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Asiatic acid
go.drugbank.com/drugs/DB14054InvestigationalFrom Centella asiatica and other plants; shows a variety of bioactivities.
Nigericin
go.drugbank.com/drugs/DB14056ExperimentalA polyether antibiotic which affects ion transport and ATPase activity in mitochondria. It is produced by Streptomyces hygroscopicus. (From Merck Index, 11th ed)
Categories: Heterocyclic Compounds, 1-Ring, Compounds used in a research, industrial, or household settingSynonyms: Helixin C, Azalomycin MValinomycin
go.drugbank.com/drugs/DB14057ExperimentalIt is composed of 3 moles each of L-valine, D-alpha-hydroxyisovaleric acid, D-valine, and L-lactic acid linked alternately to form a 36-membered ring. … (From Merck Index, 11th ed) Valinomycin is a potassium selective ionophore and is commonly used as a tool in biochemical studies.
Categories: P-glycoprotein inhibitors, P-glycoprotein substratesSynonyms: Potassium ionophore IBasifungin
go.drugbank.com/drugs/DB14058ExperimentalBasifungin, also known as _aureuobacidin A_, is a phosphorylceramide synthase inhibitor [L2960], [A33381].
Synonyms: Aureobasidin AConcanamycin A
go.drugbank.com/drugs/DB14062ExperimentalConcanamycin A is an H+-ATPase (vacuolar) inhibitor.
Categories: P-glycoprotein inhibitorsSynonyms: Concanamycin ATetrandrine
go.drugbank.com/drugs/DB14066InvestigationalSynonyms: (S,S)-Tetrandrine, D-TetrandrineCategories: P-glycoprotein inhibitors, Cytochrome P-450 SubstratesDofequidar
go.drugbank.com/drugs/DB14067InvestigationalDofequidar is an antineoplastic agent.
Categories: P-glycoprotein inhibitors, Heterocyclic Compounds, 2-RingHM-30181
go.drugbank.com/drugs/DB14070InvestigationalCategories: ATP Binding Cassette Transporter, Subfamily B, Member 1, antagonists & inhibitors, P-glycoprotein inhibitorsDesmethylsertraline
go.drugbank.com/drugs/DB14071ExperimentalDesmethylsertraline is a metabolite of sertraline.
Categories: P-glycoprotein inhibitorsSynonyms: N-Demethylsertraline, N-DesmethylsertralineReversin 121
go.drugbank.com/drugs/DB14072ExperimentalReversin 121 is a hydrophobic peptide chemosensitizer that can reverse P-glycoprotein-mediated multidrug resistance.
Categories: P-glycoprotein inhibitors