| DB00617 | Paramethadione | approved | yes | inhibitor | Details |
| DB04841 | Flunarizine | approved | yes | inhibitor | Details |
| DB01118 | Amiodarone | approved, investigational | unknown | inhibitor | Details |
| DB00909 | Zonisamide | approved, investigational | yes | inhibitor | Details |
| DB00568 | Cinnarizine | approved, investigational | yes | inhibitor | Details |
| DB01388 | Mibefradil | investigational, withdrawn | yes | inhibitor | Details |
| DB09498 | Strontium chloride Sr-89 | approved, investigational | no | inducer | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | | Details |
| DB09235 | Efonidipine | experimental | unknown | antagonist | Details |
| DB06152 | Nylidrin | approved | unknown | antagonistagonist | Details |
| DB14011 | Nabiximols | investigational | unknown | | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | | Details |
| DB00381 | Amlodipine | approved | yes | inhibitor | Details |
| DB06712 | Nilvadipine | approved, investigational | unknown | inhibitor | Details |
| DB09238 | Manidipine | approved, investigational | unknown | inhibitor | Details |
| DB00622 | Nicardipine | approved, investigational | unknown | inhibitor | Details |