| GLPG-0187 | Organic compounds | Organoheterocyclic compounds | Diazanaphthalenes | Naphthyridines | Details |
| 5-Hydroxymethylfurfural | Organic compounds | Organic oxygen compounds | Organooxygen compounds | Carbonyl compounds | Details |
| Bavisant | Organic compounds | Benzenoids | Benzene and substituted derivatives | Benzoic acids and derivatives | Details |
| P-nitrobiphenyl | Organic compounds | Benzenoids | Benzene and substituted derivatives | Biphenyls and derivatives | Details |
| Doravirine | Organic compounds | Organic oxygen compounds | Organooxygen compounds | Ethers | Details |
| CP-724714 | Organic compounds | Organoheterocyclic compounds | Diazanaphthalenes | Benzodiazines | Details |
| Motolimod | Organic compounds | Organoheterocyclic compounds | Benzazepines | Not Available | Details |
| Entolimod | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| Dasotraline | Organic compounds | Benzenoids | Tetralins | Not Available | Details |
| Cipargamin | Organic compounds | Alkaloids and derivatives | Harmala alkaloids | Not Available | Details |
| Foretinib | Organic compounds | Organic oxygen compounds | Organooxygen compounds | Ethers | Details |
| Eltanolone | Organic compounds | Lipids and lipid-like molecules | Steroids and steroid derivatives | Pregnane steroids | Details |
| GI-181771X | Organic compounds | Organoheterocyclic compounds | Benzodiazepines | Not Available | Details |
| Trehalose | Organic compounds | Organic oxygen compounds | Organooxygen compounds | Carbohydrates and carbohydrate conjugates | Details |
| CP1-1189 | Organic compounds | Benzenoids | Benzene and substituted derivatives | Benzoic acids and derivatives | Details |
| ORG-25435 | Organic compounds | Organic acids and derivatives | Carboxylic acids and derivatives | Amino acids, peptides, and analogues | Details |
| Dopexamine | Organic compounds | Benzenoids | Phenols | Benzenediols | Details |
| Chlorproguanil | Organic compounds | Benzenoids | Benzene and substituted derivatives | Halobenzenes | Details |
| 9CUAB30 | Organic compounds | Benzenoids | Tetralins | Not Available | Details |
| Vanucizumab | Organic Compounds | Organic Acids | Carboxylic Acids and Derivatives | Amino Acids, Peptides, and Analogues | Details |
| BMS-599626 | Organic compounds | Organoheterocyclic compounds | Benzopyrazoles | Indazoles | Details |
| Benzbromarone | Organic compounds | Organic oxygen compounds | Organooxygen compounds | Carbonyl compounds | Details |
| Ifetroban | Organic compounds | Phenylpropanoids and polyketides | Phenylpropanoic acids | Not Available | Details |
| GW-870086 | Organic compounds | Lipids and lipid-like molecules | Steroids and steroid derivatives | Steroid esters | Details |
| Radotinib | Organic compounds | Benzenoids | Benzene and substituted derivatives | Anilides | Details |
| Idasanutlin | Organic compounds | Phenylpropanoids and polyketides | Stilbenes | Not Available | Details |
| Antroquinonol | Organic compounds | Lipids and lipid-like molecules | Prenol lipids | Diterpenoids | Details |
| Salvinorin A | Organic compounds | Lipids and lipid-like molecules | Prenol lipids | Terpene lactones | Details |
| Cantharidin | Organic compounds | Organoheterocyclic compounds | Furofurans | Not Available | Details |
| Eravacycline | Organic compounds | Phenylpropanoids and polyketides | Tetracyclines | Not Available | Details |