| DB00007 | Leuprolide | approved, investigational | yes | agonist | Details |
| DB00106 | Abarelix | approved, investigational, withdrawn | yes | antagonist | Details |
| DB00644 | Gonadorelin | approved, investigational, vet_approved | yes | agonist | Details |
| DB00666 | Nafarelin | approved | yes | agonist | Details |
| DB00050 | Cetrorelix | approved, investigational | yes | antagonist | Details |
| DB01406 | Danazol | approved | yes | negative modulator | Details |
| DB11979 | Elagolix | approved, investigational | unknown | antagonist | Details |
| DB06494 | Sufugolix | investigational | unknown | | Details |
| DB06699 | Degarelix | approved | yes | antagonist | Details |
| DB00014 | Goserelin | approved | yes | agonist | Details |
| DB06719 | Buserelin | approved, investigational | yes | | Details |
| DB06825 | Triptorelin | approved, vet_approved | yes | agonist | Details |
| DB06785 | Ganirelix | approved | yes | antagonist | Details |
| DB06788 | Histrelin | approved, withdrawn | yes | agonist | Details |
| DB11619 | Gestrinone | approved | unknown | antagonist | Details |
| DB05624 | Teverelix | investigational | yes | antagonist | Details |
| DB11853 | Relugolix | approved, investigational | yes | antagonist | Details |
| DB17083 | Linzagolix | approved | yes | antagonist | Details |