| GSK-256066 | Organic compounds | Organoheterocyclic compounds | Quinolines and derivatives | Quinoline carboxamides | Details |
| PF-03715455 | Organic compounds | Organoheterocyclic compounds | Azoles | Pyrazoles | Details |
| Alisporivir | Organic compounds | Organic acids and derivatives | Peptidomimetics | Peptoid-peptide hybrids | Details |
| Dilmapimod | Organic compounds | Organoheterocyclic compounds | Diazines | Pyrimidines and pyrimidine derivatives | Details |
| Gilteritinib | Organic compounds | Organoheterocyclic compounds | Piperidines | Phenylpiperidines | Details |
| Duligotuzumab | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Rezatomidine | Organic compounds | Benzenoids | Benzene and substituted derivatives | Xylenes | Details |
| BMS-275183 | Organic compounds | Lipids and lipid-like molecules | Prenol lipids | Diterpenoids | Details |
| AZD-0328 | Organic compounds | Organoheterocyclic compounds | Quinuclidines | Not Available | Details |
| Rigosertib | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| Erdafitinib | Organic compounds | Organic nitrogen compounds | Organonitrogen compounds | Amines | Details |
| Menatetrenone | Organic compounds | Lipids and lipid-like molecules | Prenol lipids | Quinone and hydroquinone lipids | Details |
| S-3304 | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| Pelubiprofen | Organic compounds | Phenylpropanoids and polyketides | Phenylpropanoic acids | Not Available | Details |
| Brincidofovir | Organic compounds | Organoheterocyclic compounds | Diazines | Pyrimidines and pyrimidine derivatives | Details |
| Simtuzumab | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Citicoline | Organic compounds | Nucleosides, nucleotides, and analogues | Pyrimidine nucleotides | Pyrimidine ribonucleotides | Details |
| Itacitinib | Organic compounds | Organoheterocyclic compounds | Pyridines and derivatives | Pyridinecarboxylic acids and derivatives | Details |
| Napabucasin | Organic compounds | Organoheterocyclic compounds | Naphthofurans | Not Available | Details |
| Cordycepin | Organic compounds | Nucleosides, nucleotides, and analogues | Purine nucleosides | Purine 3'-deoxyribonucleosides | Details |
| Fasinumab | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Filorexant | Organic compounds | Benzenoids | Benzene and substituted derivatives | Benzoyl derivatives | Details |
| Dupilumab | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Bucillamine | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| Deutetrabenazine | Organic compounds | Organoheterocyclic compounds | Tetrahydroisoquinolines | Not Available | Details |
| HX-1171 | Organic compounds | Benzenoids | Phenols | 4-alkoxyphenols | Details |
| Sarpogrelate | Organic compounds | Phenylpropanoids and polyketides | Stilbenes | Not Available | Details |
| Presatovir | Organic compounds | Benzenoids | Benzene and substituted derivatives | Benzoyl derivatives | Details |
| LY-3023414 | Organic compounds | Organoheterocyclic compounds | Quinolines and derivatives | Imidazoquinolines | Details |
| MK-0557 | Organic compounds | Organoheterocyclic compounds | Azoles | Pyrazoles | Details |