Search
ABT-737
go.drugbank.com/drugs/DB17023ExperimentalAn inhibitor of members of the Bcl‑2 family of apoptosis regulators.[A252977]
Categories: Proto-Oncogene Proteins c-bcl-2, Heterocyclic Compounds, 1-RingSynonyms: Benzamide, 4-(4-((4'-chloro(1,1'-biphenyl)-2-yl)methyl)-1-piperazinyl)-n-((4-(((1r)-3-(dimethylamino)-1-((phenylthio)methyl)propyl)amino)-3-nitrophenyl)sulfonyl)-Go-6976
go.drugbank.com/drugs/DB17029ExperimentalAn inhibitor of calcium-dependent isoforms of protein kinase C.[A253002,A253007]
Categories: Heterocyclic Compounds, 2-Ring, Heterocyclic Compounds, 3-RingSynonyms: 12h-indolo(2,3-a)pyrrolo(3,4-c)carbazole-12-propanenitrile, 5,6,7,13-tetrahydro-13-methyl-5-oxo-JTC-801 free base
go.drugbank.com/drugs/DB17033ExperimentalAn antagonist of nociceptin receptor and analgesic agent, evaluated for its use in cancer treatment.
Synonyms: Benzamide, n-(4-amino-2-methyl-6-quinolinyl)-2-((4-ethylphenoxy)methyl)-Categories: Heterocyclic Compounds, 2-RingN-oleoyldopamine
go.drugbank.com/drugs/DB17036ExperimentalN-oleoyldopamine (OLDA) is an amide of dopamine and oleic acid.[A253042]
Synonyms: (9z)- n-(2-(3,4-dihydroxyphenyl)ethyl)-9-octadecenamide, N-oleoyldopamineNSC-663284
go.drugbank.com/drugs/DB17038ExperimentalNSC-663284 is a potent quinolinedione Cdc25 phosphatase inhibitor.[A253052]
Categories: Heterocyclic Compounds, 2-RingSynonyms: 5,8-quinolinedione, 6-chloro-7-((2-(4-morpholinyl)ethyl)amino)-, 6-chloro-7-((2-morpholinoethyl)amino)quinoline-5,8-dionePhorbol 12-myristate 13-acetate diester
go.drugbank.com/drugs/DB17045InvestigationalPhorbol 12-myristate 13-acetate diester is an inducer of neutrophil extracellular traps (NETs).[A253087]
Synonyms: 12-o-tetradecanoylphorbol-13-acetatePI-103
go.drugbank.com/drugs/DB17046ExperimentalPI-103 is an inhibitor of p110α of class I PI3K.[A253092]
Categories: Heterocyclic Compounds, 1-RingSynonyms: Phenol, 3-(4-(4-morpholinyl)pyrido(3',2':4,5)furo(3,2-d)pyrimidin-2-yl)-PIK-75
go.drugbank.com/drugs/DB17047ExperimentalPIK-75 is a preferential p110 alpha/gamma PI3K inhibitor.[A253097]
Categories: Phosphatidylinositol 3-Kinases, antagonists & inhibitorsSynonyms: Benzenesulfonic acid, 2-methyl-5-nitro-, 2-((6-bromoimidazo(1,2-a)pyridin-3-yl)methylene)-1-methylhydrazidePlumbagin
go.drugbank.com/drugs/DB17048InvestigationalPlumbagin is a compound investigated for its anticancer activity. It has been found that it inactivates the Akt/NF-kB, MMP-9 and VEGF pathways.[A253102]
Categories: Compounds used in a research, industrial, or household settingSynonyms: 5-hydroxy-2-methyl-1,4-naphthalenedioneRS-39604
go.drugbank.com/drugs/DB17050ExperimentalRS-39604 is a selective 5-HT4 receptor antagonist.[A253112]
Salts: RS-39604 hydrochlorideCategories: Heterocyclic Compounds, 1-Ring