| DB00030 | Insulin human | approved, investigational | yes | agonist | Details |
| DB00047 | Insulin glargine | approved | yes | agonist | Details |
| DB00071 | Insulin pork | approved | yes | binder | Details |
| DB03909 | Adenosine-5'-[Beta, Gamma-Methylene]Triphosphate | experimental | unknown | | Details |
| DB05120 | AT1391 | investigational | unknown | | Details |
| DB05115 | NN344 | investigational | unknown | | Details |
| DB01307 | Insulin detemir | approved | yes | agonist | Details |
| DB00046 | Insulin lispro | approved | yes | agonist | Details |
| DB01306 | Insulin aspart | approved | yes | agonist | Details |
| DB01309 | Insulin glulisine | approved | yes | agonist | Details |
| DB01277 | Mecasermin | approved, investigational | unknown | | Details |
| DB08513 | [4-({5-(AMINOCARBONYL)-4-[(3-METHYLPHENYL)AMINO]PYRIMIDIN-2-YL}AMINO)PHENYL]ACETIC ACID | experimental | unknown | | Details |
| DB09564 | Insulin degludec | approved | yes | agonist | Details |
| DB09129 | Chromic chloride | approved | yes | activator | Details |
| DB12267 | Brigatinib | approved, investigational | no | binding | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | inhibitor | Details |
| DB14751 | Mecasermin rinfabate | approved | unknown | | Details |
| DB16637 | KW-2450 free base | experimental | unknown | inhibitor | Details |
| DB15399 | BMS-754807 | investigational | unknown | inhibitor | Details |
| DB06075 | Linsitinib | investigational | unknown | inhibitor | Details |
| DB11567 | Insulin peglispro | investigational | unknown | | Details |
| DB11564 | Insulin argine | experimental | yes | agonist | Details |
| DB09456 | Insulin beef | approved | yes | agonist | Details |
| DB11568 | Insulin tregopil | investigational | yes | agonist | Details |