Benzbromarone

DB12319ApprovedWithdrawnSmall molecule

Benzbromarone is a uricosuric agent which is taken daily for the prevention of gout flares. Benzbromarone has been used in trials studying the basic science and treatment of Heart Failure, Hyperuricemia, Chronic Kidney Disease, Abnormal Renal Function, and Gout and Asymptomatic Hyperuricemia.

Chemical structure of Benzbromarone
Mechanism
Curator reviewed
Formula / weight
C17H12Br2O3 · 424.083 g/mol (avg)
Code names
L-2214 · MJ 10061

Resolves to

Compound
UNII4POG0RL69OCAS3562-84-3ChEMBLCHEMBL388590ChEBI3023PubChem2333KEGGD01056
Clinical / RWD
RxNorm1385ATCM04AB03
Structure
InChIKeyWHQCHUCQKNIQEC-UHFFFAOYSA-NSMILESCCC1=C(C(=O)C2=CC(Br)=C(O)C(Br)=C2)C2=CC=CC=C2O1
Targets
Q96S37SLC22A12Q5XXA6ANO1P33527ABCC1P11712CYP2C9P33261CYP2C19
Transporters
Q9Y6L6SLCO1B1O94956SLCO2B1O95342ABCB11

What you can answer from here — as of June 15, 2026

5Protein targetsEach mapped to UniProt, with action and pharmacological action
Listed above
3TransportersSubstrate / inhibitor direction, not just membership
Listed above
789Drug interactionsStructured to mechanism, not free text
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10Clinical trialsPhase, status and sponsor resolved per trial
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2Structured indicationsCondition, population, route and combination as fields, not prose
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4Marketed productsAcross 3 countries and 3 labellers
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1ATC codeIncluding every combination product, plus 17 drug categories
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29+ReferencesStructured and connected to the statements they support
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