LNS-8801

DB18091InvestigationalSmall molecule

LNS-8801: Overview.

Mechanism: Pharmacologically active on G protein-coupled estrogen receptor 1
Curator reviewed
Formula / weight: C₂₁H₁₈BrNO₃ · 412.283 g/mol (avg)
Also known as: Ethanone, 1-((3ar,4s,9bs)-4-(6-bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-3h-cyclopenta(c)quinolin-8-yl)-, rel- · G 1 (anti-tumor agent) · G 1 (g protein-coupled estrogen receptor agonist) · G 1 (gper agonist)
Code names: LNS-8801

Resolves to

Compound

Structure

InChIKeyVHSVKVWHYFBIFJ-HKZYLEAXSA-NSMILES[H][C@]12CC=C[C@@]1([H])C1=CC(=CC=C1N[C@H]2C1=CC2=C(OCO2)C=C1Br)C(C)=O

Targets

What you can answer from here — as of April 23, 2025

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

2Clinical trialsPhase, status and sponsor resolved per trial

1+ReferenceStructured and connected to the statements they support

Which drugs share a target with LNS-8801, and which of those have an active Phase 3 trial?

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