpha | target |
Quercetin | Casein kinase II subunit beta | target |
Quercetin | Eukaryotic translation initiation factor 3 subunit F | target |
Quercetin | Heat shock protein HSP 90-alpha | target |
Quercetin | Heat shock-related 70 kDa protein 2 | target |
Quercetin | RuvB-like 2 | target |
Quercetin | Splicing factor 3B subunit 3 | target |
Quercetin | Ubiquitin-like modifier-activating enzyme 1 | target |
Quercetin | Sex hormone-binding globulin | target |
Quercetin | Carbonyl reductase [NADPH] 1 | target |
Quercetin | CCAAT/enhancer-binding protein beta | target |
Quercetin | Nuclear receptor subfamily 1 group I member 2 | target |
Quercetin | Solute carrier organic anion transporter family member 1B1 | transporter |
Quercetin | Cytochrome P450 2C9 | enzyme |
Quercetin | Cytochrome P450 1A2 | enzyme |
Quercetin | Cytochrome P450 2E1 | enzyme |
Quercetin | Cytochrome P450 2C19 | enzyme |
Quercetin | Cytochrome P450 3A Subfamily | enzyme |
Quercetin | Cytochrome P450 2D6 | enzyme |
Naringenin | Solute carrier organic anion transporter family member 2B1 | transporter |
Naringenin | P-glycoprotein 1 | transporter |
Naringenin | Multidrug resistance-associated protein 1 | transporter |
Naringenin | ATP-binding cassette sub-family G member 2 | transporter |
Naringenin | HTH-type transcriptional regulator TtgR | target |
Naringenin | Estrogen receptor alpha | target |
Naringenin | Aldo-keto reductase family 1 member C1 | target |
Naringenin | Cytochrome P450 1B1 | target |
Naringenin | KAT8 regulatory NSL complex subunit 3 | target |
Naringenin | Sex hormone-binding globulin | target |
Naringenin | Cytochrome P450 19A1 | target |
Naringenin | Estrogen receptor beta | target |
Novobiocin | DNA gyrase subunit B | target |
Novobiocin | Solute carrier family 22 member 6 | transporter |
Novobiocin | Solute carrier family 22 member 8 | transporter |
Novobiocin | Solute carrier family 22 member 11 | transporter |
Novobiocin | ATP-binding cassette sub-family G member 2 | transporter |
Novobiocin | DNA topoisomerase 1 | target |
Novobiocin | Solute carrier organic anion transporter family member 1B1 | transporter |
Novobiocin | Solute carrier organic anion transporter family member 1B3 | transporter |
Novobiocin | Solute carrier organic anion transporter family member 2B1 | transporter |
Estrone | Estrogen receptor alpha | target |
Estrone | Cytochrome P450 1A2 | enzyme |
Estrone | Cytochrome P450 1A1 | enzyme |
Estrone | Serum albumin | carrier |
Estrone | Solute carrier organic anion transporter family member 2B1 | transporter |
Estrone | P-glycoprotein 1 | transporter |
Estrone | Solute carrier organic anion transporter family member 1A2 | transporter |
Estrone | ATP-binding cassette sub-family G member 2 | transporter |
Estrone | Solute carrier organic anion transporter family member 1B1 | transporter |
Estrone | Cytochrome P450 3A4 | enzyme |
Estrone | Cytochrome P450 1B1 | enzyme |
Estrone | Cytochrome P450 2B6 | enzyme |
Estrone | Cytochrome P450 2C9 | enzyme |
Estrone | Cytochrome P450 2E1 | enzyme |
Estrone | Cytochrome P450 3A5 | enzyme |
Estrone | Estrogen receptor beta | target |
Estrone | Androgen receptor | target |
Estrone | Cytochrome P450 19A1 | target |
Estrone | Sex hormone-binding globulin | target |
Estrone | Solute carrier family 22 member 8 | transporter |
Saquinavir | Human immunodeficiency virus type 1 protease | target |
Saquinavir | Cytochrome P450 3A4 | enzyme |
Saquinavir | Cytochrome P450 3A5 | enzyme |
Saquinavir | Alpha-1-acid glycoprotein 1 | carrier |
Saquinavir | Serum albumin | carrier |
Saquinavir | Cytochrome P450 3A7 | enzyme |
Saquinavir | P-glycoprotein 1 | transporter |
Saquinavir | Solute carrier family 22 member 1 | transporter |
Saquinavir | Solute carrier organic anion transporter family member 1A2 | transporter |
Saquinavir | ATP-binding cassette sub-family G member 2 | transporter |
Saquinavir | Solute carrier organic anion transporter family member 1B1 | transporter |
Saquinavir | Multidrug resistance-associated protein 1 | transporter |
Saquinavir | Canalicular multispecific organic anion transporter 1 | transporter |
Saquinavir | Cytochrome P450 2C8 | enzyme |
Saquinavir | Cytochrome P450 2D6 | enzyme |
Saquinavir | Solute carrier organic anion transporter family member 2B1 | transporter |
Saquinavir | Bile salt export pump | transporter |
Omeprazole | Potassium-transporting ATPase alpha chain 1 | target |
Omeprazole | Cytochrome P450 2C19 | enzyme |
Omeprazole | Cytochrome P450 3A4 | enzyme |
Omeprazole | Cytochrome P450 2C9 | enzyme |
Omeprazole | Cytochrome P450 1A2 | enzyme |
Omeprazole | Canalicular multispecific organic anion transporter 2 | transporter |
Omeprazole | P-glycoprotein 1 | transporter |
Omeprazole | ATP-binding cassette sub-family G member 2 | transporter |
Omeprazole | Cytochrome P450 1A1 | enzyme |
Omeprazole | Cytochrome P450 1B1 | enzyme |
Omeprazole | Cytochrome P450 2C18 | enzyme |
Omeprazole | Cytochrome P450 2C8 | enzyme |
Omeprazole | Cytochrome P450 2D6 | enzyme |
Omeprazole | Aryl hydrocarbon receptor | target |
Hesperetin | Microsomal triglyceride transfer protein large subunit | target |
Hesperetin | Sterol O-acyltransferase 1 | target |
Hesperetin | Sterol O-acyltransferase 2 | target |
Hesperetin | Cytochrome P450 1A2 | enzyme |
Hesperetin | ATP-binding cassette sub-family G member 2 | transporter |
Hesperetin | Sex hormone-binding globulin | target |
Genistein | Estrogen receptor beta | target |
Genistein | DNA topoisomerase 2-alpha | target |
Genistein | Protein-tyrosine kinase 2-beta | target |
Genistein | P-glycoprotein 1 | transporter |
Genistein | Multidrug resistance-associated protein 1 | transporter |
Genistein | ATP-binding cassette sub-family G member 2 | transporter |
Genistein | Cytochrome P450 1A2 | enzyme |
Genistein | Nuclear receptor coactivator 1 | target |
Genistein | Estrogen receptor alpha | target |
Genistein | Nuclear receptor coactivator 2 | target |
Genistein | Transthyretin | carrier |
Genistein | Steroid hormone receptor ERR2 | target |
Genistein | Steroid hormone receptor ERR1 | target |
Genistein | Nuclear receptor subfamily 1 group I member 2 | target |
Genistein | RAC-alpha serine/threonine-protein kinase | target |
Genistein | G-protein coupled estrogen receptor 1 | target |
Genistein | Cytochrome P450 1B1 | target |
Genistein | Sex hormone-binding globulin | target |
Genistein | Cytochrome P450 1A1 | enzyme |
Genistein | Solute carrier organic anion transporter family member 1B1 | transporter |
Genistein | Solute carrier organic anion transporter family member 2B1 | transporter |
Genistein | Cytochrome P450 2C8 | enzyme |
Genistein | Cytochrome P450 2C9 | enzyme |
Genistein | Cytochrome P450 3A1 | enzyme |
Genistein | Cytochrome P450 3A2 | enzyme |
Genistein | Cytochrome P450 3A4 | enzyme |
Genistein | Cystic fibrosis transmembrane conductance regulator | target |
Nelfinavir | HIV-1 protease | target |
Nelfinavir | Cytochrome P450 2C19 | enzyme |
Nelfinavir | Cytochrome P450 3A4 | enzyme |
Nelfinavir | Cytochrome P450 2B6 | enzyme |
Nelfinavir | Cytochrome P450 3A5 | enzyme |
Nelfinavir | Cytochrome P450 3A7 | enzyme |
Nelfinavir | P-glycoprotein 1 | transporter |
Nelfinavir | Solute carrier family 22 member 1 | transporter |
Nelfinavir | Solute carrier organic anion transporter family member 1A2 | transporter |
Nelfinavir | ATP-binding cassette sub-family G member 2 | transporter |
Nelfinavir | Solute carrier organic anion transporter family member 1B1 | transporter |
Nelfinavir | Cytochrome P450 2D6 | enzyme |
Nelfinavir | Serum albumin | carrier |
Nelfinavir | UDP-glucuronosyltransferase 1-1 | enzyme |
Nelfinavir | Solute carrier organic anion transporter family member 1B3 | transporter |
Nelfinavir | Solute carrier organic anion transporter family member 2B1 | transporter |
Nelfinavir | Bile salt export pump | transporter |
Nelfinavir | Cytochrome P450 2C9 | enzyme |
Nelfinavir | Alpha-1-acid glycoprotein 1 | carrier |
Diethylstilbestrol | Estrogen receptor alpha | target |
Diethylstilbestrol | Estrogen-related receptor gamma | target |
Diethylstilbestrol | Transthyretin | carrier |
Diethylstilbestrol | Catechol O-methyltransferase | enzyme |
Diethylstilbestrol | Cytochrome P450 19A1 | enzyme |
Diethylstilbestrol | ATP-binding cassette sub-family G member 2 | transporter |
Diethylstilbestrol | P-glycoprotein 1 | transporter |
Diethylstilbestrol | Estrogen receptor beta | target |
Diethylstilbestrol | Cytochrome P450 3A4 | enzyme |
Diethylstilbestrol | Cytochrome P450 2C8 | enzyme |
Diethylstilbestrol | Cytochrome P450 2C9 | enzyme |
Diethylstilbestrol | Cytochrome P450 2E1 | enzyme |
Diethylstilbestrol | Steroid hormone receptor ERR1 | target |
Diethylstilbestrol | Steroid hormone receptor ERR2 | target |
Diethylstilbestrol | Nuclear receptor coactivator 2 | target |
Diethylstilbestrol | Nuclear receptor subfamily 1 group I member 2 | target |
Diethylstilbestrol | Androgen receptor | target |
Diethylstilbestrol | Sex hormone-binding globulin | target |
Diethylstilbestrol | Solute carrier organic anion transporter family member 1B1 | transporter |
Diethylstilbestrol | Solute carrier organic anion transporter family member 2B1 | transporter |
Diethylstilbestrol | Bile salt export pump | transporter |
Ritonavir | Human immunodeficiency virus type 1 protease | target |
Ritonavir | Cytochrome P450 2D6 | enzyme |
Ritonavir | Cytochrome P450 2C9 | enzyme |
Ritonavir | Cytochrome P450 2C19 | enzyme |
Ritonavir | Cytochrome P450 2B6 | enzyme |
Ritonavir | Cytochrome P450 2C8 | enzyme |
Ritonavir | P-glycoprotein 1 | transporter |
Ritonavir | Multidrug resistance-associated protein 1 | transporter |
Ritonavir | Canalicular multispecific organic anion transporter 1 | transporter |
Ritonavir | Solute carrier organic anion transporter family member 1A2 | transporter |
Ritonavir | ATP-binding cassette sub-family G member 2 | transporter |
Ritonavir | Solute carrier organic anion transporter family member 1B1 | transporter |
Ritonavir | Cytochrome P450 1A2 | enzyme |
Ritonavir | Nuclear receptor subfamily 1 group I member 2 | target |
Ritonavir | Serum albumin | carrier |
Ritonavir | Cytochrome P450 3A4 | enzyme |
Ritonavir | Cytochrome P450 3A5 | enzyme |
Ritonavir | Cytochrome P450 3A7 | enzyme |
Ritonavir | UDP-glucuronosyltransferases (UGTs) | enzyme |
Ritonavir | Solute carrier organic anion transporter family member 2B1 | transporter |
Ritonavir | Bile salt export pump | transporter |
Ritonavir | Alpha-1-acid glycoprotein 1 | carrier |
Ritonavir | Solute carrier organic anion transporter family member 1B3 | transporter |
Pantoprazole | Potassium-transporting ATPase alpha chain 1 | target |
Pantoprazole | Cytochrome P450 2C19 | enzyme |
Pantoprazole | Cytochrome P450 3A4 | enzyme |
Pantoprazole | P-glycoprotein 1 | transporter |
Pantoprazole | ATP-binding cassette sub-family G member 2 | transporter |
Pantoprazole | Solute carrier family 22 member 8 | transporter |
Pantoprazole | N(G),N(G)-dimethylarginine dimethylaminohydrolase 1 | target |
Cyclosporine | Calcium signal-modulating cyclophilin ligand | target |
Cyclosporine | Peptidyl-prolyl cis-trans isomerase A | target |
Cyclosporine | Calcineurin subunit B type 2 | target |
Cyclosporine | Cytochrome P450 3A5 | enzyme |
Cyclosporine | Cytochrome P450 3A4 | enzyme |
Cyclosporine | P-glycoprotein 1 | transporter |
Cyclosporine | Bile salt export pump | transporter |
Cyclosporine | Ileal sodium/bile acid cotransporter | transporter |
Cyclosporine | Sodium/bile acid cotransporter | transporter |
Cyclosporine | Solute carrier family 22 member 6 | transporter |
Cyclosporine | Multidrug resistance-associated protein 7 | transporter |
Cyclosporine | Canalicular multispecific organic anion transporter 1 | transporter |
Cyclosporine | ATP-binding cassette sub-family G member 2 | transporter |
Cyclosporine | Solute carrier organic anion transporter family member 1B1 | transporter |
Cyclosporine | Cytochrome P450 2C19 | enzyme |
Cyclosporine | Cytochrome P450 2D6 | enzyme |
Cyclosporine | Peptidyl-prolyl cis-trans isomerase F, mitochondrial | target |
Cyclosporine | Solute carrier organic anion transporter family member 1B3 | transporter |
Taurocholic acid | Bile salt-activated lipase | target |
Taurocholic acid | Gastrotropin | target |
Taurocholic acid | Bile salt export pump | transporter |
Taurocholic acid | Multidrug resistance-associated protein 1 | transporter |
Taurocholic acid | Solute carrier organic anion transporter family member 1A2 | transporter |
Taurocholic acid | Ileal sodium/bile acid cotransporter | transporter |
Taurocholic acid | Canalicular multispecific organic anion transporter 1 | transporter |
Taurocholic acid | Solute carrier organic anion transporter family member 1B1 | transporter |
Taurocholic acid | Canalicular multispecific organic anion transporter 2 | transporter |
Taurocholic acid | Multidrug resistance-associated protein 4 | transporter |
Taurocholic acid | P-glycoprotein 1 | transporter |
Taurocholic acid | Solute carrier family 22 member 6 | transporter |
Taurocholic acid | Multidrug resistance-associated protein 7 | transporter |
Taurocholic acid | Solute carrier family 22 member 8 | transporter |
Taurocholic acid | Solute carrier organic anion transporter family member 4A1 | transporter |
Taurocholic acid | ATP-binding cassette sub-family C member 11 | transporter |
Taurocholic acid | Solute carrier organic anion transporter family member 1C1 | transporter |
Taurocholic acid | Solute carrier organic anion transporter family member 3A1 | transporter |
Taurocholic acid | ATP-binding cassette sub-family G member 2 | transporter |
Taurocholic acid | Solute carrier organic anion transporter family member 2B1 | transporter |
Taurocholic acid | Monocarboxylate transporter 1 | transporter |
Taurocholic acid | Sodium/bile acid cotransporter | transporter |
Taurocholic acid | Organic solute transporter subunit alpha | transporter |
Taurocholic acid | Organic solute transporter subunit beta | transporter |
Taurocholic acid | Solute carrier organic anion transporter family member 1B3 | transporter |
Taurocholic acid | Cystine/glutamate transporter | transporter |
Taurocholic acid | Bile acid receptor | target |
Imatinib | Platelet-derived growth factor receptor beta | target |
Imatinib | Tyrosine-protein kinase ABL1 | target |
Imatinib | Mast/stem cell growth factor receptor Kit | target |
Imatinib | RET proto-oncogene | target |
Imatinib | High affinity nerve growth factor receptor | target |
Imatinib | Macrophage colony-stimulating factor 1 receptor | target |
Imatinib | Platelet-derived growth factor receptor alpha | target |
Imatinib | Epithelial discoidin domain-containing receptor 1 | target |
Imatinib | Cytochrome P450 3A4 | enzyme |
Imatinib | Breakpoint cluster region protein | target |
Imatinib | Cytochrome P450 1A2 | enzyme |
Imatinib | Cytochrome P450 2D6 | enzyme |
Imatinib | Cytochrome P450 2C9 | enzyme |
Imatinib | Cytochrome P450 2C19 | enzyme |
Imatinib | Cytochrome P450 3A5 | enzyme |
Imatinib | Cytochrome P450 3A7 | enzyme |
Imatinib | Solute carrier family 22 member 1 | transporter |
Imatinib | P-glycoprotein 1 | transporter |
Imatinib | Solute carrier family 22 member 2 | transporter |
Imatinib | ATP-binding cassette sub-family G member 2 | transporter |
Imatinib | ATP-binding cassette sub-family A member 3 | transporter |
Imatinib | Prostaglandin G/H synthase 1 | enzyme |
Imatinib | Serum albumin | carrier |
Imatinib | Alpha-1-acid glycoprotein 1 | carrier |
Imatinib | Bile salt export pump | transporter |
Imatinib | Cytochrome P450 2C8 | enzyme |
Estradiol | Estrogen receptor alpha | target |
Estradiol | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol | Sex hormone-binding globulin | carrier |
Estradiol | Estrogen receptor beta | target |
Estradiol | Cytochrome P450 1A2 | enzyme |
Estradiol | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol | Serum albumin | carrier |
Estradiol | Fatty acid-binding protein, intestinal | carrier |
Estradiol | Cytochrome P450 3A4 | enzyme |
Estradiol | Cytochrome P450 3A5 | enzyme |
Estradiol | Cytochrome P450 3A7 | enzyme |
Estradiol | Solute carrier family 22 member 2 | transporter |
Estradiol | Solute carrier family 22 member 3 | transporter |
Estradiol | Multidrug resistance-associated protein 7 | transporter |
Estradiol | Solute carrier family 22 member 11 | transporter |
Estradiol | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol | P-glycoprotein 1 | transporter |
Estradiol | Cytochrome P450 1A1 | enzyme |
Estradiol | Cytochrome P450 1B1 | enzyme |
Estradiol | Cytochrome P450 2C19 | enzyme |
Estradiol | Cytochrome P450 2C8 | enzyme |
Estradiol | Cytochrome P450 2C9 | enzyme |
Estradiol | Solute carrier family 22 member 8 | transporter |
Estradiol | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol | G-protein coupled estrogen receptor 1 | target |
Estradiol | ATP synthase subunit a | target |
Estradiol | Beclin-1 | target |
Estradiol | UDP-glucuronosyltransferase 2B15 | enzyme |
Estradiol | Catechol O-methyltransferase | enzyme |
Estradiol | UDP-glucuronosyltransferases (UGTs) | enzyme |
Estradiol | Cytochrome P450 19A1 | enzyme |
Daidzin | Aldehyde dehydrogenase, mitochondrial | target |
Daidzin | ATP-binding cassette sub-family G member 2 | transporter |
Sorafenib | Serine/threonine-protein kinase B-raf | target |
Sorafenib | Receptor-type tyrosine-protein kinase FLT3 | target |
Sorafenib | RAF proto-oncogene serine/threonine-protein kinase | target |
Sorafenib | Vascular endothelial growth factor receptor 3 | target |
Sorafenib | Platelet-derived growth factor receptor beta | target |
Sorafenib | Mast/stem cell growth factor receptor Kit | target |
Sorafenib | Vascular endothelial growth factor receptor 2 | target |
Sorafenib | Cytochrome P450 3A4 | enzyme |
Sorafenib | UDP-glucuronosyltransferase 1-9 | enzyme |
Sorafenib | Cytochrome P450 2B6 | enzyme |
Sorafenib | Cytochrome P450 2C8 | enzyme |
Sorafenib | Cytochrome P450 3A5 | enzyme |
Sorafenib | Cytochrome P450 3A7 | enzyme |
Sorafenib | Cytochrome P450 2C9 | enzyme |
Sorafenib | Multidrug resistance-associated protein 4 | transporter |
Sorafenib | P-glycoprotein 1 | transporter |
Sorafenib | Canalicular multispecific organic anion transporter 1 | transporter |
Sorafenib | ATP-binding cassette sub-family G member 2 | transporter |
Sorafenib | Cytochrome P450 1A2 | enzyme |
Sorafenib | Cytochrome P450 2C19 | enzyme |
Sorafenib | Cytochrome P450 2D6 | enzyme |
Sorafenib | UDP-glucuronosyltransferase 1-1 | enzyme |
Sorafenib | RalA-binding protein 1 | transporter |
Sorafenib | Fibroblast growth factor receptor 1 | target |
Sorafenib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Sorafenib | Vascular endothelial growth factor receptor 1 | target |
Sorafenib | Solute carrier organic anion transporter family member 1B1 | transporter |
Sunitinib | Platelet-derived growth factor receptor beta | target |
Sunitinib | Vascular endothelial growth factor receptor 1 | target |
Sunitinib | Vascular endothelial growth factor receptor 2 | target |
Sunitinib | Vascular endothelial growth factor receptor 3 | target |
Sunitinib | Mast/stem cell growth factor receptor Kit | target |
Sunitinib | Receptor-type tyrosine-protein kinase FLT3 | target |
Sunitinib | Macrophage colony-stimulating factor 1 receptor | target |
Sunitinib | Platelet-derived growth factor receptor alpha | target |
Sunitinib | Cytochrome P450 3A4 | enzyme |
Sunitinib | Cytochrome P450 3A5 | enzyme |
Sunitinib | Cytochrome P450 3A7 | enzyme |
Sunitinib | Multidrug resistance-associated protein 4 | transporter |
Sunitinib | P-glycoprotein 1 | transporter |
Sunitinib | Canalicular multispecific organic anion transporter 1 | transporter |
Sunitinib | ATP-binding cassette sub-family G member 2 | transporter |
Dronabinol | Cannabinoid receptor 1 | target |
Dronabinol | Cytochrome P450 3A4 | enzyme |
Dronabinol | Cytochrome P450 2C9 | enzyme |
Dronabinol | Cannabinoid receptor 2 | target |
Dronabinol | P-glycoprotein 1 | transporter |
Dronabinol | ATP-binding cassette sub-family G member 2 | transporter |
Dronabinol | Prostaglandin G/H synthase 1 | enzyme |
Dronabinol | Cytochrome P450 2C19 | enzyme |
Dronabinol | Cytochrome P450 1A1 | enzyme |
Dronabinol | Cytochrome P450 1A2 | enzyme |
Dronabinol | Cytochrome P450 1B1 | enzyme |
Dronabinol | Cytochrome P450 2A6 | enzyme |
Dronabinol | Cytochrome P450 2B6 | enzyme |
Dronabinol | Cytochrome P450 2D6 | enzyme |
Dronabinol | Cytochrome P450 2J2 | enzyme |
Dronabinol | Cytochrome P450 3A5 | enzyme |
Dronabinol | Cytochrome P450 3A7 | enzyme |
Dronabinol | Multidrug resistance-associated protein 1 | transporter |
Dronabinol | Liver carboxylesterase 1 | enzyme |
Buprenorphine | Kappa-type opioid receptor | target |
Buprenorphine | Mu-type opioid receptor | target |
Buprenorphine | Cytochrome P450 3A4 | enzyme |
Buprenorphine | Cytochrome P450 2D6 | enzyme |
Buprenorphine | P-glycoprotein 1 | transporter |
Buprenorphine | ATP-binding cassette sub-family G member 2 | transporter |
Buprenorphine | Cytochrome P450 2C9 | enzyme |
Buprenorphine | Cytochrome P450 3A5 | enzyme |
Buprenorphine | Cytochrome P450 2C8 | enzyme |
Buprenorphine | Cytochrome P450 3A7 | enzyme |
Buprenorphine | Delta-type opioid receptor | target |
Buprenorphine | Cytochrome P450 2C18 | enzyme |
Buprenorphine | Cytochrome P450 2C19 | enzyme |
Buprenorphine | Nociceptin receptor | target |
Sulfasalazine | Acetyl-CoA acetyltransferase, mitochondrial | target |
Sulfasalazine | Cystine/glutamate transporter | target |
Sulfasalazine | ATP-binding cassette sub-family G member 2 | transporter |
Sulfasalazine | Canalicular multispecific organic anion transporter 1 | transporter |
Sulfasalazine | Inhibitor of nuclear factor kappa-B kinase subunit alpha | target |
Sulfasalazine | Inhibitor of nuclear factor kappa-B kinase subunit beta | target |
Sulfasalazine | Prostaglandin G/H synthase 2 | target |
Sulfasalazine | Peroxisome proliferator-activated receptor gamma | target |
Sulfasalazine | Prostaglandin G/H synthase 1 | target |
Sulfasalazine | Arachidonate 5-lipoxygenase | target |
Sulfasalazine | Proton-coupled folate transporter | transporter |
Sulfasalazine | Thromboxane-A synthase | target |
Sulfasalazine | Phospholipase A2 | target |
Sulfasalazine | Solute carrier organic anion transporter family member 1B1 | transporter |
Sulfasalazine | Solute carrier organic anion transporter family member 1B3 | transporter |
Sulfasalazine | Solute carrier organic anion transporter family member 2B1 | transporter |
Telmisartan | Type-1 angiotensin II receptor | target |
Telmisartan | Peroxisome proliferator-activated receptor gamma | target |
Telmisartan | P-glycoprotein 1 | transporter |
Telmisartan | Canalicular multispecific organic anion transporter 1 | transporter |
Telmisartan | ATP-binding cassette sub-family G member 2 | transporter |
Telmisartan | Cytochrome P450 2C19 | enzyme |
Telmisartan | Bile salt export pump | transporter |
Telmisartan | UDP-glucuronosyltransferase 1-3 | enzyme |
Dexamethasone | Glucocorticoid receptor | target |
Dexamethasone | Annexin A1 | target |
Dexamethasone | Nitric oxide synthase, inducible | target |
Dexamethasone | Nuclear receptor subfamily 0 group B member 1 | target |
Dexamethasone | Cytochrome P450 3A4 | enzyme |
Dexamethasone | Cytochrome P450 3A5 | enzyme |
Dexamethasone | Cytochrome P450 3A7 | enzyme |
Dexamethasone | Bile salt export pump | transporter |
Dexamethasone | P-glycoprotein 1 | transporter |
Dexamethasone | Canalicular multispecific organic anion transporter 1 | transporter |
Dexamethasone | Solute carrier organic anion transporter family member 1A2 | transporter |
Dexamethasone | ATP-binding cassette sub-family G member 2 | transporter |
Dexamethasone | Steroid 17-alpha-hydroxylase/17,20 lyase | enzyme |
Dexamethasone | Cytochrome P450 1A1 | enzyme |
Dexamethasone | Cytochrome P450 2A6 | enzyme |
Dexamethasone | Cytochrome P450 2B6 | enzyme |
Dexamethasone | Cytochrome P450 2C19 | enzyme |
Dexamethasone | Cytochrome P450 2C8 | enzyme |
Dexamethasone | Cytochrome P450 2E1 | enzyme |
Dexamethasone | Cytochrome P450 3A43 | enzyme |
Dexamethasone | Cytochrome P450 4A11 | enzyme |
Dexamethasone | Nuclear receptor subfamily 1 group I member 2 | target |
Dexamethasone | Cytochrome P450 11B1, mitochondrial | enzyme |
Dexamethasone | Serum albumin | carrier |
Dexamethasone | Corticosteroid 11-beta-dehydrogenase isozyme 2 | enzyme |
Dexamethasone | Corticosteroid 11-beta-dehydrogenase isozyme 1 | enzyme |
Dexamethasone | Solute carrier family 22 member 8 | transporter |
Dasatinib | Tyrosine-protein kinase ABL1 | target |
Dasatinib | Abelson tyrosine-protein kinase 2 | target |
Dasatinib | Proto-oncogene tyrosine-protein kinase Src | target |
Dasatinib | Tyrosine-protein kinase Fyn | target |
Dasatinib | Tyrosine-protein kinase Lck | target |
Dasatinib | Tyrosine-protein kinase Yes | target |
Dasatinib | Mast/stem cell growth factor receptor Kit | target |
Dasatinib | Platelet-derived growth factor receptor beta | target |
Dasatinib | Ephrin type-A receptor 2 | target |
Dasatinib | Signal transducer and activator of transcription 5B | target |
Dasatinib | Cytochrome P450 3A4 | enzyme |
Dasatinib | P-glycoprotein 1 | transporter |
Dasatinib | ATP-binding cassette sub-family G member 2 | transporter |
Dasatinib | Cytochrome P450 1A1 | enzyme |
Dasatinib | Cytochrome P450 1A2 | enzyme |
Dasatinib | Cytochrome P450 1B1 | enzyme |
Dasatinib | Cytochrome P450 3A5 | enzyme |
Dasatinib | Dimethylaniline monooxygenase [N-oxide-forming] 3 | enzyme |
Dasatinib | Tyrosine-protein kinase BTK | target |
Dasatinib | Nuclear receptor subfamily 4 group A member 3 | target |
Dasatinib | Breakpoint cluster region protein | target |
Dasatinib | Tyrosine-protein kinase CSK | target |
Dasatinib | Ephrin type-A receptor 5 | target |
Dasatinib | Ephrin type-B receptor 4 | target |
Dasatinib | Tyrosine-protein kinase Fgr | target |
Dasatinib | Tyrosine-protein kinase FRK | target |
Dasatinib | Heat shock cognate 71 kDa protein | target |
Dasatinib | Tyrosine-protein kinase Lyn | target |
Dasatinib | Mitogen-activated protein kinase kinase kinase MLT | target |
Dasatinib | Mitogen-activated protein kinase 14 | target |
Dasatinib | Amidophosphoribosyltransferase | target |
Rabeprazole | Potassium-transporting ATPase alpha chain 1 | target |
Rabeprazole | Cytochrome P450 3A4 | enzyme |
Rabeprazole | Cytochrome P450 2C19 | enzyme |
Rabeprazole | ATP-binding cassette sub-family G member 2 | transporter |
Rabeprazole | Cytochrome P450 1A1 | enzyme |
Rabeprazole | Cytochrome P450 1A2 | enzyme |
Rabeprazole | Cytochrome P450 2C9 | enzyme |
Rabeprazole | Cytochrome P450 2D6 | enzyme |
Rabeprazole | Cytochrome P450 2C8 | enzyme |
Elacridar | P-glycoprotein 1 | target |
Elacridar | ATP-binding cassette sub-family G member 2 | transporter |
Elacridar | P-glycoprotein 1 | transporter |
Nilotinib | Tyrosine-protein kinase ABL1 | target |
Nilotinib | Mast/stem cell growth factor receptor Kit | target |
Nilotinib | Cytochrome P450 2D6 | enzyme |
Nilotinib | Cytochrome P450 2C8 | enzyme |
Nilotinib | Cytochrome P450 2C9 | enzyme |
Nilotinib | Cytochrome P450 3A4 | enzyme |
Nilotinib | P-glycoprotein 1 | transporter |
Nilotinib | ATP-binding cassette sub-family G member 2 | transporter |
Nilotinib | UDP-glucuronosyltransferase 1-1 | transporter |
Nilotinib | Cytochrome P450 2B6 | enzyme |
Nilotinib | Solute carrier organic anion transporter family member 1B1 | transporter |
Erlotinib | Epidermal growth factor receptor | target |
Erlotinib | Cytochrome P450 3A4 | enzyme |
Erlotinib | ATP-binding cassette sub-family G member 2 | transporter |
Erlotinib | P-glycoprotein 1 | transporter |
Erlotinib | Nuclear receptor subfamily 1 group I member 2 | target |
Erlotinib | Cytochrome P450 3A5 | enzyme |
Erlotinib | Cytochrome P450 1A1 | enzyme |
Erlotinib | Cytochrome P450 1A2 | enzyme |
Erlotinib | Cytochrome P450 1B1 | enzyme |
Erlotinib | Cytochrome P450 2D6 | enzyme |
Erlotinib | Cytochrome P450 2C8 | enzyme |
Erlotinib | UDP-glucuronosyltransferase 1-1 | enzyme |
Erlotinib | Serum albumin | carrier |
Erlotinib | Alpha-1-acid glycoprotein 1 | carrier |
Erlotinib | Solute carrier organic anion transporter family member 2B1 | transporter |
Vandetanib | Vascular endothelial growth factor A | target |
Vandetanib | Epidermal growth factor receptor | target |
Vandetanib | Multidrug resistance-associated protein 1 | transporter |
Vandetanib | ATP-binding cassette sub-family G member 2 | transporter |
Vandetanib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Vandetanib | Dimethylaniline monooxygenase [N-oxide-forming] 1 | enzyme |
Vandetanib | Dimethylaniline monooxygenase [N-oxide-forming] 3 | enzyme |
Vandetanib | Protein-tyrosine kinase 6 | target |
Vandetanib | Angiopoietin-1 receptor | target |
Vandetanib | Alpha-1-acid glycoprotein 1 | carrier |
Vandetanib | Serum albumin | carrier |
Vandetanib | Cytochrome P450 3A4 | enzyme |
Vandetanib | Solute carrier family 22 member 2 | transporter |
Vandetanib | P-glycoprotein 1 | transporter |
Cabazitaxel | Cytochrome P450 3A4 | enzyme |
Cabazitaxel | Cytochrome P450 3A5 | enzyme |
Cabazitaxel | Cytochrome P450 2C8 | enzyme |
Cabazitaxel | P-glycoprotein 1 | transporter |
Cabazitaxel | ATP-binding cassette sub-family G member 2 | transporter |
Cabazitaxel | Tubulin alpha-4A chain | target |
Cabazitaxel | Tubulin beta-1 chain | target |
Cabazitaxel | Solute carrier organic anion transporter family member 1B1 | transporter |
Cabazitaxel | Solute carrier organic anion transporter family member 1B3 | transporter |
Rilpivirine | Cytochrome P450 3A4 | enzyme |
Rilpivirine | Reverse transcriptase/RNaseH | target |
Rilpivirine | Nuclear receptor subfamily 1 group I member 2 | target |
Rilpivirine | Cytochrome P450 2C19 | enzyme |
Rilpivirine | Cytochrome P450 2B6 | enzyme |
Rilpivirine | P-glycoprotein 1 | transporter |
Rilpivirine | ATP-binding cassette sub-family G member 2 | transporter |
Rilpivirine | Solute carrier organic anion transporter family member 1B1 | transporter |
Rilpivirine | Solute carrier organic anion transporter family member 1B3 | transporter |
Rilpivirine | Serum albumin | carrier |
Rilpivirine | Cytochrome P450 2D6 | enzyme |
Rilpivirine | Cytochrome P450 2C9 | enzyme |
Rilpivirine | Cytochrome P450 2C8 | enzyme |
Rilpivirine | Cytochrome P450 2E1 | enzyme |
Vismodegib | Smoothened homolog | target |
Vismodegib | Cytochrome P450 2C9 | enzyme |
Vismodegib | Cytochrome P450 3A4 | enzyme |
Vismodegib | P-glycoprotein 1 | transporter |
Vismodegib | Cytochrome P450 2C8 | enzyme |
Vismodegib | Cytochrome P450 2C19 | enzyme |
Vismodegib | ATP-binding cassette sub-family G member 2 | transporter |
Vismodegib | Serum albumin | carrier |
Vismodegib | Alpha-1-acid glycoprotein 1 | carrier |
Regorafenib | Cytochrome P450 3A4 | enzyme |
Regorafenib | UDP-glucuronosyltransferase 1-9 | enzyme |
Regorafenib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Regorafenib | Vascular endothelial growth factor receptor 1 | target |
Regorafenib | Vascular endothelial growth factor receptor 2 | target |
Regorafenib | Vascular endothelial growth factor receptor 3 | target |
Regorafenib | Mast/stem cell growth factor receptor Kit | target |
Regorafenib | Platelet-derived growth factor receptor alpha | target |
Regorafenib | Platelet-derived growth factor receptor beta | target |
Regorafenib | Fibroblast growth factor receptor 1 | target |
Regorafenib | Fibroblast growth factor receptor 2 | target |
Regorafenib | Angiopoietin-1 receptor | target |
Regorafenib | Discoidin domain-containing receptor 2 | target |
Regorafenib | High affinity nerve growth factor receptor | target |
Regorafenib | Ephrin type-A receptor 2 | target |
Regorafenib | RAF proto-oncogene serine/threonine-protein kinase | target |
Regorafenib | Serine/threonine-protein kinase B-raf | target |
Regorafenib | Cytochrome P450 2C8 | enzyme |
Regorafenib | Cytochrome P450 2C9 | enzyme |
Regorafenib | Cytochrome P450 2B6 | enzyme |
Regorafenib | Mitogen-activated protein kinase 11 | target |
Regorafenib | Tyrosine-protein kinase FRK | target |
Regorafenib | Tyrosine-protein kinase ABL1 | target |
Regorafenib | P-glycoprotein 1 | transporter |
Regorafenib | ATP-binding cassette sub-family G member 2 | transporter |
Regorafenib | UDP-glucuronosyltransferase 1-1 | enzyme |
Regorafenib | Cytochrome P450 2C19 | enzyme |
Ponatinib | Tyrosine-protein kinase ABL1 | target |
Ponatinib | Breakpoint cluster region protein | target |
Ponatinib | Mast/stem cell growth factor receptor Kit | target |
Ponatinib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Ponatinib | Angiopoietin-1 receptor | target |
Ponatinib | Receptor-type tyrosine-protein kinase FLT3 | target |
Ponatinib | Cytochrome P450 3A4 | enzyme |
Ponatinib | Cytochrome P450 2C8 | enzyme |
Ponatinib | Cytochrome P450 2D6 | enzyme |
Ponatinib | Cytochrome P450 3A5 | enzyme |
Ponatinib | P-glycoprotein 1 | transporter |
Ponatinib | ATP-binding cassette sub-family G member 2 | transporter |
Ponatinib | Fibroblast growth factor receptor 1 | target |
Ponatinib | Fibroblast growth factor receptor 2 | target |
Ponatinib | Fibroblast growth factor receptor 3 | target |
Ponatinib | Fibroblast growth factor receptor 4 | target |
Ponatinib | Tyrosine-protein kinase Lck | target |
Ponatinib | Proto-oncogene tyrosine-protein kinase Src | target |
Ponatinib | Tyrosine-protein kinase Lyn | target |
Ponatinib | Vascular endothelial growth factor receptor 2 | target |
Ponatinib | Platelet-derived growth factor receptor alpha | target |
Dabrafenib | Cytochrome P450 3A4 | enzyme |
Dabrafenib | Cytochrome P450 2C8 | enzyme |
Dabrafenib | P-glycoprotein 1 | transporter |
Dabrafenib | ATP-binding cassette sub-family G member 2 | transporter |
Dabrafenib | Solute carrier organic anion transporter family member 1B1 | transporter |
Dabrafenib | Solute carrier organic anion transporter family member 1B3 | transporter |
Dabrafenib | Solute carrier family 22 member 6 | transporter |
Dabrafenib | Solute carrier family 22 member 8 | transporter |
Dabrafenib | Serine/threonine-protein kinase B-raf | target |
Dabrafenib | RAF proto-oncogene serine/threonine-protein kinase | target |
Dabrafenib | Serine/threonine-protein kinase SIK1 | target |
Dabrafenib | Serine/threonine-protein kinase Nek11 | target |
Dabrafenib | LIM domain kinase 1 | target |
Dabrafenib | Cytochrome P450 2B6 | enzyme |
Dabrafenib | Cytochrome P450 2C9 | enzyme |
Dabrafenib | Cytochrome P450 2C19 | enzyme |
Dabrafenib | Cytochrome P450 1A2 | enzyme |
Afatinib | Epidermal growth factor receptor | target |
Afatinib | Receptor tyrosine-protein kinase erbB-2 | target |
Afatinib | Receptor tyrosine-protein kinase erbB-4 | target |
Afatinib | P-glycoprotein 1 | transporter |
Afatinib | ATP-binding cassette sub-family G member 2 | transporter |
Cobicistat | Cytochrome P450 2D6 | enzyme |
Cobicistat | P-glycoprotein 1 | transporter |
Cobicistat | ATP-binding cassette sub-family G member 2 | transporter |
Cobicistat | Cytochrome P450 3A4 | enzyme |
Cobicistat | Cytochrome P450 3A5 | enzyme |
Cobicistat | Cytochrome P450 3A7 | enzyme |
Cobicistat | Cytochrome P450 3A43 | enzyme |
Cobicistat | Solute carrier organic anion transporter family member 1B1 | transporter |
Cobicistat | Solute carrier organic anion transporter family member 1B3 | transporter |
Rolapitant | Neurokinin 1 receptor | target |
Rolapitant | Cytochrome P450 2D6 | enzyme |
Rolapitant | Cytochrome P450 3A4 | enzyme |
Rolapitant | ATP-binding cassette sub-family G member 2 | transporter |
Rolapitant | P-glycoprotein 1 | transporter |
Daclatasvir | Nonstructural protein 5A | target |
Daclatasvir | Cytochrome P450 3A5 | enzyme |
Daclatasvir | Cytochrome P450 3A4 | enzyme |
Daclatasvir | Cytochrome P450 3A43 | enzyme |
Daclatasvir | Cytochrome P450 3A7 | enzyme |
Daclatasvir | P-glycoprotein 1 | transporter |
Daclatasvir | Solute carrier organic anion transporter family member 1B1 | transporter |
Daclatasvir | Solute carrier organic anion transporter family member 1B3 | transporter |
Daclatasvir | ATP-binding cassette sub-family G member 2 | transporter |
Alectinib | ALK tyrosine kinase receptor | target |
Alectinib | ATP-binding cassette sub-family G member 2 | transporter |
Alectinib | P-glycoprotein 1 | transporter |
Dasabuvir | Nonstructural protein 5B (NS5B) | target |
Dasabuvir | Cytochrome P450 2C8 | enzyme |
Dasabuvir | Cytochrome P450 3A4 | enzyme |
Dasabuvir | Cytochrome P450 2D6 | enzyme |
Dasabuvir | UDP-glucuronosyltransferase 1-1 | enzyme |
Dasabuvir | ATP-binding cassette sub-family G member 2 | transporter |
Dasabuvir | ATP-binding cassette sub-family B member 5 | transporter |
Dasabuvir | P-glycoprotein 1 | transporter |
Velpatasvir | Cytochrome P450 2B6 | enzyme |
Velpatasvir | Cytochrome P450 2C8 | enzyme |
Velpatasvir | Cytochrome P450 3A4 | enzyme |
Velpatasvir | Nonstructural protein 5A | target |
Velpatasvir | P-glycoprotein 1 | transporter |
Velpatasvir | ATP-binding cassette sub-family G member 2 | transporter |
Velpatasvir | Solute carrier organic anion transporter family member 1B1 | transporter |
Velpatasvir | Solute carrier organic anion transporter family member 1B3 | transporter |
Velpatasvir | Solute carrier organic anion transporter family member 2B1 | transporter |
Simeprevir | NS3 protease | target |
Simeprevir | Serum albumin | carrier |
Simeprevir | Cytochrome P450 1A2 | enzyme |
Simeprevir | P-glycoprotein 1 | transporter |
Simeprevir | Solute carrier organic anion transporter family member 1B1 | transporter |
Simeprevir | Solute carrier organic anion transporter family member 1B3 | transporter |
Simeprevir | Cytochrome P450 3A4 | enzyme |
Simeprevir | Canalicular multispecific organic anion transporter 1 | transporter |
Simeprevir | ATP-binding cassette sub-family G member 2 | transporter |
Simeprevir | Solute carrier organic anion transporter family member 2B1 | transporter |
Simeprevir | Sodium/bile acid cotransporter | transporter |
Simeprevir | Bile salt export pump | transporter |
Topiroxostat | Xanthine dehydrogenase/oxidase | target |
Topiroxostat | ATP-binding cassette sub-family G member 2 | transporter |
Topiroxostat | Serum albumin | carrier |
Topiroxostat | Alpha-1-acid glycoprotein 1 | carrier |
Topiroxostat | Cytochrome P450 2C8 | enzyme |
Topiroxostat | Cytochrome P450 2C9 | enzyme |
Topiroxostat | Cytochrome P450 1A1 | enzyme |
Topiroxostat | Cytochrome P450 3A4 | enzyme |
Topiroxostat | Cytochrome P450 2C19 | enzyme |
Topiroxostat | Solute carrier family 22 member 8 | transporter |
Topiroxostat | Solute carrier family 22 member 6 | transporter |
Topiroxostat | UDP-glucuronosyltransferase 1-9 | enzyme |
Voxilaprevir | Cytochrome P450 3A4 | enzyme |
Voxilaprevir | Cytochrome P450 1A2 | enzyme |
Voxilaprevir | Cytochrome P450 2C8 | enzyme |
Voxilaprevir | NS3/4A protein | target |
Voxilaprevir | P-glycoprotein 1 | transporter |
Voxilaprevir | ATP-binding cassette sub-family G member 2 | transporter |
Voxilaprevir | Solute carrier organic anion transporter family member 1B1 | transporter |
Voxilaprevir | Solute carrier organic anion transporter family member 1B3 | transporter |
Enasidenib | Cytochrome P450 1A2 | enzyme |
Enasidenib | Cytochrome P450 2B6 | enzyme |
Enasidenib | Isocitrate dehydrogenase [NADP], mitochondrial | target |
Enasidenib | Cytochrome P450 2C8 | enzyme |
Enasidenib | Cytochrome P450 2C9 | enzyme |
Enasidenib | Cytochrome P450 2C19 | enzyme |
Enasidenib | Cytochrome P450 2D6 | enzyme |
Enasidenib | Cytochrome P450 3A4 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 1-1 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 1-3 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 1-4 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 1-9 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 2B7 | enzyme |
Enasidenib | UDP-glucuronosyltransferase 2B15 | enzyme |
Enasidenib | P-glycoprotein 1 | transporter |
Enasidenib | ATP-binding cassette sub-family G member 2 | transporter |
Enasidenib | Solute carrier family 22 member 6 | transporter |
Enasidenib | Solute carrier organic anion transporter family member 1B1 | transporter |
Enasidenib | Solute carrier family 22 member 2 | transporter |
Enasidenib | Solute carrier organic anion transporter family member 1B3 | transporter |
Enasidenib | Solute carrier family 22 member 8 | transporter |
Pibrentasvir | Nonstructural protein 5A | target |
Pibrentasvir | Cytochrome P450 3A Subfamily | enzyme |
Pibrentasvir | UDP-glucuronosyltransferase 1-1 | enzyme |
Pibrentasvir | P-glycoprotein 1 | transporter |
Pibrentasvir | ATP-binding cassette sub-family G member 2 | transporter |
Pibrentasvir | Solute carrier organic anion transporter family member 1B1 | transporter |
Pibrentasvir | Solute carrier organic anion transporter family member 1B3 | transporter |
Glecaprevir | Cytochrome P450 3A Subfamily | enzyme |
Glecaprevir | UDP-glucuronosyltransferase 1-1 | enzyme |
Glecaprevir | P-glycoprotein 1 | transporter |
Glecaprevir | ATP-binding cassette sub-family G member 2 | transporter |
Glecaprevir | Solute carrier organic anion transporter family member 1B1 | transporter |
Glecaprevir | Solute carrier organic anion transporter family member 1B3 | transporter |
Glecaprevir | NS3 protease | target |
Glecaprevir | Cytochrome P450 3A4 | enzyme |
Abemaciclib | Multidrug and toxin extrusion protein 1 | transporter |
Abemaciclib | Multidrug and toxin extrusion protein 2 | transporter |
Abemaciclib | Cyclin-dependent kinase 4 | target |
Abemaciclib | Cyclin-dependent kinase 6 | target |
Abemaciclib | Serum albumin | carrier |
Abemaciclib | alpha1-acid glycoprotein | carrier |
Abemaciclib | Cytochrome P450 3A4 | enzyme |
Abemaciclib | P-glycoprotein 1 | transporter |
Abemaciclib | ATP-binding cassette sub-family G member 2 | transporter |
Abemaciclib | Solute carrier family 22 member 2 | transporter |
Abemaciclib | Cytochrome P450 1A2 | enzyme |
Abemaciclib | Cytochrome P450 2B6 | enzyme |
Abemaciclib | Cytochrome P450 2C8 | enzyme |
Abemaciclib | Cytochrome P450 2C9 | enzyme |
Abemaciclib | Cytochrome P450 2D6 | enzyme |
Letermovir | UDP-glucuronosyltransferase 1-1 | enzyme |
Letermovir | UDP-glucuronosyltransferase 1-3 | enzyme |
Letermovir | Solute carrier organic anion transporter family member 1B1 | transporter |
Letermovir | Solute carrier organic anion transporter family member 1B3 | transporter |
Letermovir | Tripartite terminase subunit 1 | target |
Letermovir | Tripartite terminase subunit 2 | target |
Letermovir | Tripartite terminase subunit 3 | target |
Letermovir | Cytochrome P450 2D6 | enzyme |
Letermovir | Cytochrome P450 2C8 | enzyme |
Letermovir | Cytochrome P450 2C19 | enzyme |
Letermovir | Cytochrome P450 2C9 | enzyme |
Letermovir | Cytochrome P450 2B6 | enzyme |
Letermovir | P-glycoprotein 1 | transporter |
Letermovir | ATP-binding cassette sub-family G member 2 | transporter |
Letermovir | Bile salt export pump | transporter |
Letermovir | Solute carrier family 22 member 8 | transporter |
Letermovir | Canalicular multispecific organic anion transporter 1 | transporter |
Letermovir | Cytochrome P450 3A4 | enzyme |
Letermovir | Cytochrome P450 3A5 | enzyme |
Letermovir | Cytochrome P450 3A7 | enzyme |
Letermovir | Cytochrome P450 3A43 | enzyme |
Brigatinib | ALK tyrosine kinase receptor | target |
Brigatinib | Epidermal growth factor receptor | target |
Brigatinib | Tyrosine-protein kinase ABL1 | target |
Brigatinib | Insulin-like growth factor 1 receptor | target |
Brigatinib | Receptor-type tyrosine-protein kinase FLT3 | target |
Brigatinib | Cytochrome P450 2C8 | enzyme |
Brigatinib | Cytochrome P450 3A4 | enzyme |
Brigatinib | Insulin receptor | target |
Brigatinib | Hepatocyte growth factor receptor | target |
Brigatinib | Receptor tyrosine-protein kinase erbB-4 | target |
Brigatinib | Receptor tyrosine-protein kinase erbB-2 | target |
Brigatinib | ATP-binding cassette sub-family B member 5 | transporter |
Brigatinib | ATP-binding cassette sub-family G member 2 | transporter |
Brigatinib | Solute carrier family 22 member 1 | transporter |
Brigatinib | Multidrug and toxin extrusion protein 1 | transporter |
Brigatinib | Multidrug and toxin extrusion protein 2 | transporter |
Brigatinib | Cytochrome P450 3A Subfamily | enzyme |
Rucaparib | Poly [ADP-ribose] polymerase 1 | target |
Rucaparib | Poly [ADP-ribose] polymerase 2 | target |
Rucaparib | Poly [ADP-ribose] polymerase 3 | target |
Rucaparib | Cytochrome P450 2D6 | enzyme |
Rucaparib | Cytochrome P450 1A2 | enzyme |
Rucaparib | Cytochrome P450 3A4 | enzyme |
Rucaparib | P-glycoprotein 1 | transporter |
Rucaparib | ATP-binding cassette sub-family G member 2 | transporter |
Rucaparib | Multidrug and toxin extrusion protein 1 | transporter |
Rucaparib | Multidrug and toxin extrusion protein 2 | transporter |
Rucaparib | Solute carrier family 22 member 1 | transporter |
Rucaparib | Multidrug resistance-associated protein 4 | transporter |
Rucaparib | Solute carrier organic anion transporter family member 1B1 | transporter |
Rucaparib | Solute carrier organic anion transporter family member 1B3 | transporter |
Rucaparib | Solute carrier family 22 member 6 | transporter |
Rucaparib | Solute carrier family 22 member 8 | transporter |
Rucaparib | Cytochrome P450 3A5 | enzyme |
Rucaparib | Cytochrome P450 3A7 | enzyme |
Rucaparib | Cytochrome P450 3A43 | enzyme |
Rucaparib | Cytochrome P450 2C19 | enzyme |
Rucaparib | Cytochrome P450 2C9 | enzyme |
Rucaparib | Cytochrome P450 2C8 | enzyme |
Rucaparib | UDP-glucuronosyltransferase 1-1 | enzyme |
Baricitinib | Solute carrier family 22 member 8 | transporter |
Baricitinib | ATP-binding cassette sub-family G member 2 | transporter |
Baricitinib | Multidrug and toxin extrusion protein 2 | transporter |
Baricitinib | Cytochrome P450 3A4 | enzyme |
Baricitinib | Tyrosine-protein kinase JAK1 | target |
Baricitinib | Tyrosine-protein kinase JAK2 | target |
Baricitinib | Solute carrier family 22 member 6 | transporter |
Baricitinib | Solute carrier family 22 member 2 | transporter |
Baricitinib | Solute carrier organic anion transporter family member 1B3 | transporter |
Baricitinib | Tyrosine-protein kinase JAK3 | target |
Baricitinib | P-glycoprotein 1 | transporter |
Baricitinib | Non-receptor tyrosine-protein kinase TYK2 | target |
Cannabidiol | Cytochrome P450 2C9 | enzyme |
Cannabidiol | Cytochrome P450 2C19 | enzyme |
Cannabidiol | Cytochrome P450 2D6 | enzyme |
Cannabidiol | Cytochrome P450 3A4 | enzyme |
Cannabidiol | Cannabinoid receptor 1 | target |
Cannabidiol | Cannabinoid receptor 2 | target |
Cannabidiol | G-protein coupled receptor 12 | target |
Cannabidiol | Glycine receptor subunit alpha-1 | target |
Cannabidiol | Glycine receptor (alpha-1/beta) | target |
Cannabidiol | Glycine receptor subunit alpha-3 | target |
Cannabidiol | N-arachidonyl glycine receptor | target |
Cannabidiol | G-protein coupled receptor 55 | target |
Cannabidiol | 5-hydroxytryptamine receptor 1A | target |
Cannabidiol | 5-hydroxytryptamine receptor 2A | target |
Cannabidiol | Neuronal acetylcholine receptor subunit alpha-7 | target |
Cannabidiol | Delta-type opioid receptor | target |
Cannabidiol | Mu-type opioid receptor | target |
Cannabidiol | Peroxisome proliferator-activated receptor gamma | target |
Cannabidiol | Cytochrome P450 3A5 | enzyme |
Cannabidiol | Arylalkylamine N-acetyltransferase | enzyme |
Cannabidiol | Cytochrome P450 1A1 | enzyme |
Cannabidiol | Fatty-acid amide hydrolase 1 | enzyme |
Cannabidiol | Arachidonate 5-lipoxygenase | enzyme |
Cannabidiol | Arachidonate 15-lipoxygenase | enzyme |
Cannabidiol | Quinone oxidoreductase | enzyme |
Cannabidiol | Multidrug resistance-associated protein 1 | transporter |
Cannabidiol | ATP-binding cassette sub-family G member 2 | transporter |
Cannabidiol | Equilibrative nucleoside transporter 1 | transporter |
Cannabidiol | Transient receptor potential cation channel subfamily V member 1 | target |
Cannabidiol | Voltage-dependent T-type calcium channel subunit alpha-1G | target |
Cannabidiol | Voltage-dependent T-type calcium channel subunit alpha-1H | target |
Cannabidiol | Voltage-dependent T-type calcium channel subunit alpha-1I | target |
Cannabidiol | Transient receptor potential cation channel subfamily A member 1 | target |
Cannabidiol | Transient receptor potential cation channel subfamily M member 8 | target |
Cannabidiol | Transient receptor potential cation channel subfamily V member 2 | target |
Cannabidiol | Transient receptor potential cation channel subfamily V member 3 | target |
Cannabidiol | Transient receptor potential cation channel subfamily V member 4 | target |
Cannabidiol | Voltage-dependent anion-selective channel protein 1 | target |
Cannabidiol | 5-hydroxytryptamine receptor 3A | target |
Cannabidiol | Adenosine receptor A1 | target |
Cannabidiol | Prostaglandin G/H synthase 1 | target |
Cannabidiol | Prostaglandin G/H synthase 2 | target |
Cannabidiol | Acetyl-CoA acetyltransferase, mitochondrial | target |
Cannabidiol | Steroid 17-alpha-hydroxylase/17,20 lyase | target |
Cannabidiol | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | target |
Cannabidiol | Glutathione reductase, mitochondrial | target |
Cannabidiol | Glutathione peroxidase 1 | target |
Cannabidiol | Indoleamine 2,3-dioxygenase 1 | target |
Cannabidiol | Cytochrome P450 1B1 | target |
Cannabidiol | NAD(P)H dehydrogenase [quinone] 1 | target |
Cannabidiol | Catalase | target |
Cannabidiol | Cytochrome P450 3A5 | target |
Cannabidiol | Cytochrome P450 2D6 | target |
Cannabidiol | Superoxide dismutase [Cu-Zn] | target |
Cannabidiol | Cytochrome P450 1A2 | target |
Cannabidiol | Cytochrome P450 3A7 | target |
Cannabidiol | Arylalkylamine N-acetyltransferase | target |
Cannabidiol | N-acylethanolamine-hydrolyzing acid amidase | target |
Cannabidiol | Cytochrome P450 1A2 | enzyme |
Cannabidiol | Cytochrome P450 1B1 | enzyme |
Cannabidiol | Cytochrome P450 2A6 | enzyme |
Cannabidiol | Cytochrome P450 2B6 | enzyme |
Cannabidiol | Cytochrome P450 2C8 | enzyme |
Cannabidiol | Cytochrome P450 2E1 | enzyme |
Cannabidiol | Cytochrome P450 3A7 | enzyme |
Cannabidiol | UDP-glucuronosyltransferase 1-7 | enzyme |
Cannabidiol | UDP-glucuronosyltransferase 1-9 | enzyme |
Cannabidiol | UDP-glucuronosyltransferase 2B7 | enzyme |
Cannabidiol | UDP-glucuronosyltransferase 2B17 | enzyme |
Cannabidiol | P-glycoprotein 1 | transporter |
Cannabidiol | Cytochrome P450 2J2 | enzyme |
Cannabidiol | Liver carboxylesterase 1 | enzyme |
Estradiol acetate | Estrogen receptor alpha | target |
Estradiol acetate | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol acetate | Sex hormone-binding globulin | carrier |
Estradiol acetate | Estrogen receptor beta | target |
Estradiol acetate | Cytochrome P450 1A2 | enzyme |
Estradiol acetate | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol acetate | Serum albumin | carrier |
Estradiol acetate | Fatty acid-binding protein, intestinal | carrier |
Estradiol acetate | Cytochrome P450 3A4 | enzyme |
Estradiol acetate | Cytochrome P450 3A5 | enzyme |
Estradiol acetate | Cytochrome P450 3A7 | enzyme |
Estradiol acetate | Solute carrier family 22 member 2 | transporter |
Estradiol acetate | Solute carrier family 22 member 1 | transporter |
Estradiol acetate | Solute carrier family 22 member 3 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 2B1 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 1A2 | transporter |
Estradiol acetate | Multidrug resistance-associated protein 7 | transporter |
Estradiol acetate | Solute carrier family 22 member 11 | transporter |
Estradiol acetate | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol acetate | P-glycoprotein 1 | transporter |
Estradiol acetate | Cytochrome P450 1A1 | enzyme |
Estradiol acetate | Cytochrome P450 1B1 | enzyme |
Estradiol acetate | Cytochrome P450 2C19 | enzyme |
Estradiol acetate | Cytochrome P450 2C8 | enzyme |
Estradiol acetate | Cytochrome P450 2C9 | enzyme |
Estradiol acetate | Solute carrier family 22 member 8 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol acetate | Solute carrier organic anion transporter family member 4A1 | transporter |
Estradiol acetate | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol acetate | Nuclear receptor coactivator 2 | target |
Estradiol acetate | G-protein coupled estrogen receptor 1 | target |
Estradiol acetate | ATP synthase subunit a | target |
Estradiol acetate | Beclin-1 | target |
Estradiol acetate | Estradiol 17-beta-dehydrogenase 2 | target |
Estradiol acetate | Estrogen-related receptor gamma | target |
Estradiol benzoate | Estrogen receptor alpha | target |
Estradiol benzoate | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol benzoate | Sex hormone-binding globulin | carrier |
Estradiol benzoate | Estrogen receptor beta | target |
Estradiol benzoate | Cytochrome P450 1A2 | enzyme |
Estradiol benzoate | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol benzoate | Serum albumin | carrier |
Estradiol benzoate | Fatty acid-binding protein, intestinal | carrier |
Estradiol benzoate | Cytochrome P450 3A4 | enzyme |
Estradiol benzoate | Cytochrome P450 3A5 | enzyme |
Estradiol benzoate | Cytochrome P450 3A7 | enzyme |
Estradiol benzoate | Solute carrier family 22 member 2 | transporter |
Estradiol benzoate | Solute carrier family 22 member 1 | transporter |
Estradiol benzoate | Solute carrier family 22 member 3 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 2B1 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 1A2 | transporter |
Estradiol benzoate | Multidrug resistance-associated protein 7 | transporter |
Estradiol benzoate | Solute carrier family 22 member 11 | transporter |
Estradiol benzoate | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol benzoate | P-glycoprotein 1 | transporter |
Estradiol benzoate | Cytochrome P450 1A1 | enzyme |
Estradiol benzoate | Cytochrome P450 1B1 | enzyme |
Estradiol benzoate | Cytochrome P450 2C19 | enzyme |
Estradiol benzoate | Cytochrome P450 2C8 | enzyme |
Estradiol benzoate | Cytochrome P450 2C9 | enzyme |
Estradiol benzoate | Solute carrier family 22 member 8 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol benzoate | Solute carrier organic anion transporter family member 4A1 | transporter |
Estradiol benzoate | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol benzoate | Nuclear receptor coactivator 2 | target |
Estradiol benzoate | G-protein coupled estrogen receptor 1 | target |
Estradiol benzoate | ATP synthase subunit a | target |
Estradiol benzoate | Beclin-1 | target |
Estradiol benzoate | Estradiol 17-beta-dehydrogenase 2 | target |
Estradiol benzoate | Estrogen-related receptor gamma | target |
Estradiol cypionate | Estrogen receptor alpha | target |
Estradiol cypionate | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol cypionate | Sex hormone-binding globulin | carrier |
Estradiol cypionate | Estrogen receptor beta | target |
Estradiol cypionate | Cytochrome P450 1A2 | enzyme |
Estradiol cypionate | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol cypionate | Serum albumin | carrier |
Estradiol cypionate | Fatty acid-binding protein, intestinal | carrier |
Estradiol cypionate | Cytochrome P450 3A4 | enzyme |
Estradiol cypionate | Cytochrome P450 3A5 | enzyme |
Estradiol cypionate | Cytochrome P450 3A7 | enzyme |
Estradiol cypionate | Solute carrier family 22 member 2 | transporter |
Estradiol cypionate | Solute carrier family 22 member 1 | transporter |
Estradiol cypionate | Solute carrier family 22 member 3 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 2B1 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 1A2 | transporter |
Estradiol cypionate | Multidrug resistance-associated protein 7 | transporter |
Estradiol cypionate | Solute carrier family 22 member 11 | transporter |
Estradiol cypionate | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol cypionate | P-glycoprotein 1 | transporter |
Estradiol cypionate | Cytochrome P450 1A1 | enzyme |
Estradiol cypionate | Cytochrome P450 1B1 | enzyme |
Estradiol cypionate | Cytochrome P450 2C19 | enzyme |
Estradiol cypionate | Cytochrome P450 2C8 | enzyme |
Estradiol cypionate | Cytochrome P450 2C9 | enzyme |
Estradiol cypionate | Solute carrier family 22 member 8 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol cypionate | Solute carrier organic anion transporter family member 4A1 | transporter |
Estradiol cypionate | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol cypionate | Nuclear receptor coactivator 2 | target |
Estradiol cypionate | G-protein coupled estrogen receptor 1 | target |
Estradiol cypionate | ATP synthase subunit a | target |
Estradiol cypionate | Beclin-1 | target |
Estradiol cypionate | Estradiol 17-beta-dehydrogenase 2 | target |
Estradiol cypionate | Estrogen-related receptor gamma | target |
Estradiol dienanthate | Estrogen receptor alpha | target |
Estradiol dienanthate | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol dienanthate | Sex hormone-binding globulin | carrier |
Estradiol dienanthate | Estrogen receptor beta | target |
Estradiol dienanthate | Cytochrome P450 1A2 | enzyme |
Estradiol dienanthate | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol dienanthate | Serum albumin | carrier |
Estradiol dienanthate | Fatty acid-binding protein, intestinal | carrier |
Estradiol dienanthate | Cytochrome P450 3A4 | enzyme |
Estradiol dienanthate | Cytochrome P450 3A5 | enzyme |
Estradiol dienanthate | Cytochrome P450 3A7 | enzyme |
Estradiol dienanthate | Solute carrier family 22 member 2 | transporter |
Estradiol dienanthate | Solute carrier family 22 member 1 | transporter |
Estradiol dienanthate | Solute carrier family 22 member 3 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 2B1 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 1A2 | transporter |
Estradiol dienanthate | Multidrug resistance-associated protein 7 | transporter |
Estradiol dienanthate | Solute carrier family 22 member 11 | transporter |
Estradiol dienanthate | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol dienanthate | P-glycoprotein 1 | transporter |
Estradiol dienanthate | Cytochrome P450 1A1 | enzyme |
Estradiol dienanthate | Cytochrome P450 1B1 | enzyme |
Estradiol dienanthate | Cytochrome P450 2C19 | enzyme |
Estradiol dienanthate | Cytochrome P450 2C8 | enzyme |
Estradiol dienanthate | Cytochrome P450 2C9 | enzyme |
Estradiol dienanthate | Solute carrier family 22 member 8 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol dienanthate | Solute carrier organic anion transporter family member 4A1 | transporter |
Estradiol dienanthate | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol dienanthate | Nuclear receptor coactivator 2 | target |
Estradiol dienanthate | G-protein coupled estrogen receptor 1 | target |
Estradiol dienanthate | ATP synthase subunit a | target |
Estradiol dienanthate | Beclin-1 | target |
Estradiol dienanthate | Estradiol 17-beta-dehydrogenase 2 | target |
Estradiol dienanthate | Estrogen-related receptor gamma | target |
Estradiol valerate | Estrogen receptor alpha | target |
Estradiol valerate | Nuclear receptor subfamily 1 group I member 2 | target |
Estradiol valerate | Sex hormone-binding globulin | carrier |
Estradiol valerate | Estrogen receptor beta | target |
Estradiol valerate | Cytochrome P450 1A2 | enzyme |
Estradiol valerate | UDP-glucuronosyltransferase 1-1 | enzyme |
Estradiol valerate | Serum albumin | carrier |
Estradiol valerate | Fatty acid-binding protein, intestinal | carrier |
Estradiol valerate | Cytochrome P450 3A4 | enzyme |
Estradiol valerate | Cytochrome P450 3A5 | enzyme |
Estradiol valerate | Cytochrome P450 3A7 | enzyme |
Estradiol valerate | Solute carrier family 22 member 2 | transporter |
Estradiol valerate | Solute carrier family 22 member 1 | transporter |
Estradiol valerate | Solute carrier family 22 member 3 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 2B1 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 1A2 | transporter |
Estradiol valerate | Multidrug resistance-associated protein 7 | transporter |
Estradiol valerate | Solute carrier family 22 member 11 | transporter |
Estradiol valerate | ATP-binding cassette sub-family G member 2 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 1B1 | transporter |
Estradiol valerate | P-glycoprotein 1 | transporter |
Estradiol valerate | Cytochrome P450 1A1 | enzyme |
Estradiol valerate | Cytochrome P450 1B1 | enzyme |
Estradiol valerate | Cytochrome P450 2C19 | enzyme |
Estradiol valerate | Cytochrome P450 2C8 | enzyme |
Estradiol valerate | Cytochrome P450 2C9 | enzyme |
Estradiol valerate | Solute carrier family 22 member 8 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 1B3 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 1C1 | transporter |
Estradiol valerate | Solute carrier organic anion transporter family member 4A1 | transporter |
Estradiol valerate | Neuronal acetylcholine receptor subunit alpha-4 | target |
Estradiol valerate | Nuclear receptor coactivator 2 | target |
Estradiol valerate | G-protein coupled estrogen receptor 1 | target |
Estradiol valerate | ATP synthase subunit a | target |
Estradiol valerate | Beclin-1 | target |
Estradiol valerate | Estradiol 17-beta-dehydrogenase 2 | target |
Estradiol valerate | Estrogen-related receptor gamma | target |
Isavuconazole | Cytochrome P450 3A4 | enzyme |
Isavuconazole | Cytochrome P450 3A5 | enzyme |
Isavuconazole | Cytochrome P450 2C8 | enzyme |
Isavuconazole | Cytochrome P450 2C9 | enzyme |
Isavuconazole | Cytochrome P450 2C19 | enzyme |
Isavuconazole | Cytochrome P450 2D6 | enzyme |
Isavuconazole | Cytochrome P450 2B6 | enzyme |
Isavuconazole | UDP-glucuronosyltransferase 1-9 | enzyme |
Isavuconazole | UDP-glucuronosyltransferase 1-8 | enzyme |
Isavuconazole | P-glycoprotein 1 | transporter |
Isavuconazole | ATP-binding cassette sub-family G member 2 | transporter |
Isavuconazole | Solute carrier family 22 member 2 | transporter |
Isavuconazole | Lanosterol 14-alpha demethylase | target |
Isavuconazole | Potassium voltage-gated channel subfamily H member 2 | target |
Isavuconazole | Voltage-dependent L-type calcium channel subunit alpha-1C | target |
Isavuconazole | G protein-activated inward rectifier potassium channel 2 | target |
Isavuconazole | G protein-activated inward rectifier potassium channel 3 | target |
Isavuconazole | ATP-sensitive inward rectifier potassium channel 11 | target |
Isavuconazole | Potassium voltage-gated channel subfamily A member 5 | target |
Isavuconazole | Potassium voltage-gated channel subfamily D member 3 | target |
Isavuconazole | Potassium voltage-gated channel subfamily KQT member 1 | target |
Isavuconazole | Sodium channel protein type 5 subunit alpha | target |
Nabiximols | Cannabinoid receptor 1 | target |
Nabiximols | Cannabinoid receptor 2 | target |
Nabiximols | G-protein coupled receptor 12 | target |
Nabiximols | Cytochrome P450 2C9 | enzyme |
Nabiximols | Cytochrome P450 2C19 | enzyme |
Nabiximols | Cytochrome P450 2D6 | enzyme |
Nabiximols | Cytochrome P450 3A4 | enzyme |
Nabiximols | Glycine receptor subunit alpha-1 | target |
Nabiximols | Glycine receptor (alpha-1/beta) | target |
Nabiximols | Glycine receptor subunit alpha-3 | target |
Nabiximols | N-arachidonyl glycine receptor | target |
Nabiximols | G-protein coupled receptor 55 | target |
Nabiximols | 5-hydroxytryptamine receptor 1A | target |
Nabiximols | 5-hydroxytryptamine receptor 2A | target |
Nabiximols | Neuronal acetylcholine receptor subunit alpha-7 | target |
Nabiximols | Delta-type opioid receptor | target |
Nabiximols | Mu-type opioid receptor | target |
Nabiximols | Peroxisome proliferator-activated receptor gamma | target |
Nabiximols | Cytochrome P450 3A5 | enzyme |
Nabiximols | Arachidonate 5-lipoxygenase | enzyme |
Nabiximols | Arachidonate 15-lipoxygenase | enzyme |
Nabiximols | Multidrug resistance-associated protein 1 | transporter |
Nabiximols | ATP-binding cassette sub-family G member 2 | transporter |
Nabiximols | Equilibrative nucleoside transporter 1 | transporter |
Nabiximols | Transient receptor potential cation channel subfamily V member 1 | target |
Nabiximols | Voltage-dependent T-type calcium channel subunit alpha-1G | target |
Nabiximols | Voltage-dependent T-type calcium channel subunit alpha-1H | target |
Nabiximols | Voltage-dependent T-type calcium channel subunit alpha-1I | target |
Nabiximols | Transient receptor potential cation channel subfamily A member 1 | target |
Nabiximols | Transient receptor potential cation channel subfamily M member 8 | target |
Nabiximols | Transient receptor potential cation channel subfamily V member 2 | target |
Nabiximols | Transient receptor potential cation channel subfamily V member 3 | target |
Nabiximols | Transient receptor potential cation channel subfamily V member 4 | target |
Nabiximols | Voltage-dependent anion-selective channel protein 1 | target |
Nabiximols | Prostaglandin G/H synthase 1 | target |
Nabiximols | Prostaglandin G/H synthase 2 | target |
Nabiximols | Acetyl-CoA acetyltransferase, mitochondrial | target |
Nabiximols | Steroid 17-alpha-hydroxylase/17,20 lyase | target |
Nabiximols | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | target |
Nabiximols | Glutathione reductase, mitochondrial | target |
Nabiximols | Glutathione peroxidase 1 | target |
Nabiximols | Indoleamine 2,3-dioxygenase 1 | target |
Nabiximols | Arylalkylamine N-acetyltransferase | target |
Nabiximols | Cytochrome P450 1B1 | target |
Nabiximols | Cytochrome P450 3A5 | target |
Nabiximols | Cytochrome P450 2D6 | target |
Nabiximols | Cytochrome P450 1A2 | target |
Nabiximols | Cytochrome P450 1A1 | target |
Nabiximols | Cytochrome P450 3A7 | target |
Nabiximols | Quinone oxidoreductase | target |
Nabiximols | Catalase | target |
Nabiximols | Fatty-acid amide hydrolase 1 | target |
Nabiximols | Superoxide dismutase [Cu-Zn] | target |
Nabiximols | N-acylethanolamine-hydrolyzing acid amidase | target |
Medical Cannabis | Cannabinoid receptor 1 | target |
Medical Cannabis | Cannabinoid receptor 2 | target |
Medical Cannabis | Cytochrome P450 2C9 | enzyme |
Medical Cannabis | Cytochrome P450 2C19 | enzyme |
Medical Cannabis | Cytochrome P450 2D6 | enzyme |
Medical Cannabis | Cytochrome P450 3A4 | enzyme |
Medical Cannabis | G-protein coupled receptor 12 | target |
Medical Cannabis | Glycine receptor subunit alpha-1 | target |
Medical Cannabis | Glycine receptor (alpha-1/beta) | target |
Medical Cannabis | Glycine receptor subunit alpha-3 | target |
Medical Cannabis | N-arachidonyl glycine receptor | target |
Medical Cannabis | G-protein coupled receptor 55 | target |
Medical Cannabis | 5-hydroxytryptamine receptor 1A | target |
Medical Cannabis | 5-hydroxytryptamine receptor 2A | target |
Medical Cannabis | Neuronal acetylcholine receptor subunit alpha-7 | target |
Medical Cannabis | Delta-type opioid receptor | target |
Medical Cannabis | Mu-type opioid receptor | target |
Medical Cannabis | Peroxisome proliferator-activated receptor gamma | target |
Medical Cannabis | Cytochrome P450 3A5 | enzyme |
Medical Cannabis | Cytochrome P450 3A7 | enzyme |
Medical Cannabis | Cytochrome P450 1A1 | enzyme |
Medical Cannabis | Cytochrome P450 1A2 | enzyme |
Medical Cannabis | Cytochrome P450 1B1 | enzyme |
Medical Cannabis | Arachidonate 5-lipoxygenase | enzyme |
Medical Cannabis | Arachidonate 15-lipoxygenase | enzyme |
Medical Cannabis | Superoxide dismutase [Cu-Zn] | enzyme |
Medical Cannabis | Multidrug resistance-associated protein 1 | transporter |
Medical Cannabis | ATP-binding cassette sub-family G member 2 | transporter |
Medical Cannabis | Equilibrative nucleoside transporter 1 | transporter |
Medical Cannabis | Transient receptor potential cation channel subfamily V member 1 | target |
Medical Cannabis | Voltage-dependent T-type calcium channel subunit alpha-1G | target |
Medical Cannabis | Voltage-dependent T-type calcium channel subunit alpha-1H | target |
Medical Cannabis | Voltage-dependent T-type calcium channel subunit alpha-1I | target |
Medical Cannabis | Transient receptor potential cation channel subfamily A member 1 | target |
Medical Cannabis | Transient receptor potential cation channel subfamily M member 8 | target |
Medical Cannabis | Transient receptor potential cation channel subfamily V member 2 | target |
Medical Cannabis | Transient receptor potential cation channel subfamily V member 3 | target |
Medical Cannabis | Transient receptor potential cation channel subfamily V member 4 | target |
Medical Cannabis | Voltage-dependent anion-selective channel protein 1 | target |
Medical Cannabis | N-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D | target |
Medical Cannabis | N-acylethanolamine-hydrolyzing acid amidase | target |
Medical Cannabis | Arylalkylamine N-acetyltransferase | target |
Medical Cannabis | Phospholipase A2 | target |
Medical Cannabis | Superoxide dismutase [Cu-Zn] | target |
Medical Cannabis | Fatty-acid amide hydrolase 1 | target |
Medical Cannabis | Catalase | target |
Medical Cannabis | Quinone oxidoreductase | target |
Medical Cannabis | Sphingomyelin phosphodiesterase | target |
Medical Cannabis | Glutathione peroxidase 1 | target |
Medical Cannabis | Glutathione reductase, mitochondrial | target |
Medical Cannabis | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | target |
Medical Cannabis | Indoleamine 2,3-dioxygenase 1 | target |
Medical Cannabis | Prostaglandin G/H synthase 1 | target |
Medical Cannabis | Prostaglandin G/H synthase 2 | target |
Medical Cannabis | Steroid 17-alpha-hydroxylase/17,20 lyase | target |
Medical Cannabis | Acetyl-CoA acetyltransferase, mitochondrial | target |
Medical Cannabis | Cytochrome P450 2A6 | enzyme |
Medical Cannabis | Cytochrome P450 2B6 | enzyme |
Medical Cannabis | Cytochrome P450 2C8 | enzyme |
Medical Cannabis | Cytochrome P450 2E1 | enzyme |
Medical Cannabis | Cytochrome P450 2J2 | enzyme |
Medical Cannabis | UDP-glucuronosyltransferase 1-7 | enzyme |
Medical Cannabis | UDP-glucuronosyltransferase 1-8 | enzyme |
Medical Cannabis | UDP-glucuronosyltransferase 1-9 | enzyme |
Medical Cannabis | UDP-glucuronosyltransferase 1-10 | enzyme |
Medical Cannabis | UDP-glucuronosyltransferase 2B17 | enzyme |
Medical Cannabis | Liver carboxylesterase 1 | enzyme |
Medical Cannabis | P-glycoprotein 1 | transporter |
Medical Cannabis | UDP-glucuronosyltransferase 2B7 | enzyme |
Avatrombopag | ATP-binding cassette sub-family G member 2 | target |
Avatrombopag | Cytochrome P450 2C8 | enzyme |
Avatrombopag | Cytochrome P450 2C9 | enzyme |
Avatrombopag | Thrombopoietin receptor | target |
Avatrombopag | P-glycoprotein 1 | transporter |
Avatrombopag | Solute carrier family 22 member 8 | target |
Gefitinib | Epidermal growth factor receptor | target |
Gefitinib | Cytochrome P450 3A4 | enzyme |
Gefitinib | Cytochrome P450 2D6 | enzyme |
Gefitinib | P-glycoprotein 1 | transporter |
Gefitinib | ATP-binding cassette sub-family G member 2 | transporter |
Gefitinib | Cytochrome P450 3A5 | enzyme |
Gefitinib | Cytochrome P450 1A1 | enzyme |
Gefitinib | Cytochrome P450 2C9 | enzyme |
Gefitinib | Cytochrome P450 2C19 | enzyme |
Gefitinib | Serum albumin | carrier |
Gefitinib | Alpha-1-acid glycoprotein 1 | carrier |
Safinamide | Amine oxidase [flavin-containing] B | target |
Safinamide | Amine oxidase [flavin-containing] A | enzyme |
Safinamide | ATP-binding cassette sub-family G member 2 | transporter |
Safinamide | Solute carrier organic anion transporter family member 3A1 | transporter |
Safinamide | Cytochrome P450 3A4 | enzyme |
Safinamide | Cytochrome P450 1A1 | enzyme |
Safinamide | Cytochrome P450 1A2 | enzyme |
Safinamide | Cytochrome P450 2D6 | enzyme |
Safinamide | Cytochrome P450 2C19 | enzyme |
Safinamide | Cytochrome P450 3A5 | enzyme |
Paritaprevir | NS3/4A protein | target |
Paritaprevir | Cytochrome P450 3A4 | enzyme |
Paritaprevir | Cytochrome P450 3A5 | enzyme |
Paritaprevir | ATP-binding cassette sub-family G member 2 | transporter |
Paritaprevir | P-glycoprotein 1 | transporter |
Paritaprevir | Solute carrier organic anion transporter family member 1B1 | transporter |
Paritaprevir | Solute carrier organic anion transporter family member 1B3 | transporter |
Paritaprevir | UDP-glucuronosyltransferase 1-1 | enzyme |
Fostamatinib | Adenosine receptor A3 | target |
Fostamatinib | vesicular monoamine transporter 2 (VMAT2) | target |
Fostamatinib | Fatty-acid amide hydrolase 1 | target |
Fostamatinib | Equilibrative nucleoside transporter 1 | target |
Fostamatinib | UDP-glucuronosyltransferase 1-1 | target |
Fostamatinib | cGMP-specific 3',5'-cyclic phosphodiesterase | target |
Fostamatinib | Arachidonate 5-lipoxygenase | target |
Fostamatinib | Cathepsin S | target |
Fostamatinib | Cathepsin L1 | target |
Fostamatinib | Tyrosine-protein kinase ABL1 | target |
Fostamatinib | Calcium-dependent protein kinase 1 | target |
Fostamatinib | Serine/threonine-protein kinase PknB | target |
Fostamatinib | Ribosomal protein S6 kinase alpha-6 | target |
Fostamatinib | Non-receptor tyrosine-protein kinase TYK2 | target |
Fostamatinib | Atypical kinase COQ8A, mitochondrial | target |
Fostamatinib | Tyrosine-protein kinase JAK1 | target |
Fostamatinib | Hepatocyte growth factor receptor | target |
Fostamatinib | Serine/threonine-protein kinase NIM1 | target |
Fostamatinib | Serine/threonine-protein kinase MST4 | target |
Fostamatinib | cAMP-dependent protein kinase catalytic subunit alpha | target |
Fostamatinib | Serine/threonine-protein kinase 24 | target |
Fostamatinib | Serine/threonine-protein kinase 3 | target |
Fostamatinib | Tyrosine-protein kinase Tec | target |
Fostamatinib | Tyrosine-protein kinase SYK | target |
Fostamatinib | Serine/threonine-protein kinase 33 | target |
Fostamatinib | Serine/threonine-protein kinase 35 | target |
Fostamatinib | Serine/threonine-protein kinase 36 | target |
Fostamatinib | Serine/threonine-protein kinase 38 | target |
Fostamatinib | Serine/threonine-protein kinase 38-like | target |
Fostamatinib | STE20/SPS1-related proline-alanine-rich protein kinase | target |
Fostamatinib | Serine/threonine-protein kinase TAO1 | target |
Fostamatinib | Serine/threonine-protein kinase TAO2 | target |
Fostamatinib | Serine/threonine-protein kinase TAO3 | target |
Fostamatinib | Serine/threonine-protein kinase TBK1 | target |
Fostamatinib | Angiopoietin-1 receptor | target |
Fostamatinib | Dual specificity testis-specific protein kinase 1 | target |
Fostamatinib | TGF-beta receptor type-1 | target |
Fostamatinib | TGF-beta receptor type-2 | target |
Fostamatinib | Tyrosine-protein kinase receptor Tie-1 | target |
Fostamatinib | Serine/threonine-protein kinase tousled-like 1 | target |
Fostamatinib | Serine/threonine-protein kinase tousled-like 2 | target |
Fostamatinib | TRAF2 and NCK-interacting protein kinase | target |
Fostamatinib | Non-receptor tyrosine-protein kinase TNK1 | target |
Fostamatinib | Activated CDC42 kinase 1 | target |
Fostamatinib | Serine/threonine-protein kinase TNNI3K | target |
Fostamatinib | Testis-specific serine/threonine-protein kinase 1 | target |
Fostamatinib | Dual specificity protein kinase TTK | target |
Fostamatinib | Tyrosine-protein kinase TXK | target |
Fostamatinib | Tyrosine-protein kinase receptor TYRO3 | target |
Fostamatinib | Serine/threonine-protein kinase ULK1 | target |
Fostamatinib | Serine/threonine-protein kinase ULK2 | target |
Fostamatinib | Serine/threonine-protein kinase ULK3 | target |
Fostamatinib | Wee1-like protein kinase | target |
Fostamatinib | Tyrosine-protein kinase Yes | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 19 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase MLT | target |
Fostamatinib | Tyrosine-protein kinase ZAP-70 | target |
Fostamatinib | AP2-associated protein kinase 1 | target |
Fostamatinib | Abelson tyrosine-protein kinase 2 | target |
Fostamatinib | Activin receptor type-1 | target |
Fostamatinib | Activin receptor type-1B | target |
Fostamatinib | Atypical kinase COQ8B, mitochondrial | target |
Fostamatinib | ALK tyrosine kinase receptor | target |
Fostamatinib | Ankyrin repeat and protein kinase domain-containing protein 1 | target |
Fostamatinib | Aurora kinase A | target |
Fostamatinib | Aurora kinase B | target |
Fostamatinib | Aurora kinase C | target |
Fostamatinib | Tyrosine-protein kinase receptor UFO | target |
Fostamatinib | Tyrosine-protein kinase Blk | target |
Fostamatinib | BMP-2-inducible protein kinase | target |
Fostamatinib | Bone morphogenetic protein receptor type-1B | target |
Fostamatinib | Bone morphogenetic protein receptor type-2 | target |
Fostamatinib | Cytoplasmic tyrosine-protein kinase BMX | target |
Fostamatinib | Serine/threonine-protein kinase B-raf | target |
Fostamatinib | Tyrosine-protein kinase BTK | target |
Fostamatinib | Calcium/calmodulin-dependent protein kinase type 1 | target |
Fostamatinib | Calcium/calmodulin-dependent protein kinase type 1D | target |
Fostamatinib | Calcium/calmodulin-dependent protein kinase type 1G | target |
Fostamatinib | Calcium/calmodulin-dependent protein kinase type II subunit alpha | target |
Fostamatinib | Calcium/calmodulin-dependent protein kinase type II subunit beta | target |
Fostamatinib | Calcium/calmodulin-dependent protein kinase type II subunit delta | target |
Fostamatinib | Calcium/calmodulin-dependent protein kinase type II subunit gamma | target |
Fostamatinib | Calcium/calmodulin-dependent protein kinase kinase 1 | target |
Fostamatinib | Calcium/calmodulin-dependent protein kinase kinase 2 | target |
Fostamatinib | Peripheral plasma membrane protein CASK | target |
Fostamatinib | Kappa-casein | target |
Fostamatinib | Cyclin-dependent kinase 1 | target |
Fostamatinib | Serine/threonine-protein kinase MRCK gamma | target |
Fostamatinib | Cyclin-dependent kinase 4 | target |
Fostamatinib | Cyclin-dependent kinase-like 1 | target |
Fostamatinib | Cyclin-dependent kinase-like 2 | target |
Fostamatinib | Serine/threonine-protein kinase Chk1 | target |
Fostamatinib | Serine/threonine-protein kinase Chk2 | target |
Fostamatinib | Citron Rho-interacting kinase | target |
Fostamatinib | Dual specificity protein kinase CLK1 | target |
Fostamatinib | Dual specificity protein kinase CLK2 | target |
Fostamatinib | Dual specificity protein kinase CLK3 | target |
Fostamatinib | Dual specificity protein kinase CLK4 | target |
Fostamatinib | Macrophage colony-stimulating factor 1 receptor | target |
Fostamatinib | Tyrosine-protein kinase CSK | target |
Fostamatinib | Casein kinase I isoform alpha | target |
Fostamatinib | Casein kinase II subunit alpha | target |
Fostamatinib | Casein kinase II subunit alpha' | target |
Fostamatinib | Death-associated protein kinase 1 | target |
Fostamatinib | Death-associated protein kinase 2 | target |
Fostamatinib | Death-associated protein kinase 3 | target |
Fostamatinib | Serine/threonine-protein kinase DCLK1 | target |
Fostamatinib | Serine/threonine-protein kinase DCLK2 | target |
Fostamatinib | Serine/threonine-protein kinase DCLK3 | target |
Fostamatinib | Epithelial discoidin domain-containing receptor 1 | target |
Fostamatinib | Discoidin domain-containing receptor 2 | target |
Fostamatinib | Dual specificity tyrosine-phosphorylation-regulated kinase 1A | target |
Fostamatinib | Dual specificity tyrosine-phosphorylation-regulated kinase 1B | target |
Fostamatinib | Epidermal growth factor receptor | target |
Fostamatinib | Eukaryotic translation initiation factor 2-alpha kinase 1 | target |
Fostamatinib | Interferon-induced, double-stranded RNA-activated protein kinase | target |
Fostamatinib | eIF-2-alpha kinase GCN2 | target |
Fostamatinib | Ephrin type-A receptor 1 | target |
Fostamatinib | Ephrin type-A receptor 2 | target |
Fostamatinib | Ephrin type-A receptor 3 | target |
Fostamatinib | Ephrin type-A receptor 4 | target |
Fostamatinib | Ephrin type-A receptor 5 | target |
Fostamatinib | Ephrin type-A receptor 6 | target |
Fostamatinib | Ephrin type-A receptor 7 | target |
Fostamatinib | Ephrin type-A receptor 8 | target |
Fostamatinib | Ephrin type-B receptor 1 | target |
Fostamatinib | Ephrin type-B receptor 2 | target |
Fostamatinib | Ephrin type-B receptor 4 | target |
Fostamatinib | Ephrin type-B receptor 6 | target |
Fostamatinib | Receptor tyrosine-protein kinase erbB-2 | target |
Fostamatinib | Receptor tyrosine-protein kinase erbB-4 | target |
Fostamatinib | Serine/threonine-protein kinase/endoribonuclease IRE1 | target |
Fostamatinib | Tyrosine-protein kinase Fer | target |
Fostamatinib | Tyrosine-protein kinase Fes/Fps | target |
Fostamatinib | Fibroblast growth factor receptor 1 | target |
Fostamatinib | Fibroblast growth factor receptor 2 | target |
Fostamatinib | Fibroblast growth factor receptor 3 | target |
Fostamatinib | Tyrosine-protein kinase Fgr | target |
Fostamatinib | Vascular endothelial growth factor receptor 1 | target |
Fostamatinib | Receptor-type tyrosine-protein kinase FLT3 | target |
Fostamatinib | Vascular endothelial growth factor receptor 3 | target |
Fostamatinib | Serine/threonine-protein kinase mTOR | target |
Fostamatinib | Tyrosine-protein kinase FRK | target |
Fostamatinib | Tyrosine-protein kinase Fyn | target |
Fostamatinib | Cyclin-G-associated kinase | target |
Fostamatinib | Glycogen synthase kinase-3 alpha | target |
Fostamatinib | Glycogen synthase kinase-3 beta | target |
Fostamatinib | Tyrosine-protein kinase HCK | target |
Fostamatinib | Homeodomain-interacting protein kinase 2 | target |
Fostamatinib | Homeodomain-interacting protein kinase 3 | target |
Fostamatinib | Serine/threonine-protein kinase ICK | target |
Fostamatinib | Inhibitor of nuclear factor kappa-B kinase subunit beta | target |
Fostamatinib | Inhibitor of nuclear factor kappa-B kinase subunit epsilon | target |
Fostamatinib | Insulin receptor | target |
Fostamatinib | Insulin receptor-related protein | target |
Fostamatinib | Interleukin-1 receptor-associated kinase 1 | target |
Fostamatinib | Interleukin-1 receptor-associated kinase 3 | target |
Fostamatinib | Interleukin-1 receptor-associated kinase 4 | target |
Fostamatinib | Tyrosine-protein kinase ITK/TSK | target |
Fostamatinib | Tyrosine-protein kinase JAK2 | target |
Fostamatinib | Tyrosine-protein kinase JAK3 | target |
Fostamatinib | Vascular endothelial growth factor receptor 2 | target |
Fostamatinib | Serine/threonine-protein kinase SIK3 | target |
Fostamatinib | Mast/stem cell growth factor receptor Kit | target |
Fostamatinib | Serine/threonine-protein kinase LATS1 | target |
Fostamatinib | Tyrosine-protein kinase Lck | target |
Fostamatinib | LIM domain kinase 1 | target |
Fostamatinib | LIM domain kinase 2 | target |
Fostamatinib | Leucine-rich repeat serine/threonine-protein kinase 2 | target |
Fostamatinib | Leukocyte tyrosine kinase receptor | target |
Fostamatinib | Tyrosine-protein kinase Lyn | target |
Fostamatinib | Dual specificity mitogen-activated protein kinase kinase 2 | target |
Fostamatinib | Dual specificity mitogen-activated protein kinase kinase 3 | target |
Fostamatinib | Dual specificity mitogen-activated protein kinase kinase 5 | target |
Fostamatinib | Dual specificity mitogen-activated protein kinase kinase 6 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 1 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 10 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 11 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 12 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 13 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 15 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 2 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 3 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 4 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 6 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase 9 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase kinase 1 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase kinase 2 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase kinase 3 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase kinase 4 | target |
Fostamatinib | Mitogen-activated protein kinase kinase kinase kinase 5 | target |
Fostamatinib | Mitogen-activated protein kinase 10 | target |
Fostamatinib | Mitogen-activated protein kinase 13 | target |
Fostamatinib | Mitogen-activated protein kinase 14 | target |
Fostamatinib | Mitogen-activated protein kinase 15 | target |
Fostamatinib | Mitogen-activated protein kinase 4 | target |
Fostamatinib | Mitogen-activated protein kinase 7 | target |
Fostamatinib | Mitogen-activated protein kinase 9 | target |
Fostamatinib | MAP kinase-activated protein kinase 5 | target |
Fostamatinib | Serine/threonine-protein kinase MARK1 | target |
Fostamatinib | Serine/threonine-protein kinase MARK2 | target |
Fostamatinib | MAP/microtubule affinity-regulating kinase 3 | target |
Fostamatinib | MAP/microtubule affinity-regulating kinase 4 | target |
Fostamatinib | CLIP-associating protein 1 | target |
Fostamatinib | Microtubule-associated serine/threonine-protein kinase 1 | target |
Fostamatinib | Megakaryocyte-associated tyrosine-protein kinase | target |
Fostamatinib | Maternal embryonic leucine zipper kinase | target |
Fostamatinib | Tyrosine-protein kinase Mer | target |
Fostamatinib | Misshapen-like kinase 1 | target |
Fostamatinib | MAP kinase-interacting serine/threonine-protein kinase 1 | target |
Fostamatinib | MAP kinase-interacting serine/threonine-protein kinase 2 | target |
Fostamatinib | Macrophage-stimulating protein receptor | target |
Fostamatinib | Muscle, skeletal receptor tyrosine-protein kinase | target |
Fostamatinib | Myosin light chain kinase, smooth muscle | target |
Fostamatinib | Myosin light chain kinase 2, skeletal/cardiac muscle | target |
Fostamatinib | Myosin light chain kinase 3 | target |
Fostamatinib | Myosin light chain kinase family member 4 | target |
Fostamatinib | Myosin-IIIa | target |
Fostamatinib | Serine/threonine-protein kinase Nek1 | target |
Fostamatinib | Serine/threonine-protein kinase Nek11 | target |
Fostamatinib | Serine/threonine-protein kinase Nek2 | target |
Fostamatinib | Serine/threonine-protein kinase Nek3 | target |
Fostamatinib | Serine/threonine-protein kinase Nek4 | target |
Fostamatinib | Serine/threonine-protein kinase Nek5 | target |
Fostamatinib | Serine/threonine-protein kinase Nek9 | target |
Fostamatinib | High affinity nerve growth factor receptor | target |
Fostamatinib | BDNF/NT-3 growth factors receptor | target |
Fostamatinib | NT-3 growth factor receptor | target |
Fostamatinib | NUAK family SNF1-like kinase 1 | target |
Fostamatinib | NUAK family SNF1-like kinase 2 | target |
Fostamatinib | Serine/threonine-protein kinase OSR1 | target |
Fostamatinib | Serine/threonine-protein kinase PAK 1 | target |
Fostamatinib | Serine/threonine-protein kinase PAK 2 | target |
Fostamatinib | Serine/threonine-protein kinase PAK 3 | target |
Fostamatinib | Serine/threonine-protein kinase PAK 4 | target |
Fostamatinib | Serine/threonine-protein kinase PAK 6 | target |
Fostamatinib | Serine/threonine-protein kinase PAK 5 | target |
Fostamatinib | Cyclin-dependent kinase 16 | target |
Fostamatinib | Cyclin-dependent kinase 17 | target |
Fostamatinib | Platelet-derived growth factor receptor alpha | target |
Fostamatinib | Platelet-derived growth factor receptor beta | target |
Fostamatinib | 3-phosphoinositide-dependent protein kinase 1 | target |
Fostamatinib | Cyclin-dependent kinase 15 | target |
Fostamatinib | Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform | target |
Fostamatinib | Phosphatidylinositol 4-kinase beta | target |
Fostamatinib | Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta | target |
Fostamatinib | Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma | target |
Fostamatinib | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | target |
Fostamatinib | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | target |
Fostamatinib | Serine/threonine-protein kinase pim-1 | target |
Fostamatinib | Serine/threonine-protein kinase pim-3 | target |
Fostamatinib | Phosphatidylinositol 5-phosphate 4-kinase type-2 beta | target |
Fostamatinib | Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma | target |
Fostamatinib | Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | target |
Fostamatinib | Serine/threonine-protein kinase N1 | target |
Fostamatinib | Serine/threonine-protein kinase N2 | target |
Fostamatinib | Serine/threonine-protein kinase PLK1 | target |
Fostamatinib | Serine/threonine-protein kinase PLK2 | target |
Fostamatinib | Serine/threonine-protein kinase PLK3 | target |
Fostamatinib | Serine/threonine-protein kinase PLK4 | target |
Fostamatinib | 5'-AMP-activated protein kinase catalytic subunit alpha-1 | target |
Fostamatinib | 5'-AMP-activated protein kinase | target |
Fostamatinib | cAMP-dependent protein kinase catalytic subunit beta | target |
Fostamatinib | Protein kinase C delta type | target |
Fostamatinib | Protein kinase C epsilon type | target |
Fostamatinib | Protein kinase C gamma type (PRKCG) | target |
Fostamatinib | Protein kinase C iota type | target |
Fostamatinib | Protein kinase C theta type | target |
Fostamatinib | Serine/threonine-protein kinase D1 | target |
Fostamatinib | cGMP-dependent protein kinase 2 | target |
Fostamatinib | Serine/threonine-protein kinase PRP4 homolog | target |
Fostamatinib | Focal adhesion kinase 1 | target |
Fostamatinib | Protein-tyrosine kinase 2-beta | target |
Fostamatinib | Protein-tyrosine kinase 6 | target |
Fostamatinib | RAF proto-oncogene serine/threonine-protein kinase | target |
Fostamatinib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Fostamatinib | Serine/threonine-protein kinase RIO1 | target |
Fostamatinib | Serine/threonine-protein kinase RIO2 | target |
Fostamatinib | Serine/threonine-protein kinase RIO3 | target |
Fostamatinib | Receptor-interacting serine/threonine-protein kinase 1 | target |
Fostamatinib | Receptor-interacting serine/threonine-protein kinase 2 | target |
Fostamatinib | Receptor-interacting serine/threonine-protein kinase 4 | target |
Fostamatinib | Rho-associated protein kinase 2 | target |
Fostamatinib | Proto-oncogene tyrosine-protein kinase ROS | target |
Fostamatinib | Ribosomal protein S6 kinase alpha-1 | target |
Fostamatinib | Ribosomal protein S6 kinase alpha-3 | target |
Fostamatinib | Serine/threonine-protein kinase SBK1 | target |
Fostamatinib | Uncharacterized serine/threonine-protein kinase SBK3 | target |
Fostamatinib | Serine/threonine-protein kinase Sgk3 | target |
Fostamatinib | Serine/threonine-protein kinase SIK1 | target |
Fostamatinib | Serine/threonine-protein kinase SIK2 | target |
Fostamatinib | STE20-like serine/threonine-protein kinase | target |
Fostamatinib | SNF-related serine/threonine-protein kinase | target |
Fostamatinib | Proto-oncogene tyrosine-protein kinase Src | target |
Fostamatinib | Tyrosine-protein kinase Srms | target |
Fostamatinib | Serine/threonine-protein kinase 10 | target |
Fostamatinib | Serine/threonine-protein kinase 16 | target |
Fostamatinib | Serine/threonine-protein kinase 17A | target |
Fostamatinib | Serine/threonine-protein kinase 17B | target |
Fostamatinib | Serine/threonine-protein kinase 32A | target |
Fostamatinib | Cytochrome P450 3A4 | enzyme |
Fostamatinib | ATP-binding cassette sub-family G member 2 | transporter |
Fostamatinib | ATP-binding cassette sub-family B member 5 | transporter |
Fostamatinib | UDP-glucuronosyltransferase 1-9 | enzyme |
Lansoprazole | Potassium-transporting ATPase alpha chain 1 | target |
Lansoprazole | Cytochrome P450 2C19 | enzyme |
Lansoprazole | Cytochrome P450 2C9 | enzyme |
Lansoprazole | Cytochrome P450 3A4 | enzyme |
Lansoprazole | P-glycoprotein 1 | transporter |
Lansoprazole | ATP-binding cassette sub-family G member 2 | transporter |
Lansoprazole | Cytochrome P450 1A1 | enzyme |
Lansoprazole | Cytochrome P450 1B1 | enzyme |
Lansoprazole | Cytochrome P450 2C18 | enzyme |
Lansoprazole | Cytochrome P450 2C8 | enzyme |
Lansoprazole | Cytochrome P450 2D6 | enzyme |
Lansoprazole | Microtubule-associated protein tau | target |
Lansoprazole | Solute carrier family 22 member 8 | transporter |
Lansoprazole | Solute carrier family 22 member 1 | transporter |
Lansoprazole | Solute carrier family 22 member 2 | transporter |
Lansoprazole | Solute carrier family 22 member 3 | transporter |
Pravastatin | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | target |
Pravastatin | Solute carrier organic anion transporter family member 2B1 | transporter |
Pravastatin | P-glycoprotein 1 | transporter |
Pravastatin | Solute carrier organic anion transporter family member 1A2 | transporter |
Pravastatin | Solute carrier family 22 member 6 | transporter |
Pravastatin | Solute carrier family 22 member 8 | transporter |
Pravastatin | Canalicular multispecific organic anion transporter 1 | transporter |
Pravastatin | Solute carrier family 22 member 11 | transporter |
Pravastatin | ATP-binding cassette sub-family G member 2 | transporter |
Pravastatin | Solute carrier family 22 member 7 | transporter |
Pravastatin | Solute carrier organic anion transporter family member 1B1 | transporter |
Pravastatin | Monocarboxylate transporter 1 | transporter |
Pravastatin | Bile salt export pump | transporter |
Pravastatin | Solute carrier organic anion transporter family member 1B3 | transporter |
Pravastatin | Histone deacetylase 2 | target |
Dovitinib | Cytochrome P450 1A1 | enzyme |
Dovitinib | Cytochrome P450 1A2 | enzyme |
Dovitinib | Canalicular multispecific organic anion transporter 2 | transporter |
Dovitinib | ATP-binding cassette sub-family G member 2 | transporter |
Dovitinib | UDP-glucuronosyltransferase 1-3 | enzyme |
Dovitinib | UDP-glucuronosyltransferase 2B7 | enzyme |
Dovitinib | Nuclear receptor subfamily 1 group I member 2 | target |
Dovitinib | Solute carrier organic anion transporter family member 1B1 | transporter |
Dovitinib | Solute carrier organic anion transporter family member 2B1 | transporter |
Dovitinib | Cytochrome P450 2C19 | enzyme |
Dovitinib | Cytochrome P450 3A4 | enzyme |
Dovitinib | Solute carrier organic anion transporter family member 1B3 | transporter |
Dovitinib | P-glycoprotein 1 | transporter |
Eltrombopag | Thrombopoietin receptor | target |
Eltrombopag | Cytochrome P450 2C8 | enzyme |
Eltrombopag | Cytochrome P450 1A2 | enzyme |
Eltrombopag | UDP-glucuronosyltransferase 1-1 | enzyme |
Eltrombopag | UDP-glucuronosyltransferase 1-3 | enzyme |
Eltrombopag | Solute carrier organic anion transporter family member 1B1 | transporter |
Eltrombopag | ATP-binding cassette sub-family G member 2 | transporter |
Eltrombopag | UDP-glucuronosyltransferase 1-9 | enzyme |
Teriflunomide | ATP-binding cassette sub-family G member 2 | transporter |
Teriflunomide | Dihydroorotate dehydrogenase (quinone), mitochondrial | target |
Teriflunomide | Cytochrome P450 2C8 | enzyme |
Teriflunomide | Solute carrier organic anion transporter family member 1B1 | transporter |
Teriflunomide | Cytochrome P450 1A2 | enzyme |
Vemurafenib | Serum albumin | carrier |
Vemurafenib | Alpha-1-acid glycoprotein 1 | carrier |
Vemurafenib | Cytochrome P450 1A2 | enzyme |
Vemurafenib | Cytochrome P450 2D6 | enzyme |
Vemurafenib | Cytochrome P450 3A4 | enzyme |
Vemurafenib | Serine/threonine-protein kinase B-raf | target |
Vemurafenib | Multidrug resistance-associated protein 1 | transporter |
Vemurafenib | ATP-binding cassette sub-family G member 2 | transporter |
Vemurafenib | Cytochrome P450 2C9 | enzyme |
Vemurafenib | Cytochrome P450 2C8 | enzyme |
Vemurafenib | Cytochrome P450 2B6 | enzyme |
Vemurafenib | P-glycoprotein 1 | transporter |
Progesterone | Progesterone receptor | target |
Progesterone | Estrogen receptor alpha | target |
Progesterone | Steroid 17-alpha-hydroxylase/17,20 lyase | target |
Progesterone | Cytochrome P450 2C19 | enzyme |
Progesterone | Cytochrome P450 2C9 | enzyme |
Progesterone | Cytochrome P450 3A4 | enzyme |
Progesterone | Cytochrome P450 3A5 | enzyme |
Progesterone | Cytochrome P450 3A7 | enzyme |
Progesterone | P-glycoprotein 1 | transporter |
Progesterone | Solute carrier family 22 member 2 | transporter |
Progesterone | Solute carrier family 22 member 1 | transporter |
Progesterone | Solute carrier family 22 member 3 | transporter |
Progesterone | Bile salt export pump | transporter |
Progesterone | Multidrug resistance-associated protein 1 | transporter |
Progesterone | Sodium/bile acid cotransporter | transporter |
Progesterone | Steroid 17-alpha-hydroxylase/17,20 lyase | enzyme |
Progesterone | Cytochrome P450 1A1 | enzyme |
Progesterone | Cytochrome P450 1B1 | enzyme |
Progesterone | Cytochrome P450 2A6 | enzyme |
Progesterone | Cytochrome P450 2D6 | enzyme |
Progesterone | Mineralocorticoid receptor | target |
Progesterone | Kappa-type opioid receptor | target |
Progesterone | Alpha-1-acid glycoprotein 1 | target |
Progesterone | Glucocorticoid receptor | target |
Progesterone | Androgen receptor | target |
Progesterone | Sex hormone-binding globulin | target |
Progesterone | Solute carrier organic anion transporter family member 1B1 | transporter |
Progesterone | ATP-binding cassette sub-family G member 2 | transporter |
Progesterone | Estrogen receptor beta | target |
Progesterone | Solute carrier organic anion transporter family member 1B3 | transporter |
Fusidic acid | Chloramphenicol acetyltransferase 3 | target |
Fusidic acid | Chloramphenicol acetyltransferase | target |
Fusidic acid | Bile salt export pump | transporter |
Fusidic acid | Canalicular multispecific organic anion transporter 1 | transporter |
Fusidic acid | Elongation factor G | target |
Fusidic acid | Cytochrome P450 2D6 | enzyme |
Fusidic acid | Cytochrome P450 3A4 | enzyme |
Fusidic acid | UDP-glucuronosyltransferase 1-1 | enzyme |
Fusidic acid | ATP-binding cassette sub-family G member 2 | transporter |
Fusidic acid | Solute carrier organic anion transporter family member 1B1 | transporter |
Netupitant | Neurokinin 1 receptor | target |
Netupitant | Cytochrome P450 3A43 | enzyme |
Netupitant | Cytochrome P450 2C9 | enzyme |
Netupitant | Cytochrome P450 2D6 | enzyme |
Netupitant | Cytochrome P450 3A4 | enzyme |
Netupitant | P-glycoprotein 1 | transporter |
Ledipasvir | Nonstructural protein 5A | target |
Ledipasvir | P-glycoprotein 1 | transporter |
Ledipasvir | ATP-binding cassette sub-family G member 2 | transporter |
Osimertinib | Epidermal growth factor receptor | target |
Osimertinib | P-glycoprotein 1 | transporter |
Osimertinib | ATP-binding cassette sub-family G member 2 | transporter |
Osimertinib | Cytochrome P450 3A4 | enzyme |
Osimertinib | Cytochrome P450 1A2 | enzyme |
Grazoprevir | P-glycoprotein 1 | transporter |
Grazoprevir | Solute carrier organic anion transporter family member 1B1 | transporter |
Grazoprevir | Solute carrier organic anion transporter family member 1B3 | transporter |
Grazoprevir | Cytochrome P450 3A4 | enzyme |
Grazoprevir | NS3/4A protein | target |
Grazoprevir | Serum albumin | carrier |
Grazoprevir | Alpha-1-acid glycoprotein 1 | carrier |
Elbasvir | Nonstructural protein 5A | target |
Elbasvir | P-glycoprotein 1 | transporter |
Elbasvir | Cytochrome P450 3A4 | enzyme |
Elbasvir | Cytochrome P450 3A5 | enzyme |
Elbasvir | Cytochrome P450 3A7 | enzyme |
Elbasvir | Cytochrome P450 3A43 | enzyme |
Sapropterin | Phenylalanine-4-hydroxylase | target |
Sapropterin | Nitric oxide synthase, endothelial | target |
Sapropterin | Tyrosine 3-monooxygenase | target |
Sapropterin | Tryptophan 5-hydroxylase 1 | target |
Sapropterin | Prostaglandin G/H synthase 2 | enzyme |
Sapropterin | P-glycoprotein 1 | transporter |
Tedizolid | 23S ribosomal RNA | target |
Tedizolid | Amine oxidase [flavin-containing] A | enzyme |
Tedizolid | Amine oxidase [flavin-containing] B | enzyme |
Dacomitinib | Cytochrome P450 2D6 | enzyme |
Dacomitinib | Serum albumin | carrier |
Dacomitinib | Cytochrome P450 3A4 | enzyme |
Dacomitinib | Cytochrome P450 2C9 | enzyme |
Dacomitinib | UDP-glucuronosyltransferase 1-1 | enzyme |
Dacomitinib | P-glycoprotein 1 | transporter |
Dacomitinib | ATP-binding cassette sub-family G member 2 | transporter |
Dacomitinib | Solute carrier family 22 member 1 | transporter |
Dacomitinib | Epidermal growth factor receptor | target |
Venetoclax | Apoptosis regulator Bcl-2 | target |
Venetoclax | Cytochrome P450 3A4 | enzyme |
Venetoclax | P-glycoprotein 1 | transporter |
Venetoclax | ATP-binding cassette sub-family G member 2 | transporter |
Venetoclax | Solute carrier organic anion transporter family member 1B1 | transporter |
Gilteritinib | Serum albumin | carrier |
Gilteritinib | Cytochrome P450 3A4 | enzyme |
Gilteritinib | Receptor-type tyrosine-protein kinase FLT3 | target |
Gilteritinib | Serotonin Receptors | target |
Gilteritinib | P-glycoprotein 1 | transporter |
Gilteritinib | Multidrug and toxin extrusion protein 1 | transporter |
Gilteritinib | ATP-binding cassette sub-family G member 2 | transporter |
Gilteritinib | Solute carrier family 22 member 1 | transporter |
Gilteritinib | Tyrosine-protein kinase receptor UFO | target |
Gilteritinib | ALK tyrosine kinase receptor | target |
Glasdegib | Cytochrome P450 3A4 | enzyme |
Glasdegib | Smoothened homolog | target |
Glasdegib | Cytochrome P450 2C8 | enzyme |
Glasdegib | UDP-glucuronosyltransferase 1-9 | enzyme |
Glasdegib | Serum albumin | carrier |
Glasdegib | P-glycoprotein 1 | transporter |
Glasdegib | ATP-binding cassette sub-family G member 2 | transporter |
Glasdegib | Multidrug and toxin extrusion protein 1 | transporter |
Glasdegib | Multidrug and toxin extrusion protein 2 | transporter |
Olaparib | Poly [ADP-ribose] polymerase 1 | target |
Olaparib | Cytochrome P450 3A4 | enzyme |
Olaparib | Cytochrome P450 2B6 | enzyme |
Olaparib | Poly [ADP-ribose] polymerase 2 | target |
Olaparib | Poly [ADP-ribose] polymerase 3 | target |
Olaparib | Cytochrome P450 3A5 | enzyme |
Olaparib | P-glycoprotein 1 | transporter |
Olaparib | ATP-binding cassette sub-family G member 2 | transporter |
Olaparib | Aldo-keto reductase family 1 member C3 | target |
Olaparib | UDP-glucuronosyltransferase 1-1 | enzyme |
Olaparib | Serum albumin | carrier |
Olaparib | Alpha-1-acid glycoprotein 1 | carrier |
Itraconazole | Lanosterol 14-alpha demethylase | target |
Itraconazole | Lanosterol 14-alpha demethylase | target |
Itraconazole | Cytochrome P450 3A4 | enzyme |
Itraconazole | Cytochrome P450 3A5 | enzyme |
Itraconazole | Cytochrome P450 3A7 | enzyme |
Itraconazole | Cytochrome P450 2B6 | enzyme |
Itraconazole | P-glycoprotein 1 | transporter |
Itraconazole | Cytochrome P450 1A1 | enzyme |
Itraconazole | Cytochrome P450 2E1 | enzyme |
Itraconazole | Solute carrier organic anion transporter family member 2B1 | transporter |
Palbociclib | Cyclin-dependent kinase 4 | target |
Palbociclib | Cyclin-dependent kinase 6 | target |
Palbociclib | Cytochrome P450 3A4 | enzyme |
Palbociclib | Bile salt sulfotransferase | enzyme |
Palbociclib | P-glycoprotein 1 | transporter |
Palbociclib | ATP-binding cassette sub-family G member 2 | transporter |
Palbociclib | Serum albumin | carrier |
Palbociclib | Solute carrier family 22 member 1 | transporter |
Alpelisib | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | target |
Alpelisib | Cytochrome P450 3A4 | enzyme |
Alpelisib | Cytochrome P450 2C9 | enzyme |
Alpelisib | Cytochrome P450 2C8 | enzyme |
Alpelisib | Cytochrome P450 2C19 | enzyme |
Alpelisib | ATP-binding cassette sub-family G member 2 | transporter |
Alpelisib | P-glycoprotein 1 | transporter |
Beclomethasone dipropionate | Corticosteroid-binding globulin | carrier |
Beclomethasone dipropionate | Glucocorticoid receptor | target |
Beclomethasone dipropionate | Cytochrome P450 3A5 | enzyme |
Beclomethasone dipropionate | Cytochrome P450 3A4 | enzyme |
Beclomethasone dipropionate | P-glycoprotein 1 | transporter |
Beclomethasone dipropionate | ATP-binding cassette sub-family G member 2 | transporter |
Beclomethasone dipropionate | Solute carrier organic anion transporter family member 1B1 | transporter |
Beclomethasone dipropionate | Solute carrier organic anion transporter family member 1B3 | transporter |
Fedratinib | P-glycoprotein 1 | transporter |
Fedratinib | ATP-binding cassette sub-family G member 2 | transporter |
Fedratinib | Solute carrier organic anion transporter family member 1B1 | transporter |
Fedratinib | Solute carrier organic anion transporter family member 1B3 | transporter |
Fedratinib | POU domain, class 2, transcription factor 2 | transporter |
Fedratinib | Multidrug and toxin extrusion protein 1 | transporter |
Fedratinib | Multidrug and toxin extrusion protein 2 | transporter |
Fedratinib | Cytochrome P450 3A4 | enzyme |
Fedratinib | Cytochrome P450 2C19 | enzyme |
Fedratinib | Dimethylaniline monooxygenase [N-oxide-forming] 3 | enzyme |
Fedratinib | Tyrosine-protein kinase JAK2 | target |
Fedratinib | Receptor-type tyrosine-protein kinase FLT3 | target |
Fedratinib | Tyrosine-protein kinase JAK1 | target |
Fedratinib | Cytochrome P450 2D6 | enzyme |
Istradefylline | Cytochrome P450 1A1 | enzyme |
Istradefylline | Cytochrome P450 3A4 | enzyme |
Istradefylline | Cytochrome P450 3A5 | enzyme |
Istradefylline | Cytochrome P450 1A2 | enzyme |
Istradefylline | Cytochrome P450 2B6 | enzyme |
Istradefylline | Cytochrome P450 2C8 | enzyme |
Istradefylline | Cytochrome P450 2C9 | enzyme |
Istradefylline | Cytochrome P450 2C18 | enzyme |
Istradefylline | Cytochrome P450 2D6 | enzyme |
Istradefylline | Cytochrome P450 3A Subfamily | enzyme |
Istradefylline | P-glycoprotein 1 | transporter |
Istradefylline | Adenosine receptor A2a | target |
Istradefylline | Adenosine receptor A1 | target |
Istradefylline | Serum albumin | carrier |
Istradefylline | alpha1-acid glycoprotein | carrier |
Istradefylline | ATP-binding cassette sub-family G member 2 | transporter |
Istradefylline | Solute carrier organic anion transporter family member 1B1 | transporter |
Istradefylline | Solute carrier organic anion transporter family member 1B3 | transporter |
Istradefylline | Solute carrier family 22 member 6 | transporter |
Istradefylline | POU domain, class 2, transcription factor 2 | transporter |
Istradefylline | Multidrug and toxin extrusion protein 1 | transporter |
Istradefylline | Multidrug and toxin extrusion protein 2 | transporter |
Caffeine | Adenosine receptor A1 | target |
Caffeine | cAMP-specific 3',5'-cyclic phosphodiesterase 4B | target |
Caffeine | Adenosine receptor A2a | target |
Caffeine | Cytochrome P450 1A2 | enzyme |
Caffeine | Ryanodine receptor 1 | target |
Caffeine | Cytochrome P450 3A4 | enzyme |
Caffeine | Cytochrome P450 2E1 | enzyme |
Caffeine | Cytochrome P450 2C8 | enzyme |
Caffeine | Cytochrome P450 2C9 | enzyme |
Caffeine | Cytochrome P450 1A1 | enzyme |
Caffeine | Cytochrome P450 1B1 | enzyme |
Caffeine | Cytochrome P450 2D6 | enzyme |
Caffeine | Cyclic nucleotide phosphodiesterase | target |
Caffeine | DNA-dependent protein kinase catalytic subunit | target |
Caffeine | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | target |
Caffeine | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | target |
Caffeine | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform | target |
Caffeine | Inositol 1,4,5-trisphosphate receptor | target |
Caffeine | Serine-protein kinase ATM | target |
Caffeine | ATP-binding cassette sub-family G member 2 | transporter |
Caffeine | Adenosine receptor A2b | target |
Caffeine | Adenosine receptor A3 | target |
Caffeine | Phosphodiesterase enzymes | target |
Lasmiditan | 5-hydroxytryptamine receptor 1F | target |
Lasmiditan | P-glycoprotein 1 | transporter |
Lasmiditan | ATP-binding cassette sub-family G member 2 | transporter |
Lasmiditan | Solute carrier family 22 member 1 | transporter |
Lasmiditan | Multidrug and toxin extrusion protein 1 | transporter |
Lasmiditan | Multidrug and toxin extrusion protein 2 | transporter |
Lasmiditan | Cytochrome P450 2D6 | enzyme |
Darolutamide | Cytochrome P450 3A4 | enzyme |
Darolutamide | UDP-glucuronosyltransferase 1-9 | enzyme |
Darolutamide | Androgen receptor | target |
Darolutamide | ATP-binding cassette sub-family G member 2 | transporter |
Darolutamide | P-glycoprotein 1 | transporter |
Darolutamide | Serum albumin | carrier |
Darolutamide | Progesterone receptor | target |
Darolutamide | Solute carrier organic anion transporter family member 1B1 | transporter |
Darolutamide | Solute carrier organic anion transporter family member 1B3 | transporter |
Upadacitinib | Tyrosine-protein kinase JAK1 | target |
Upadacitinib | Cytochrome P450 3A4 | enzyme |
Upadacitinib | Cytochrome P450 2D6 | enzyme |
Upadacitinib | P-glycoprotein 1 | transporter |
Upadacitinib | ATP-binding cassette sub-family G member 2 | transporter |
Upadacitinib | Solute carrier organic anion transporter family member 1B1 | transporter |
Tafamidis | Transthyretin | target |
Tafamidis | Solute carrier family 22 member 6 | transporter |
Tafamidis | Solute carrier family 22 member 8 | transporter |
Tafamidis | ATP-binding cassette sub-family G member 2 | transporter |
Capmatinib | Cytochrome P450 3A4 | enzyme |
Capmatinib | Aldehyde oxidase | enzyme |
Capmatinib | Hepatocyte growth factor receptor | target |
Capmatinib | P-glycoprotein 1 | transporter |
Capmatinib | Multidrug and toxin extrusion protein 1 | transporter |
Capmatinib | Multidrug and toxin extrusion protein 2 | transporter |
Capmatinib | Cytochrome P450 1A2 | enzyme |
Capmatinib | ATP-binding cassette sub-family G member 2 | transporter |
Selpercatinib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Selpercatinib | Vascular endothelial growth factor receptor 1 | target |
Selpercatinib | Vascular endothelial growth factor receptor 3 | target |
Selpercatinib | Fibroblast growth factor receptor 1 | target |
Selpercatinib | Fibroblast growth factor receptor 2 | target |
Selpercatinib | Fibroblast growth factor receptor 3 | target |
Selpercatinib | Cytochrome P450 3A4 | enzyme |
Selpercatinib | Cytochrome P450 2C8 | enzyme |
Selpercatinib | Cytochrome P450 3A Subfamily | enzyme |
Selpercatinib | P-glycoprotein 1 | transporter |
Selpercatinib | ATP-binding cassette sub-family G member 2 | transporter |
Selpercatinib | Multidrug and toxin extrusion protein 1 | transporter |
Ripretinib | Mast/stem cell growth factor receptor Kit | target |
Ripretinib | Platelet-derived growth factor receptor beta | target |
Ripretinib | Angiopoietin-1 receptor | target |
Ripretinib | Vascular endothelial growth factor receptor 2 | target |
Ripretinib | Serine/threonine-protein kinase B-raf | target |
Ripretinib | Platelet-derived growth factor receptor alpha | target |
Ripretinib | Cytochrome P450 2C8 | enzyme |
Ripretinib | Platelet-derived growth factor receptor alpha | enzyme |
Ripretinib | Serum albumin | carrier |
Ripretinib | alpha1-acid glycoprotein | carrier |
Ripretinib | P-glycoprotein 1 | transporter |
Ripretinib | ATP-binding cassette sub-family G member 2 | transporter |
Ripretinib | Multidrug and toxin extrusion protein 1 | transporter |
Ripretinib | Cytochrome P450 3A4 | enzyme |
Ripretinib | Cytochrome P450 2D6 | enzyme |
Ripretinib | Cytochrome P450 2E1 | enzyme |
Clofazimine | Cytochrome P450 3A4 | enzyme |
Clofazimine | Peroxisome proliferator-activated receptor gamma | target |
Clofazimine | Cytochrome P450 2C8 | enzyme |
Clofazimine | Cytochrome P450 2D6 | enzyme |
Clofazimine | Cytochrome P450 3A5 | enzyme |
Clofazimine | Potassium voltage-gated channel subfamily A member 3 | target |
Clofazimine | Serum albumin | carrier |
Clofazimine | P-glycoprotein 1 | transporter |
Clofazimine | ATP-binding cassette sub-family G member 2 | transporter |
Clofazimine | Multidrug resistance-associated protein 1 | transporter |
Dexamethasone acetate | Glucocorticoid receptor | target |
Dexamethasone acetate | Annexin A1 | target |
Dexamethasone acetate | Nitric oxide synthase, inducible | target |
Dexamethasone acetate | Nuclear receptor subfamily 0 group B member 1 | target |
Dexamethasone acetate | Cytochrome P450 3A4 | enzyme |
Dexamethasone acetate | Cytochrome P450 3A5 | enzyme |
Dexamethasone acetate | Cytochrome P450 3A7 | enzyme |
Dexamethasone acetate | Bile salt export pump | transporter |
Dexamethasone acetate | P-glycoprotein 1 | transporter |
Dexamethasone acetate | Canalicular multispecific organic anion transporter 1 | transporter |
Dexamethasone acetate | Solute carrier organic anion transporter family member 1A2 | transporter |
Dexamethasone acetate | ATP-binding cassette sub-family G member 2 | transporter |
Dexamethasone acetate | Steroid 17-alpha-hydroxylase/17,20 lyase | enzyme |
Dexamethasone acetate | Cytochrome P450 1A1 | enzyme |
Dexamethasone acetate | Cytochrome P450 2A6 | enzyme |
Dexamethasone acetate | Cytochrome P450 2B6 | enzyme |
Dexamethasone acetate | Cytochrome P450 2C19 | enzyme |
Dexamethasone acetate | Cytochrome P450 2C8 | enzyme |
Dexamethasone acetate | Cytochrome P450 2E1 | enzyme |
Dexamethasone acetate | Cytochrome P450 3A43 | enzyme |
Dexamethasone acetate | Cytochrome P450 4A11 | enzyme |
Dexamethasone acetate | Nuclear receptor subfamily 1 group I member 2 | target |
Dexamethasone acetate | Cytochrome P450 11B1, mitochondrial | enzyme |
Dexamethasone acetate | Serum albumin | carrier |
Dexamethasone acetate | Corticosteroid 11-beta-dehydrogenase isozyme 2 | enzyme |
Dexamethasone acetate | Corticosteroid 11-beta-dehydrogenase isozyme 1 | enzyme |
Dexamethasone acetate | Solute carrier family 22 member 8 | transporter |
Fostemsavir | Cytochrome P450 3A4 | enzyme |
Fostemsavir | UDP-glucuronosyltransferases (UGTs) | enzyme |
Fostemsavir | P-glycoprotein 1 | transporter |
Fostemsavir | ATP-binding cassette sub-family G member 2 | transporter |
Fostemsavir | Solute carrier organic anion transporter family member 1B1 | transporter |
Fostemsavir | Solute carrier organic anion transporter family member 1B3 | transporter |
Fostemsavir | Serum albumin | carrier |
Fostemsavir | Envelope glycoprotein gp160 | target |
Pralsetinib | Proto-oncogene tyrosine-protein kinase receptor Ret | target |
Pralsetinib | Epithelial discoidin domain-containing receptor 1 | target |
Pralsetinib | NT-3 growth factor receptor | target |
Pralsetinib | Receptor-type tyrosine-protein kinase FLT3 | target |
Pralsetinib | Tyrosine-protein kinase JAK1 | target |
Pralsetinib | Tyrosine-protein kinase JAK2 | target |
Pralsetinib | High affinity nerve growth factor receptor | target |
Pralsetinib | Vascular endothelial growth factor receptor 2 | target |
Pralsetinib | Platelet-derived growth factor receptor beta | target |
Pralsetinib | Fibroblast growth factor receptor 1 | target |
Pralsetinib | Fibroblast growth factor receptor 2 | target |
Pralsetinib | Cytochrome P450 3A4 | enzyme |
Pralsetinib | Cytochrome P450 3A5 | enzyme |
Pralsetinib | Cytochrome P450 2D6 | enzyme |
Pralsetinib | Cytochrome P450 1A2 | enzyme |
Pralsetinib | Cytochrome P450 2C8 | enzyme |
Pralsetinib | Cytochrome P450 2C9 | enzyme |
Pralsetinib | P-glycoprotein 1 | transporter |
Pralsetinib | ATP-binding cassette sub-family G member 2 | transporter |
Pralsetinib | Solute carrier organic anion transporter family member 1B1 | transporter |
Pralsetinib | Solute carrier organic anion transporter family member 1B3 | transporter |
Pralsetinib | Solute carrier family 22 member 6 | transporter |
Pralsetinib | Multidrug and toxin extrusion protein 1 | transporter |
Pralsetinib | Multidrug and toxin extrusion protein 2 | transporter |
Pralsetinib | Bile salt export pump | transporter |
Lonafarnib | Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha | target |
Lonafarnib | P-glycoprotein 1 | transporter |
Lonafarnib | Protein farnesyltransferase subunit beta | target |
Lonafarnib | Cytochrome P450 3A Subfamily | enzyme |
Lonafarnib | Cytochrome P450 2C8 | enzyme |
Lonafarnib | Cytochrome P450 2C19 | enzyme |
Lonafarnib | Cytochrome P450 1A2 | enzyme |
Lonafarnib | Cytochrome P450 2A6 | enzyme |
Lonafarnib | Cytochrome P450 2C9 | enzyme |
Lonafarnib | Cytochrome P450 2E1 | enzyme |
Lonafarnib | Solute carrier organic anion transporter family member 1B1 | transporter |
Lonafarnib | Solute carrier organic anion transporter family member 1B3 | transporter |
Lonafarnib | ATP-binding cassette sub-family G member 2 | transporter |
Lonafarnib | Cytochrome P450 3A4 | enzyme |
Lonafarnib | Cytochrome P450 3A5 | enzyme |
Lonafarnib | Canalicular multispecific organic anion transporter 1 | transporter |
Relugolix | Serum albumin | carrier |
Relugolix | Alpha-1-acid glycoprotein 1 | carrier |
Relugolix | P-glycoprotein 1 | transporter |
Relugolix | ATP-binding cassette sub-family G member 2 | transporter |
Relugolix | Cytochrome P450 3A Subfamily | enzyme |
Relugolix | Cytochrome P450 2C8 | enzyme |
Relugolix | Cytochrome P450 2B6 | enzyme |
Relugolix | Gonadotropin-releasing hormone receptor | target |
Tepotinib | P-glycoprotein 1 | transporter |
Tepotinib | Cytochrome P450 3A4 | enzyme |
Tepotinib | Cytochrome P450 2C8 | enzyme |
Tepotinib | ATP-binding cassette sub-family G member 2 | transporter |
Tepotinib | Hepatocyte growth factor receptor | target |
Tepotinib | Nischarin | target |
Tepotinib | Melatonin receptor type 1B | target |
Tepotinib | Serum albumin | carrier |
Tepotinib | Alpha-1-acid glycoprotein 1 | carrier |
Febuxostat | Serum albumin | carrier |
Febuxostat | Xanthine dehydrogenase/oxidase | target |
Febuxostat | UDP-glucuronosyltransferase 1-1 | enzyme |
Febuxostat | UDP-glucuronosyltransferase 1-3 | enzyme |
Febuxostat | UDP-glucuronosyltransferase 1-9 | enzyme |
Febuxostat | UDP-glucuronosyltransferase 2B7 | enzyme |
Febuxostat | Cytochrome P450 1A2 | enzyme |
Febuxostat | Cytochrome P450 2C8 | enzyme |
Febuxostat | Cytochrome P450 2C9 | enzyme |
Febuxostat | ATP-binding cassette sub-family G member 2 | transporter |
Avanafil | cGMP-specific 3',5'-cyclic phosphodiesterase | target |
Avanafil | Cytochrome P450 3A4 | enzyme |
Avanafil | Serum albumin | carrier |
Avanafil | Alpha-1-acid glycoprotein 1 | carrier |
Avanafil | P-glycoprotein 1 | transporter |
Avanafil | ATP-binding cassette sub-family G member 2 | transporter |
Avanafil | Cytochrome P450 2C9 | enzyme |
Tivozanib | Cytochrome P450 3A4 | enzyme |
Tivozanib | Serum albumin | carrier |
Tivozanib | Vascular endothelial growth factor receptor 1 | target |
Tivozanib | Vascular endothelial growth factor receptor 2 | target |
Tivozanib | Vascular endothelial growth factor receptor 3 | target |
Tivozanib | Mast/stem cell growth factor receptor Kit | target |
Tivozanib | Platelet-derived growth factor receptor beta | target |
Tivozanib | P-glycoprotein 1 | transporter |
Tivozanib | ATP-binding cassette sub-family G member 2 | transporter |
Tivozanib | Receptor-type tyrosine-protein kinase FLT3 | target |
Tivozanib | Platelet-derived growth factor receptor alpha | target |
Tivozanib | Protein-tyrosine kinase 6 | target |
Tivozanib | Angiopoietin-1 receptor | target |
Tivozanib | Fibroblast growth factor receptor 1 | target |
Tivozanib | Hepatocyte growth factor receptor | target |
Infigratinib | Cytochrome P450 3A4 | enzyme |
Infigratinib | Multidrug and toxin extrusion protein 1 | transporter |
Infigratinib | ATP-binding cassette sub-family G member 2 | transporter |
Infigratinib | Bile salt export pump | transporter |
Infigratinib | Solute carrier family 22 member 1 | transporter |
Infigratinib | Solute carrier family 22 member 2 | transporter |
Infigratinib | Multidrug and toxin extrusion protein 2 | transporter |
Infigratinib | P-glycoprotein 1 | transporter |
Infigratinib | Solute carrier organic anion transporter family member 1B1 | transporter |
Infigratinib | Solute carrier organic anion transporter family member 1B3 | transporter |
Infigratinib | Apolipoproteins | carrier |
Infigratinib | Dimethylaniline monooxygenase [N-oxide-forming] 3 | enzyme |
Infigratinib | Fibroblast growth factor receptor 1 | target |
Infigratinib | Fibroblast growth factor receptor 2 | target |
Infigratinib | Fibroblast growth factor receptor 3 | target |
Infigratinib | Fibroblast growth factor receptor 4 | target |
Sotorasib | GTPase KRas | target |
Sotorasib | Cytochrome P450 3A Subfamily | enzyme |
Sotorasib | Cytochrome P450 2C8 | enzyme |
Sotorasib | Cytochrome P450 2C9 | enzyme |
Sotorasib | Cytochrome P450 2B6 | enzyme |
Sotorasib | ATP-binding cassette sub-family G member 2 | transporter |
Sotorasib | P-glycoprotein 1 | transporter |
Tecovirimat | Envelope protein F13 | target |
Tecovirimat | UDP-glucuronosyltransferase 1-1 | enzyme |
Tecovirimat | UDP-glucuronosyltransferase 1-4 | enzyme |
Tecovirimat | Cytochrome P450 3A4 | enzyme |
Tecovirimat | Cytochrome P450 2C8 | enzyme |
Tecovirimat | Cytochrome P450 2C19 | enzyme |
Tecovirimat | UDP-glucuronosyltransferase 1-3 | enzyme |
Tecovirimat | ATP-binding cassette sub-family G member 2 | transporter |
Tecovirimat | Cytochrome P450 2B6 | enzyme |
Avapritinib | Platelet derived growth factor receptor alpha | target |
Avapritinib | Mast/stem cell growth factor receptor Kit | target |
Avapritinib | P-glycoprotein 1 | transporter |
Avapritinib | ATP-binding cassette sub-family G member 2 | transporter |
Avapritinib | Cytochrome P450 3A4 | enzyme |
Avapritinib | Cytochrome P450 2C9 | enzyme |
Avapritinib | Bile salt export pump | transporter |
Avapritinib | Multidrug and toxin extrusion protein 1 | transporter |
Avapritinib | Multidrug and toxin extrusion protein 2 | transporter |
Brincidofovir | Leukotriene-B(4) omega-hydroxylase 1 | enzyme |
Brincidofovir | Sphingomyelin phosphodiesterase | enzyme |
Brincidofovir | DNA polymerase | target |
Brincidofovir | Cytochrome P450 1A2 | enzyme |
Brincidofovir | Cytochrome P450 2B6 | enzyme |
Brincidofovir | Cytochrome P450 2C8 | enzyme |
Brincidofovir | Cytochrome P450 2C9 | enzyme |
Brincidofovir | Cytochrome P450 2C19 | enzyme |
Brincidofovir | Cytochrome P450 2D6 | enzyme |
Brincidofovir | ATP-binding cassette sub-family G member 2 | transporter |
Brincidofovir | Canalicular multispecific organic anion transporter 1 | transporter |
Brincidofovir | Bile salt export pump | transporter |
Brincidofovir | Solute carrier organic anion transporter family member 1B1 | transporter |
Brincidofovir | Solute carrier family 22 member 6 | transporter |
Brincidofovir | Solute carrier family 22 member 8 | transporter |
Brincidofovir | Solute carrier organic anion transporter family member 1B3 | transporter |
Brincidofovir | Variola virus DNA | target |
Belumosudil | Rho-associated protein kinase 2 | target |
Belumosudil | Serum albumin | carrier |
Belumosudil | Alpha-1-acid glycoprotein 1 | carrier |
Belumosudil | Rho-associated protein kinase 1 | target |
Belumosudil | Cytochrome P450 3A4 | enzyme |
Belumosudil | Cytochrome P450 2C8 | enzyme |
Belumosudil | Cytochrome P450 2D6 | enzyme |
Belumosudil | UDP-glucuronosyltransferase 1-9 | enzyme |
Belumosudil | Cytochrome P450 1A2 | enzyme |
Belumosudil | Cytochrome P450 2C19 | enzyme |
Belumosudil | UDP-glucuronosyltransferase 1-1 | enzyme |
Belumosudil | P-glycoprotein 1 | transporter |
Belumosudil | ATP-binding cassette sub-family G member 2 | transporter |
Belumosudil | Solute carrier organic anion transporter family member 1B1 | transporter |
Lorlatinib | ALK tyrosine kinase receptor | target |
Lorlatinib | Cytochrome P450 3A Subfamily | enzyme |
Lorlatinib | Cytochrome P450 3A5 | enzyme |
Lorlatinib | Cytochrome P450 2B6 | enzyme |
Lorlatinib | Cytochrome P450 2C8 | enzyme |
Lorlatinib | Cytochrome P450 2C19 | enzyme |
Lorlatinib | UDP-glucuronosyltransferase 1-3 | enzyme |
Lorlatinib | Cytochrome P450 3A4 | enzyme |
Mobocertinib | Epidermal growth factor receptor | target |
Mobocertinib | Cytochrome P450 3A4 | enzyme |
Mobocertinib | Cytochrome P450 3A5 | enzyme |
Mobocertinib | Cytochrome P450 3A7 | enzyme |
Mobocertinib | P-glycoprotein 1 | transporter |
Mobocertinib | ATP-binding cassette sub-family G member 2 | transporter |
Asciminib | Cytochrome P450 3A4 | enzyme |
Asciminib | UDP-glucuronosyltransferase 2B7 | enzyme |
Asciminib | UDP-glucuronosyltransferase 2B17 | enzyme |
Asciminib | Tyrosine-protein kinase ABL1 | target |
Asciminib | ATP-binding cassette sub-family G member 2 | transporter |
Asciminib | UDP-glucuronosyltransferase 1-1 | enzyme |
Asciminib | Cytochrome P450 2C19 | enzyme |
Asciminib | P-glycoprotein 1 | transporter |
Asciminib | Solute carrier organic anion transporter family member 1B1 | transporter |
Asciminib | Solute carrier organic anion transporter family member 1B3 | transporter |
Asciminib | Solute carrier family 22 member 1 | transporter |
Asciminib | Cytochrome P450 2C9 | enzyme |
Maribavir | Serine/threonine protein kinase UL97 | target |
Maribavir | Cytochrome P450 3A4 | enzyme |
Maribavir | Cytochrome P450 1A2 | enzyme |
Maribavir | Serum albumin | carrier |
Maribavir | Alpha-1-acid glycoprotein 1 | carrier |
Maribavir | ATP-binding cassette sub-family G member 2 | transporter |
Maribavir | P-glycoprotein 1 | transporter |
Sotagliflozin | UDP-glucuronosyltransferase 1-9 | enzyme |
Sotagliflozin | UDP-glucuronosyltransferase 1-1 | enzyme |
Sotagliflozin | UDP-glucuronosyltransferase 2B7 | enzyme |
Sotagliflozin | Cytochrome P450 3A4 | enzyme |
Sotagliflozin | Sodium/glucose cotransporter 2 | target |
Sotagliflozin | Sodium/glucose cotransporter 1 | target |
Sotagliflozin | Cytochrome P450 2D6 | enzyme |
Sotagliflozin | P-glycoprotein 1 | transporter |
Sotagliflozin | ATP-binding cassette sub-family G member 2 | transporter |
Sotagliflozin | Solute carrier organic anion transporter family member 1B1 | transporter |
Sotagliflozin | Solute carrier organic anion transporter family member 1B3 | transporter |
Sotagliflozin | Canalicular multispecific organic anion transporter 1 | transporter |
Roxadustat | Egl nine homolog 1 | target |
Roxadustat | Egl nine homolog 2 | target |
Roxadustat | Egl nine homolog 3 | target |
Roxadustat | Cytochrome P450 2C8 | enzyme |
Roxadustat | ATP-binding cassette sub-family G member 2 | transporter |
Roxadustat | Solute carrier organic anion transporter family member 1B1 | transporter |
Roxadustat | Serum albumin | carrier |
Roxadustat | UDP-glucuronosyltransferase 1-9 | enzyme |
Roxadustat | Solute carrier family 22 member 6 | transporter |
Roxadustat | Solute carrier family 22 member 8 | transporter |
Cannabinol | Cytochrome P450 3A4 | enzyme |
Cannabinol | Cytochrome P450 2C19 | enzyme |
Cannabinol | Cytochrome P450 1A1 | enzyme |
Cannabinol | Cytochrome P450 1A2 | enzyme |
Cannabinol | Cytochrome P450 1B1 | enzyme |
Cannabinol | Cytochrome P450 2A6 | enzyme |
Cannabinol | Cytochrome P450 2B6 | enzyme |
Cannabinol | Cytochrome P450 2C9 | enzyme |
Cannabinol | Cytochrome P450 2D6 | enzyme |
Cannabinol | Cytochrome P450 3A5 | enzyme |
Cannabinol | Cytochrome P450 3A7 | enzyme |
Cannabinol | UDP-glucuronosyltransferase 1-7 | enzyme |
Cannabinol | UDP-glucuronosyltransferase 1-8 | enzyme |
Cannabinol | UDP-glucuronosyltransferase 1-9 | enzyme |
Cannabinol | UDP-glucuronosyltransferase 1-10 | enzyme |
Cannabinol | UDP-glucuronosyltransferase 2B7 | enzyme |
Cannabinol | P-glycoprotein 1 | transporter |
Cannabinol | ATP-binding cassette sub-family G member 2 | transporter |
Cannabinol | Multidrug resistance-associated protein 1 | transporter |
Cannabinol | Cytochrome P450 2E1 | enzyme |
Cannabinol | Cytochrome P450 2J2 | enzyme |
Cannabinol | Liver carboxylesterase 1 | enzyme |
Pacritinib | Cytochrome P450 3A4 | enzyme |
Pacritinib | Cytochrome P450 1A2 | enzyme |
Pacritinib | Tyrosine-protein kinase JAK2 | target |
Pacritinib | Receptor-type tyrosine-protein kinase FLT3 | target |
Pacritinib | P-glycoprotein 1 | transporter |
Pacritinib | ATP-binding cassette sub-family G member 2 | transporter |
Pacritinib | Solute carrier family 22 member 1 | transporter |
Pacritinib | Cytochrome P450 2C19 | enzyme |
Pacritinib | Solute carrier family 22 member 2 | transporter |
Oteseconazole | Cytochrome P450 51 | target |
Oteseconazole | ATP-binding cassette sub-family G member 2 | transporter |